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1-(cyclopropylmethyl)-5-[2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
8-(2,4-difluorobenzenesulfonyl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-2-methyl-4-(2-methylphenyl)piperazine
8-cyclopropyl-N-(2-ethoxyphenyl)-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
3-[(3S,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[2-(trifluoromethyl)phenyl]urea
2,3,6-trimethyl-4-[3-(pyridin-2-yl)azetidine-1-carbonyl]quinoline
1-ethyl-N-methyl-2-oxo-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1,2-dihydropyridine-4-carboxamide
5-[(2-chloro-4,5-difluorophenyl)methyl]-1-methyl-1H-1,2,4-triazole
N-[(3-tert-butyl-1,2,4-oxadiazol-5-yl)methyl]-5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-amine
1-cyclopentyl-5-(2,3-dimethoxyphenyl)-3-methyl-1H,4H-pyrazolo[3,4-d]imidazole
8-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-1-(2-methylpropyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-amino-4-chloro-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-1H-pyrazole-3-carboxamide
1-(3-{[3-(3-hydroxyazetidine-1-carbonyl)-1,2-oxazol-5-yl]methoxy}phenyl)ethan-1-one
2-(2,5-dimethoxyphenyl)-8-methyl-3-(morpholin-4-ylmethyl)quinoline
1-[1-(3-phenylpropyl)piperidin-4-yl]-4-(piperidine-1-carbonyl)piperidine
2-methyl-N-({4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenyl}methyl)propanamide
1-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3-methylbutan-1-one
(1S,5R)-3-(2H-1,3-benzodioxol-5-ylmethyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonane
2-({[2-(ethanesulfonyl)ethyl]amino}methyl)-6,8-dimethylquinolin-4-ol
2-{4-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]-1-(furan-3-ylmethyl)piperazin-2-yl}ethan-1-ol
4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}-N-[(1S)-1-phenylethyl]piperidine-1-carboxamide
N-ethyl-2-[(1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonan-3-yl]-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
N-[(1-ethyl-1H-indazol-3-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
3-({[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl](methyl)amino}methyl)-6-methoxy-1,2-dihydroquinolin-2-one
1-{2-[1-(2,4-difluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]ethyl}-1,2-dihydropyridin-2-one
1-(4-methyl-1,3-oxazole-5-carbonyl)-3-(4-phenylbenzoyl)piperidine
3-fluoro-N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]pyridine-4-carboxamide
N-phenyl-2-[(1R,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
6-(1-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}piperidin-3-yl)-3,4-dihydropyrimidin-4-one
methyl 6-[(2-methylpiperidin-1-yl)methyl]-3-(thiophene-3-amido)thieno[2,3-b]pyridine-2-carboxylate
2-(1-{4-[(pyridin-2-ylsulfanyl)methyl]benzoyl}piperidin-2-yl)ethan-1-ol
3-(1-methyl-1H-imidazol-4-yl)-5-[3-(2-methylpropyl)-1H-pyrazol-5-yl]-1,2,4-oxadiazole
1-{4-[({2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}amino)methyl]phenoxy}-3-(piperidin-1-yl)propan-2-ol
4-(8-methoxyquinolin-5-yl)-N,6-dimethylpyrimidin-2-amine
2-methoxy-4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]phenol
3-(1-cyclopentyl-1H-pyrazol-5-yl)-1-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)urea
4-butyl-N-{4-[(2-methoxyethyl)carbamoyl]-2-methylphenyl}piperazine-1-carboxamide
2-(phenoxymethyl)-5-[(1S,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl]pyrimidin-4-ol
2-({4-phenyl-5-[4-(1H-1,2,4-triazol-1-yl)phenyl]-1H-imidazol-1-yl}methyl)pyridine
1-{[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-4-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]piperazine
N-[3-(1H-imidazol-1-yl)propyl]-3-(morpholine-4-carbonyl)benzene-1-sulfonamide
4-[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]piperazin-2-one
8-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}-1-oxa-8-azaspiro[4.5]decane
3-(1-ethyl-1H-1,2,3-triazol-4-yl)-1-[(1-methanesulfonylpiperidin-3-yl)methyl]urea
2-(3-chloro-4-hydroxyphenyl)-N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]acetamide
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carboxamide
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-2-ethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-(2-methoxyethyl)-3-{methyl[2-(methylsulfanyl)ethyl]sulfamoyl}benzamide
6-[4-(furan-2-carbonyl)piperazine-1-carbonyl]-5-methyl-N-(2-phenylethyl)thieno[2,3-d]pyrimidin-4-amine
[4-({2-[2-(propan-2-yl)pyrimidin-4-yl]-1H-imidazol-1-yl}methyl)oxan-4-yl]methanol