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8-{2-[methyl(phenyl)amino]acetyl}-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
N,5-dimethyl-4-{[(6-methylpyridin-2-yl)methyl]amino}-N-(propan-2-yl)thieno[2,3-d]pyrimidine-6-carboxamide
4-{[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}-1-phenyl-1H-1,2,3-triazole
1-{3-fluoro-5-methylimidazo[1,2-a]pyridine-2-carbonyl}-2-(3-methoxypropyl)piperidine
(4aS,7aR)-1-(3,3-dimethylbutanoyl)-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-amino-4-(5-chloro-2,3-dimethoxyphenyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
3-phenyl-2-{2-[1-(propan-2-yl)piperidin-4-yl]-1H-imidazol-1-yl}propanoic acid
N-[4-(propan-2-yloxy)-1-(2,2,2-trifluoroethyl)-1H-indazol-3-yl]oxolane-3-carboxamide
N-[(3R,4S)-1-[2-(benzyloxy)acetyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
N-cyclopropyl-1-[1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidin-4-yl]piperidine-4-carboxamide
(2S,4R)-4-amino-1-[2-(2,5-dimethylphenyl)acetyl]-N-ethylpyrrolidine-2-carboxamide
6-{1-[(1,2-dimethyl-1H-imidazol-4-yl)sulfonyl]piperidin-3-yl}-2-methyl-3,4-dihydropyrimidin-4-one
2-methyl-6-{[6-(propan-2-yl)pyrimidin-4-yl]amino}heptan-2-ol
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
3-(4-chlorophenyl)-1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperidine
N-{[1-({4-oxo-3H,4H-thieno[3,2-d]pyrimidin-2-yl}methyl)-1,2,5,6-tetrahydropyridin-3-yl]methyl}acetamide
N2-[(1-benzyl-1H-imidazol-2-yl)methyl]-N4-methylpyrimidine-2,4-diamine
2-{3-oxo-9-[(2S)-oxolane-2-carbonyl]-2,9-diazaspiro[5.5]undecan-2-yl}acetic acid
N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-2-(3,5-dimethyl-1H-pyrazol-1-yl)acetamide
{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
N-(1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-1H-indole-2-carboxamide
3-[1-(4-propylpyrimidine-5-carbonyl)piperidin-4-yl]phenol
7-methyl-2-{2-[5-(oxolan-3-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}-1H-1,3-benzodiazole
1-(2-chloro-4-fluoro-5-methylphenyl)-3-ethyl-3-[2-(1H-pyrazol-1-yl)ethyl]urea
4-[1-(3-methylphenyl)-1H-pyrazol-4-yl]-2-[2-(pyridin-2-yl)pyrrolidin-1-yl]pyrimidine
2-{[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl](propan-2-yl)amino}-2-(4-fluoro-3-methylphenyl)acetic acid
N-[(3S,4R)-1-({2-methyl-5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-7-yl}methyl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
(3E)-5,5-dimethyl-2-[4-(pyrazin-2-yl)piperazin-1-yl]hex-3-enoic acid
(3S,4R)-1-{3-[(2R,6S)-2,6-dimethylmorpholin-4-yl]propanoyl}-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
1-[(2,6-dimethoxyphenyl)methyl]-5-oxopyrrolidine-3-carboxylic acid
3-[(propan-2-yl)(quinolin-4-ylmethyl)amino]propanamide
1-(3-chlorophenyl)-4-{[4-(2-hydroxyethoxy)phenyl]methyl}-5-methylpiperazin-2-one
3-(2-{4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-oxoethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-{[(furan-2-ylmethyl)[2-(morpholin-4-yl)ethyl]amino]methyl}phenol
2-[(5-methylpyrazin-2-yl)methyl]-8-(thiophene-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
(1R,7S)-3-(2-methoxyethyl)-N-methyl-4-oxo-N-[2-(1H-pyrazol-1-yl)ethyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-1-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
2-(methylamino)-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}-1,3-thiazole-4-carboxamide
2-(4-{1-[3-(1H-pyrazol-1-yl)propyl]pyrrolidin-3-yl}piperidin-1-yl)pyrimidine
N2-({2-[(dimethylamino)methyl]phenyl}methyl)-N4,N4,5-trimethylpyrimidine-2,4-diamine
2-[(2-methanesulfonamidoethyl)amino]-N-(1,3-thiazol-2-yl)propanamide
N-{4-[2-(4-butylpiperazin-1-yl)-2-oxoethoxy]phenyl}propanamide
2-[(4-chlorophenyl)methyl]-8-(propan-2-yl)-2,8-diazaspiro[4.5]decan-3-one
(2,1,3-benzoxadiazol-4-ylmethyl)(ethyl)[2-(1H-pyrazol-1-yl)ethyl]amine
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2-{2-[(4-phenylpiperazin-1-yl)methyl]-4-(thiophen-3-yl)phenoxy}acetamide
2-(cyclohex-1-en-1-yl)-N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]acetamide
3-(1-{6-amino-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-4-yl)-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-1-(4-methylphenyl)piperazin-2-one
3-{[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]sulfonyl}benzoic acid