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2-(4-chloro-2-{[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]methyl}phenoxy)acetamide
(1R,5R)-N-[(4-chlorophenyl)methyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-(8-chloroquinolin-2-yl)-4-hydroxypiperidine-4-carboxylic acid
(3R,5S)-1-benzyl-N3-(2,3-dihydro-1H-inden-5-yl)-N5-[(2-methoxyphenyl)methyl]piperidine-3,5-dicarboxamide
1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-N-[3-(3-methylphenyl)phenyl]piperidine-3-carboxamide
N-[1-(butan-2-yl)-1H-pyrazol-5-yl]-4-[(3-methoxyphenyl)methyl]-3-oxopiperazine-1-carboxamide
3-(2H-1,3-benzodioxol-5-yl)-2-methyl-6-(4H-1,2,4-triazol-4-yl)pyridine
(3R,4S)-1-(2,6-difluoro-3-methoxybenzoyl)-4-(propan-2-yl)pyrrolidin-3-amine
3-(3-chlorobenzoyl)-1-cyclohexylpiperidine
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
ethyl 1-[(2-methyl-1,3-thiazol-5-yl)methyl]-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
(2S,4S,5R)-2-ethyl-5-(4-fluorophenyl)-4-(4-hydroxypiperidine-1-carbonyl)-1-methylpyrrolidine-2-carboxylic acid
(2S)-4-methyl-2-phenyl-1-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]piperazine
N-(1-{[3-(morpholin-4-ylmethyl)phenyl]methyl}piperidin-4-yl)methanesulfonamide
1-[2-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-2-oxoethyl]pyrrolidin-2-one
1-(3-{[6-(2-aminoethyl)-2-methylpyrimidin-4-yl]amino}propyl)pyrrolidin-2-one
1-{[3-(2-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-4-(oxolan-3-yl)-1H-1,2,3-triazole
1-(3-fluoropyridin-4-yl)-4-[3-(furan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
1-(5-chloropyridin-2-yl)-4-[3-(methylsulfanyl)propyl]piperazine
1-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepane
6-(3,5-difluorophenyl)-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
3-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
{[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl}[(8-methoxyquinolin-5-yl)methyl]methylamine
3-(3-methylbut-2-en-1-yl)-1-(2-methylpyrimidin-4-yl)piperidine-3-carboxylic acid
3-phenyl-N-(1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-1,2-oxazole-4-carboxamide
2-{[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1H-imidazole
2-[({5-[1-(5-methoxypyrimidin-2-yl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)(methyl)amino]ethan-1-ol
N-[(3-ethoxyphenyl)methyl]-N-(2-hydroxyethyl)furan-2-carboxamide
2-[3-(4H-1,2,4-triazol-4-yl)benzoyl]-2,3-dihydro-1H-isoindole
2-{5-[3-(3-methoxyphenyl)-1H-pyrazole-5-carbonyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
2,5-dioxo-6-(2-propoxypropyl)-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
6-methyl-2-(2-{[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethyl)-3,4-dihydropyrimidin-4-one
N-[2-oxo-2-(pyrrolidin-1-yl)ethyl]-4-(1H-pyrazol-3-yl)benzamide
4-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-sulfonyl}-2,1,3-benzoxadiazole
1-[(5-methylfuran-2-yl)methyl]-3-[5-(thiophen-2-yl)-1,3,4-thiadiazol-2-yl]urea
1-(3-methyl-3-phenylpiperidin-1-yl)-2-(morpholin-4-yl)ethan-1-one
N-benzyl[(2-methoxypyridin-3-yl)amino]sulfonamide
(1S,5R)-6-(2-methoxyethyl)-3-[1-(pyrazine-2-carbonyl)piperidin-4-yl]-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(3-methoxypropyl)-9-{3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-2,9-diazaspiro[5.5]undecan-3-one
2-(3-methoxyphenoxy)-N-[(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]acetamide
2-{2-[3-(4-chlorophenoxy)phenyl]-1H-imidazol-1-yl}acetamide
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-4-methyl-1H-imidazole-5-carboxamide
[(3-chloro-5-fluoro-4-methoxyphenyl)methyl][(2-fluorophenyl)methyl](2-methoxyethyl)amine
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylpyrimidin-2-amine
1-{4-[3-(4-methoxyphenoxymethyl)piperidine-1-carbonyl]piperidin-1-yl}ethan-1-one
3-[3-(1-cyclopentyl-1H-pyrazol-3-yl)phenyl]-6-methoxypyridazine
1-[(2-fluorophenyl)methyl]-2-methyl-3-[2-oxo-2-(thiomorpholin-4-yl)ethyl]-4,5,6,7-tetrahydro-1H-indol-4-one
(2S,4S)-4-amino-N-ethyl-1-(4,4,4-trifluorobutanoyl)pyrrolidine-2-carboxamide
N-[2-(4-fluoro-2-methoxyphenyl)pyridin-3-yl]-2-methylpropanamide
N-(2-methoxyethyl)-4-methyl-3-{[(piperidin-4-yl)carbamoyl]methyl}-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide