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1-methyl-4-[1-(pyrrolidin-1-yl)cyclopentanecarbonyl]piperazine-2-carboxylic acid
1'-(1,3-benzothiazol-2-yl)-5-butyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-{1-[(4-ethoxyphenyl)methyl]-4-[(3-methyl-1H-indol-2-yl)methyl]piperazin-2-yl}ethan-1-ol
N,6-dimethyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]pyridazin-3-amine
3-[(4-fluorophenyl)formamido]-N-(oxan-2-ylmethyl)propanamide
3-[4-(methylsulfanyl)benzoyl]piperidine
N-methyl-3-(5-methylfuran-2-yl)-N-(piperidin-4-yl)benzamide
ethyl 1-{5-[(dimethylamino)methyl]furan-2-carbonyl}-3-(2-phenoxyethyl)piperidine-3-carboxylate
1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-8-(thiophen-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-ethyl-4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
(4aR,7aS)-1-(cyclopropylmethyl)-4-(3-hydroxynaphthalene-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3,3-dimethyl-1-[(5-{[3-(methylsulfanyl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]urea
7-methoxy-3-(1-methyl-1H-1,3-benzodiazol-2-yl)quinolin-2-ol
3-[4-(prop-2-en-1-yl)piperazine-1-carbonyl]-N-(1H-pyrazol-3-ylmethyl)benzene-1-sulfonamide
(1R,5R)-6-(2-methoxyethyl)-3-(2-methyl-1-benzofuran-7-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
4-[4-(1-methoxyethyl)phenyl]-6-(pyrrolidin-1-yl)pyrimidin-2-amine
5-{3-oxa-9-azaspiro[5.5]undecane-9-carbonyl}-2-(propan-2-yl)-3,4-dihydropyrimidin-4-one
(1R,2R,6S,7S)-4-[8-(trifluoromethyl)quinolin-4-yl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane
3-(1-{1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-2-yl)pyridine
5-{1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]pyrrolidin-2-yl}-3-phenyl-1,2,4-oxadiazole
1-{4-methyl-2-[(2-{[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]methyl}propyl)amino]pyrimidin-5-yl}ethan-1-one
N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,9-dioxaspiro[5.5]undecan-4-amine
N-[(3-fluorophenyl)methyl]-9-methoxy-7-oxo-3-[2-(phenylsulfanyl)acetyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
2-(oxolan-2-ylmethyl)-8-[3-(pyridin-4-yl)propanoyl]-2,8-diazaspiro[4.5]decan-3-one
2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(3-hydroxy-2,2-dimethylpropyl)acetamide
1-[5-({[(2,5-difluorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
13-(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
4-(4-methoxy-2-methylbenzoyl)-1-(4-methylphenyl)piperazin-2-one
5-{2-[2-(dimethylamino)ethyl]piperidine-1-carbonyl}-2-methyl-3,4-dihydropyrimidin-4-one
2-[(2-cyclohexylacetamido)methyl]-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
3-ethoxy-6-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyridazine
3-{1-[(2-chlorophenyl)methyl]-1H-pyrazol-5-yl}-1-(5-oxo-1-propylpyrrolidin-3-yl)urea
N-[(6-ethoxyquinolin-2-yl)methyl]-N-methyloxan-4-amine
1-(2-chlorophenyl)-3-{1-[1-(oxolan-3-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
2-(2,5-dioxoimidazolidin-1-yl)-N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]acetamide
1-[(2-chlorophenyl)methyl]-N-({2,3-dimethylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-1H-1,2,3-triazole-4-carboxamide
(2H-1,3-benzodioxol-5-ylmethyl)(pyridin-3-ylmethyl){[4-(pyrimidin-2-yloxy)phenyl]methyl}amine
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-4-(1H-pyrazol-3-yl)benzamide
1-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(3-methylbutyl)acetamide
3-(5-cyclohexyl-1,3,4-oxadiazol-2-yl)-1-[(2S)-4-methyl-2-phenylpiperazin-1-yl]propan-1-one
1-{3-[2-({[2-(2-fluorophenyl)ethyl]amino}methyl)-4-methoxyphenoxy]-2-hydroxypropyl}piperidin-4-ol
ethyl 2-{1-[3-(dimethylamino)benzoyl]piperidin-2-yl}acetate
5-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrole-1-carbonyl]-N-(2-methoxyethyl)-1-methyl-1H-1,3-benzodiazol-2-amine
7-(cyclopropylmethyl)-2-[6-(dimethylamino)pyridine-3-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
N-(furan-2-ylmethyl)-6-[(3-hydroxy-4-methoxyphenyl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
7-(2,3-dimethoxyphenyl)-4-[(2-ethoxyphenyl)methyl]-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-{[2-(2,3-dimethoxyphenyl)ethyl]carbamoyl}-1H-imidazole-4-carboxylic acid
N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-{[2-(naphthalen-2-yl)pyrimidin-5-yl]methyl}cyclopropanamine
3-(4-methyl-1,3-thiazol-5-yl)-1-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one