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2-({methyl[3-(1H-pyrazol-1-yl)propyl]amino}methyl)benzoic acid
(3S)-4-{4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzoyl}-1-ethyl-3-methylpiperazin-2-one
N-{4-[2-(2-aminoethyl)phenyl]phenyl}acetamide
3-[1-(cyclohexylmethyl)piperidin-3-yl]-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
2-(2-acetyl-4,5-dimethoxyphenyl)-N-{1-azabicyclo[2.2.2]octan-3-yl}acetamide
N-{1-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]ethyl}pyrimidin-4-amine
3-(4-fluorophenyl)-3-{[3-(1H-pyrazol-1-ylmethyl)phenyl]formamido}propanoic acid
(3ar,6ar)-N-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N-[(4-fluorophenyl)methyl]-N-(2-methoxyethyl)-2,2-dimethylcyclopropane-1-carboxamide
N-ethyl-N-methyl-6-{3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}pyrimidin-4-amine
(3aR,6aS)-2-methyl-5-[(4-methyl-1H-imidazol-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-1,3-dione
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-(4-methoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-ethyl-1-methyl-3-{1-[(3-methylthiophen-2-yl)sulfonyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-4-{[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methyl}-1,3-oxazole
4-({5-[1-(oxolan-2-ylmethyl)-1H-1,2,3-triazol-4-yl]-1,2,4-oxadiazol-3-yl}methyl)morpholine
2-{2-[1-(4-oxo-1,4-dihydroquinoline-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
6-[3-(furan-2-yl)benzoyl]-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
3-{[(cyclopropylmethyl)amino]methyl}-1-[(4-fluorophenyl)methyl]-3-hydroxypiperidin-2-one
N'-cycloheptyl-N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]butanediamide
2-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-{4-[(4-ethoxyphenyl)methyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
2-(morpholin-2-yl)-N-{2-[3-(trifluoromethyl)phenyl]ethyl}acetamide
1-({3-methoxy-4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}methyl)azepan-4-ol
1-{4-[3-({methyl[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)phenoxy]piperidin-1-yl}-2-(thiophen-3-yl)ethan-1-one
2-{4-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}acetamide
1-[(3S,4R)-4-amino-3-methoxypiperidin-1-yl]-3-(pyridin-3-yl)propan-1-one
N-methyl-N-[(5-methylfuran-2-yl)methyl]-6-oxo-1-(prop-2-en-1-yl)piperidine-3-carboxamide
2-{5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}pyrimidin-4-amine
N-[3-(cyclopentyloxy)propyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
{[1-(benzenesulfonyl)-1H-pyrrol-2-yl]methyl}(methyl)[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amine
(4aS,7aR)-1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
ethyl(2-methoxyethyl)[(2-phenyl-1H-imidazol-4-yl)methyl]amine
3-({[6-(azocane-1-carbonyl)-5-methylthieno[2,3-d]pyrimidin-4-yl]amino}methyl)-1λ6-thiolane-1,1-dione
2-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]-6-(propan-2-yl)pyridine-3-carbonitrile
2-oxo-6-(propan-2-yl)-N-{2-[(pyridin-3-yl)amino]ethyl}-1,2-dihydropyridine-3-carboxamide
N-[2-(dimethylamino)ethyl]-N-({1-[(2-fluorophenyl)methyl]piperidin-3-yl}methyl)-1H-imidazole-5-carboxamide
N-[1-(4-methylbenzoyl)piperidin-4-yl]-2,7-dioxo-1,3-diazepane-4-carboxamide
4-[(5-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}-1,2,4-oxadiazol-3-yl)methyl]-1-propylpiperidine
2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]-1-[2-(4-methylpiperazine-1-carbonyl)morpholin-4-yl]ethan-1-one
1-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-(thian-4-yl)piperazine
1-[2-(3,4-dimethoxyphenyl)ethyl]-1-methyl-3-(2-methyl-2H-1,2,3-benzotriazol-4-yl)urea
7-[2-(1H-imidazol-2-yl)benzoyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(3-ethoxypropyl)acetamide
3-{5-[2-(ethylsulfanyl)pyrimidin-5-yl]-4-phenyl-1H-imidazol-1-yl}-1-methylpyrrolidin-2-one
8-[(3,4-dimethoxypyridin-2-yl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
1-{6-ethyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-(pyrrolidin-1-yl)piperidine
(1s,4s)-4-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]cyclohexan-1-ol
1-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]-2-(2-methoxyphenyl)ethan-1-one
N-[4-(3-methoxyphenyl)phenyl]-1-(1,3-thiazole-4-carbonyl)piperidine-3-carboxamide
6-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]pyrimidine-2,4-diamine
1-[(2R,3S,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one