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1-{1-[2-(4-chlorophenyl)acetyl]piperidin-3-yl}-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
3-{[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]sulfonyl}benzoic acid
5-(2-{3-[ethyl(pyridin-4-ylmethyl)amino]piperidin-1-yl}-2-oxoethyl)-2-methyl-3,4-dihydropyrimidin-4-one
N,N-dimethyl-4-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]piperidine-1-carboxamide
4-(3-hydroxy-3-methylbutyl)-N-{[1-(hydroxymethyl)cyclopropyl]methyl}-N-methylbenzamide
N-{2-[ethyl(3-methylphenyl)amino]ethyl}-1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2,2-dimethyl-1-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}propan-1-one
2-(3-methylpyridine-2-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
(3aR,7aS)-N-[5-(5-ethyl-1,3,4-oxadiazol-2-yl)-2-methoxyphenyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-(3-methoxypropyl)pyrrolidin-3-yl]-5-fluoro-2-methoxybenzamide
N-[(4-phenyloxan-4-yl)methyl]-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(2,5-dioxoimidazolidin-1-yl)-N-ethyl-N-(pyridin-4-ylmethyl)acetamide
[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl][(2-fluoro-4-methoxyphenyl)methyl]methylamine
2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]-N-(3-phenylprop-2-yn-1-yl)-N-propylacetamide
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2,2,3,3-tetramethylcyclopropane-1-carboxamide
4-(3-fluorophenoxy)-1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidine
N-(2-{1-[(2-methylnaphthalen-1-yl)methyl]piperidin-3-yl}ethyl)acetamide
1-methyl-6-oxo-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]-1,6-dihydropyridazine-3-carboxamide
4-methoxy-2-({methyl[(5-{[(2-methylphenyl)methyl]sulfanyl}-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl)methyl]amino}methyl)phenol
1-methyl-4-({1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidin-3-yl}methyl)piperazine
9-[(2R)-2-cyclohexyl-2-hydroxyacetyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
(butan-2-yl)(pyridin-4-ylmethyl)(quinolin-4-ylmethyl)amine
3-butyl-4-ethyl-1-(2-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-2-oxoethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
7-fluoro-3-({4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}methyl)-1,2-dihydroquinolin-2-one
7-ethoxy-4-(6-methoxypyridin-3-yl)-1,2,3,4-tetrahydroquinolin-2-one
2-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]pyridine-4-carbonitrile
(1R,5R)-6-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
2-methyl-4-(4-{[methyl(oxan-4-yl)amino]methyl}phenyl)butan-2-ol
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-{2-[(3-methylpyridin-2-yl)amino]ethyl}acetamide
2-(5-acetylthiophen-3-yl)-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]acetamide
N-[3-(1H-imidazol-1-yl)propyl]-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propanamide
4-(1-{1-[(6-methoxypyridin-3-yl)methyl]piperidin-4-yl}ethyl)morpholine
9-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
methyl 3-(3-{2-cyano-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}propanamido)thiophene-2-carboxylate
4-{[2-(oxolan-3-yl)-1H-imidazol-1-yl]methyl}-2-phenyl-2H-1,2,3-triazole
1-(cyclohexylmethyl)-5-[(cyclopropylmethyl)amino]-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(2R,3S,6R)-5-[(2-ethylpyrimidin-5-yl)methyl]-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-amino-1-{5-[5-(3,5-dimethyl-1H-pyrrol-2-yl)-1,2,4-oxadiazol-3-yl]-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl}ethan-1-one
5-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidine-1-carbonyl]-2-(thiophen-2-yl)pyrimidin-4-ol
2-(4-{[(1R,5R)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}phenyl)ethan-1-amine
2-methyl-8-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
[1-({1-[3-(methylsulfanyl)butyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]methanol
2-hydroxy-N-methyl-N-[2-(morpholin-4-yl)propyl]-5-(1H-pyrrol-1-yl)benzamide
3-{[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl](methyl)amino}-1-(3-methylpiperidin-1-yl)propan-1-one
8-({3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}methyl)quinoline
[(1-cyclopentylpiperidin-4-yl)methyl][(3-methyl-1,2-oxazol-5-yl)methyl](oxolan-2-ylmethyl)amine
1-(2-phenoxyethyl)-5-[4-(thiophen-2-ylmethyl)piperazin-1-yl]azepan-2-one
N-[1-(dimethyl-1,3-thiazol-2-yl)propyl]-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
N-[2-(2-methoxynaphthalen-1-yl)ethyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
dimethyl[(4-methyl-5-{1-[3-(pyrrolidin-1-yl)pyrazin-2-yl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]amine