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N'-(furan-2-ylmethyl)-N-(5-methyl-1,3,4-thiadiazol-2-yl)-N'-(3-methylbutan-2-yl)ethanediamide
methyl 6-[(3,4-difluorophenyl)methyl]-2-[(4-fluorophenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-hydroxy-N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine-5-carboxamide
1-(2-cyclohexylethyl)-N-[2-(1H-indol-3-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
4-{5-fluoro-2-[(E)-2-phenylethenyl]pyrimidin-4-yl}morpholine
methyl[(1-methyl-1H-imidazol-2-yl)methyl]({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)amine
5-{2-[3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2-oxazol-3-ol
4-{4-[1-(morpholin-4-yl)ethyl]phenyl}-2-(1,2-oxazol-5-yl)phenol
2-(azepan-1-yl)-N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]acetamide
3-ethyl-8-[(3-methoxyphenyl)methyl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{[3-(methylsulfanyl)phenyl]methyl}-1-(pyrimidin-2-yl)piperidin-3-amine
(2S)-4-carbamoyl-2-(5-cyclopropyl-4-phenyl-1H-imidazol-1-yl)butanoic acid
1-[(1-propyl-1H-imidazol-2-yl)methyl]-3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
5-(2-fluorophenoxymethyl)-N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)-1H-pyrazole-3-carboxamide
1-[4-(2-methoxyethyl)piperazin-1-yl]-2-[(3-methoxyphenyl)amino]butan-1-one
5-{5-[pyridin-3-yl(pyrrolidin-1-yl)methyl]-1,2,4-oxadiazol-3-yl}-1H-1,3-benzodiazole
6-{dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-N,1-dimethyl-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-2-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-[(2,3-difluoro-6-methoxyphenyl)methyl]pyrrolidin-3-yl]-2-methoxyacetamide
4-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidine-1-carbonyl]-1,2-dihydrophthalazin-1-one
6-{2-benzyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl}-2-methyl-2,3-dihydropyridazin-3-one
4-[(4-methylphenyl)sulfanyl]-1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperidine
3,5-dimethoxy-2-({methyl[(1-methylpiperidin-4-yl)methyl]amino}methyl)benzoic acid
2-(2H-1,2,3-benzotriazol-2-yl)-1-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)ethan-1-one
(1R,3S)-3-(2-aminoethoxy)-7-(2,8-dimethylquinoline-4-carbonyl)-7-azaspiro[3.5]nonan-1-ol
1-[4-(2-cyclobutyl-5-fluoro-1H-1,3-benzodiazol-1-yl)piperidin-1-yl]-2-(3-fluorophenyl)ethan-1-one
(2R)-1-[2-methyl-6-(piperidin-4-yl)pyrimidin-4-yl]pyrrolidine-2-carboxamide
1-[(2-fluorophenyl)methyl]-N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
1-(difluoromethyl)-N-methyl-N-{[2-(2-methylpropoxy)phenyl]methyl}-1H-pyrazole-5-carboxamide
5-methoxy-N-methyl-4-oxo-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}-4H-pyran-2-carboxamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[2-(pyridin-4-yl)ethyl]benzamide
4-[4-(oxan-4-yl)piperazin-1-yl]-8-(trifluoromethyl)quinoline
(4aS,8aR)-6-[(3-methyl-1,2-oxazol-5-yl)methyl]-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
6-(2,5-dimethoxyphenyl)-N-[(3-fluorophenyl)methyl]-2-(4-methylpiperazin-1-yl)pyridine-3-carboxamide
2-(dimethylamino)-8-(2,4,5-trimethylphenyl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
N-benzyl-5-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]pyrimidin-2-amine
N-(1-{[3-(furan-2-yl)phenyl]methyl}piperidin-4-yl)methanesulfonamide
N2-(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)-N4-methyl-5H,6H,7H-cyclopenta[d]pyrimidine-2,4-diamine
4-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyridine
(2S)-2-[(2-amino-6-methylpyrimidin-4-yl)amino]-2-phenylethan-1-ol
6-{[(5-methylthiophen-2-yl)methyl]amino}-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
4-{3-[2-(1-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]propyl}morpholine
N-(4-{[3-hydroxy-3-(2-methylphenyl)pyrrolidin-1-yl]methyl}phenyl)acetamide
4-(cyclopropylmethyl)-3-(propan-2-yl)-1-(4,4,4-trifluorobutyl)-1,4-diazepan-5-one
3-[2-oxo-2-(thiomorpholin-4-yl)ethyl]-4-(thiophen-2-ylmethyl)piperazin-2-one
N-(2,3-dimethylphenyl)-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-carboxamide
1-[(3-fluoropyridin-2-yl)methyl]-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
2-{[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-3,4-dimethoxypyridine
5-cyclopropyl-N-(6-hydroxy-6-methylheptan-2-yl)-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-2-(1H-1,2,4-triazol-3-yl)benzamide
N-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)-1-(propan-2-yl)-1H-pyrazole-4-carboxamide