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1-(isoquinolin-5-yl)-3-methyl-3-[3-(oxolan-2-yl)propyl]urea
1-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-4-(2-methoxyphenoxy)piperidine
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}pyridine-3-sulfonamide
(4aS,8aR)-1-[3-(methylsulfanyl)propyl]-6-(pyrazin-2-yl)-decahydro-1,6-naphthyridine-4a-carboxylic acid
5-(2-oxo-2-{4-[(2-oxopyrrolidin-1-yl)methyl]piperidin-1-yl}ethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-({1-[(3-hydroxy-4-methoxyphenyl)methyl]pyrrolidin-3-yl}methyl)-3-(propan-2-yl)urea
1-(dimethyl-1,2-oxazole-4-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
N-[1-(2-chlorophenyl)cyclopropyl]-N'-(2-methylphenyl)propanediamide
N-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
3-[methyl(oxan-4-yl)sulfamoyl]-N-(2,2,2-trifluoroethyl)benzamide
1-[(4aS,8aS)-7-cyclobutanecarbonyl-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2-phenylethane-1,2-dione
2-(4,6-dimethyl-1-benzofuran-3-yl)-1-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
3-(1-butyl-3-methyl-1H-pyrazol-5-yl)-1-[(2,6-dimethoxyphenyl)methyl]urea
1'-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
(2S,4R)-1-[(2-fluorophenyl)methyl]-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide
5-methyl-2-(2-methylphenyl)-4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}-1,3-oxazole
2-[1-(3-ethyl-1,2,4-oxadiazol-5-yl)-2-methylbutyl]-2,3-dihydro-1H-isoindol-1-one
N-butyl-2-{N-methyl-1-[1-methyl-2-(morpholin-4-yl)-1H-1,3-benzodiazol-5-yl]formamido}acetamide
4-{[1-(cyclohexylmethyl)piperidin-3-yl]carbamoyl}pyridin-1-ium-1-olate
N-(2-methoxyethyl)-1-(3-methylbutyl)-4-oxo-5-{1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl}-1,4-dihydropyridine-3-carboxamide
[(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-(3-methoxyphenyl)-4H-1,2,4-triazol-3-yl)methyl](furan-3-ylmethyl)methylamine
2-[4-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-1-(thiophen-3-ylmethyl)piperazin-2-yl]ethan-1-ol
N-[(1,3-diphenyl-1H-pyrazol-4-yl)methyl]-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
4-cyclopentyl-N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]pyrimidin-2-amine
N-cyclopropyl-4-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}piperazine-2-carboxamide
1-{2-[3-(2-methoxyethyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-cyclohexyl-2-[(isoquinolin-5-yloxy)methyl]-1,3-oxazole-4-carboxamide
1-(4-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-3-(pyridin-4-yl)propan-1-one
5-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidine-1-carbonyl}-4,6-dimethyl-2H-pyran-2-one
4-{[4-(3-methyl-3-phenylpiperidine-1-carbonyl)furan-2-yl]methyl}morpholine
5-acetyl-2,4-dimethyl-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1H-pyrrole-3-carboxamide
5,6-dichloro-2-[2,5-dimethyl-1-(4H-1,2,4-triazol-4-yl)-1H-pyrrol-3-yl]-1H-1,3-benzodiazole
2-[(2-chlorophenyl)methyl]-4-{4-[(4-ethoxyphenyl)methyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
[(1-ethyl-1H-imidazol-2-yl)methyl](methyl){[3-(3-methylbutyl)-1,2,4-oxadiazol-5-yl]methyl}amine
5-[6-(hydroxymethyl)-1,4-oxazepane-4-carbonyl]pyridine-2-carbonitrile
1-(1H-1,2,3-benzotriazole-5-carbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
6-fluoro-4-[(1-methylpiperidin-2-yl)methyl]-3,4-dihydro-2H-1,4-benzoxazin-3-one
5-oxo-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)-2,5-dihydro-1H-pyrazole-3-carboxamide
5-methanesulfonyl-1'-[3-(methylsulfanyl)butyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-benzyl-4-(5-fluoro-3-methyl-1H-indole-2-carbonyl)piperazin-2-one
N-(1H-1,3-benzodiazol-2-ylmethyl)-5-[(4-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
3-(2-phenylethyl)-8-(pyrrolidin-3-ylmethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-{4H-thieno[3,2-b]pyrrole-5-carbonyl}-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)-3-methyl-1H-indole-2-carboxamide
N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]pyrazolo[1,5-a]pyridine-2-carboxamide
N-[1-(butan-2-yl)-1H-pyrazol-5-yl]-4-methyl-3-(3-methylbutanamido)benzamide
1-(2,3-dihydro-1H-inden-2-yl)-N-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
methyl 3-(2-amino-6-butanoyl-3-cyano-5,6,7,8-tetrahydro-1,6-naphthyridin-4-yl)benzoate
6-chloro-2-{1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
N5-cyclooctyl-N3-methyl-4-oxo-1-(oxolan-2-ylmethyl)-N3-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide