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(2S,4R)-N-[2-(4-fluorophenyl)ethyl]-1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
(4aS,7aR)-1-(2,3-dichlorobenzoyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2,6,8-trimethyl-N-[1-(1,3-thiazol-5-yl)propan-2-yl]quinoline-4-carboxamide
N-methyl-N-[2-({1H-pyrrolo[2,3-b]pyridin-6-yl}amino)ethyl]methanesulfonamide
1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-4-(5-methyl-1,2,4-oxadiazol-3-yl)piperidine
methyl (4aR,7aS)-4-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxylate
3-{[1-(4-methylpiperazine-1-carbonyl)pyrrolidin-3-yl]methyl}benzoic acid
N-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]oxane-4-carboxamide
1-[(4-methyl-1,3-benzoxazol-2-yl)methyl]-3-(3-phenyl-1,2,4-thiadiazol-5-yl)urea
N-methyl-N-{3-[(4-methylphenyl)sulfanyl]propyl}-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-(2-oxoazepan-1-yl)propanamide
8-(2-amino-6-methoxypyrimidin-4-yl)-2-cyclopropyl-2,8-diazaspiro[5.5]undecan-3-one
3-(5-{[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]methyl}thiophen-3-yl)prop-2-yn-1-ol
methyl 2-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-6-methylpyrimidine-4-carboxylate
[(5-cyclopropyl-1,2-oxazol-3-yl)methyl](methyl)({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)amine
1-(8-fluoroquinoline-2-carbonyl)-N,N-dimethylazepan-4-amine
2-{2-[(dimethylamino)methyl]-4-(pyrimidin-2-yl)phenoxy}-N-[1-(naphthalen-1-yl)ethyl]acetamide
2,5-dimethyl-N-(2-phenylpropyl)-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
4-(3-{1-[(2,3-difluorophenyl)methyl]piperidin-4-yl}pyrrolidine-1-carbonyl)pyridin-1-ium-1-olate
2-[3-(1-methyl-1H-imidazole-2-carbonyl)piperidin-1-yl]-4-(pyrrolidine-1-carbonyl)pyridine
4-{[1-(2-fluoro-4-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1-methyl-1H-pyrazole
2-(3-chlorophenyl)-N-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]acetamide
(3S,4S)-1-[(4-fluoro-2-methoxyphenyl)methyl]-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
methyl 4-{[(1R,3S,5S)-3-(4-methoxyphenyl)-8-azabicyclo[3.2.1]octan-8-yl]methyl}-1H-pyrazole-3-carboxylate
3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-1-[(4-phenyloxan-4-yl)methyl]urea
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-{1-[(5-methoxy-3-methyl-1H-indol-2-yl)methyl]piperidin-4-yl}propanamide
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-{[7-fluoro-5-(pyridin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-5-propyl-1,2-oxazole-3-carboxamide
{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}(oxolan-2-ylmethyl)(pyridin-4-ylmethyl)amine
5,6-dimethyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}pyrimidin-4-amine
N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-1-[4-(1H-pyrazol-1-yl)phenyl]piperidin-4-amine
9-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
3-hydroxy-1-(3-phenylpropyl)-3-({[1-(propan-2-yl)piperidin-4-yl]amino}methyl)piperidin-2-one
3-[({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]piperidin-3-ol
N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
3-cyclopentyl-6-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
N-methyl-N-(2-phenyl-1-{1-[2-(thiophen-3-yl)acetyl]piperidin-4-yl}ethyl)pyridine-2-carboxamide
4-[3-(azepane-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]piperazine-1-carbaldehyde
{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(methyl)({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine
N,N-dimethyl-2-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-yl}pyridine-3-carboxamide
[(5-ethylpyridin-2-yl)methyl](methyl){[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}amine
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(1H-1,2,4-triazol-1-yl)benzamide
4-(2-fluoro-6-methoxybenzoyl)-1-(2-methylphenyl)piperazin-2-one
(3S,4R)-4-(4-fluorophenyl)-1-(1-methyl-1H-pyrazole-4-carbonyl)pyrrolidine-3-carboxylic acid
N-ethyl-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-2,5-dimethyl-1,3-thiazole-4-carboxamide
3-cyclobutyl-4-(5-fluoro-2-methylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(cyclopropylmethyl)-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}-N-propylpiperidine-4-carboxamide
(5S,9aS,9bS)-5-(5-acetylthiophen-3-yl)-2-[(3-chlorophenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-[1-(3-methylfuran-2-carbonyl)pyrrolidin-3-yl]-2-(pyridin-4-yl)pyridine