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1-{3-[3-(trifluoromethyl)benzoyl]piperidine-1-carbonyl}cyclopropane-1-carboxamide
2-(dimethyl-1,3-thiazol-5-yl)-N-[2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]acetamide
4-{4-[(propylamino)methyl]phenyl}benzoic acid
N-(5-methyl-1,2-oxazol-3-yl)-2-[4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperazin-1-yl]-2-oxoacetamide
5-acetyl-N-[2-(4-ethylphenoxy)ethyl]-N-methylthiophene-2-carboxamide
4-methyl-N-{2-methyl-5-[2-(2-methyl-1H-1,3-benzodiazol-5-yl)acetamido]phenyl}benzamide
(2S,4S)-4-{[(2,4-difluorophenyl)methyl]amino}-1-(2,3-dihydro-1H-inden-2-yl)-N-methylpyrrolidine-2-carboxamide
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-(2-ethoxyethyl)-1H-pyrazole-3-carboxamide
N-(1-ethyl-1H-1,2,4-triazol-3-yl)-3-propoxypiperidine-1-carboxamide
2-methyl-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}pyrido[2,3-d]pyrimidin-4-amine
3-methyl-5-(2-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}ethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-[1-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)pyrrolidin-2-yl]pyridine
3-[(1-{3-[(3-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazole-5-carbonyl}piperidin-4-yl)oxy]pyridine
1-(4-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}piperazin-1-yl)ethan-1-one
4-hydroxy-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
N4-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-2-{[(4-methylphenyl)methyl]sulfanyl}pyrimidine-4,6-diamine
N-[2-hydroxy-2-(1-methyl-1H-imidazol-2-yl)ethyl]-2-[(2-methylprop-2-en-1-yl)oxy]benzamide
3-(2-amino-1,3-thiazol-4-yl)-N-methyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]propanamide
2-(2-phenyl-1H-imidazol-1-yl)-1-[3-(pyridin-3-yl)azetidin-1-yl]ethan-1-one
4-{[2-(2,5-dimethylphenyl)ethyl](ethyl)amino}butan-1-ol
1-[(3-methoxyphenyl)methyl]-4-[2-(methylsulfanyl)benzoyl]piperazin-2-one
{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[1-(4-methoxyphenyl)ethyl]methylamine
3-(2-methoxyethyl)-1-(pyrrolidine-1-sulfonyl)piperidine-3-carboxylic acid
2-benzyl-N-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-1,3-thiazole-4-carboxamide
1-cyclopropyl-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-5-oxopyrrolidine-3-carboxamide
N-{[(3S,4S)-1-(1-ethenyl-1H-pyrazole-4-carbonyl)-3-hydroxypiperidin-4-yl]methyl}-2-methylpropanamide
N-[2-(dimethylsulfamoyl)ethyl]-2-(methylamino)pyridine-3-carboxamide
(3aS,7aR)-5-methyl-2-{2-[(4-methylphenyl)methyl]benzoyl}-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
2-{1-[1-(2H-1,3-benzodioxol-5-yl)piperidin-4-yl]piperidin-3-yl}-1,2,3,4-tetrahydroisoquinoline
1-[1-(5-acetylpyridin-2-yl)piperidin-4-yl]-N-cyclopropylpiperidine-3-carboxamide
N,4-dimethyl-N-({4-oxo-3H,4H-thieno[3,2-d]pyrimidin-2-yl}methyl)-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
N-methyl-2-(2-oxo-1,3-oxazolidin-3-yl)-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]acetamide
2-[4-(1-benzofuran-2-ylmethyl)-6-hydroxy-1,4-diazepan-1-yl]acetamide
2-(4-methanesulfonylphenyl)-4,6-dimethylpyrimidine
N-{[3-(4-fluorophenyl)oxolan-3-yl]methyl}-3-(1,2-oxazinan-2-yl)propanamide
4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-6-methyl-2-propylpyrimidine
2-(4-chloro-2-{[(2,2-dimethyloxan-4-yl)(methyl)amino]methyl}phenoxy)acetic acid
3-propyl-5-[3-(1H-pyrazol-1-ylmethyl)phenyl]-1,2,4-oxadiazole
3-({methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amino}methyl)-4H-chromen-4-one
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-4-(pyrrolidin-1-ylmethyl)benzamide
4-[1-(2-chlorophenyl)-1H-pyrazol-4-yl]-N-(furan-3-ylmethyl)pyrimidin-2-amine
2-hydroxy-1-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
1-[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-hydroxy-4-methylpentan-1-one
4-[(6-methoxy-3-methyl-1-benzofuran-2-yl)formamido]-N,4-dimethylpentanamide
(2S,4S,5R)-5-(4-chlorophenyl)-4-[(2-methoxyethyl)carbamoyl]-1,2-dimethylpyrrolidine-2-carboxylic acid
(1R,9aR)-1-({[1-(morpholin-4-ylmethyl)cyclopentyl]amino}methyl)-octahydro-1H-quinolizin-1-ol
1-[(3,5-dimethyl-1H-indol-2-yl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-(propan-2-yl)-3-(4H-1,2,4-triazol-4-yl)benzamide
4-(1,3-benzothiazol-2-yl)-2-{[4-(furan-2-carbonyl)piperazin-1-yl]methyl}phenol
(1S,5R)-3-[1-(2H-1,3-benzodioxol-5-yl)piperidin-4-yl]-6-methyl-3,6-diazabicyclo[3.2.2]nonan-7-one