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3-(1-{[2-(2-aminoethyl)quinazolin-4-yl]amino}ethyl)adamantan-1-ol
N-[(3R,5S)-5-(ethylcarbamoyl)-1-(3-methylbut-2-en-1-yl)pyrrolidin-3-yl]pyridine-4-carboxamide
1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-2-(4-chloro-3-methyl-1H-pyrazol-1-yl)ethan-1-one
3-(1-methyl-4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-1H-pyrazolo[3,4-d]pyrimidin-6-yl)pyridine
N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)methanesulfonamide
(1S,5R)-6-(morpholine-4-carbonyl)-3-(pyridine-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
6-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-9H-purin-2-amine
3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]-1-[2-(trifluoromethyl)morpholin-4-yl]propan-1-one
1-methyl-2-{[4-(1H-pyrazol-3-yl)piperidin-1-yl]methyl}-1H-indole
6,7-dimethyl-4-({methyl[1-(1,2-oxazol-3-yl)ethyl]amino}methyl)-2H-chromen-2-one
1-[2-fluoro-6-(trifluoromethyl)phenyl]-3-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]urea
2-[(1S,5R)-6-[2-(3,4-dimethylphenoxy)ethyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
1-ethyl-3-methyl-4-(5-{[2-(methylsulfanyl)phenyl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)-1H-pyrazole
2-[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-{2-[(3R,4S)-3-(3-hydroxypropyl)-4-(morpholin-4-yl)piperidin-1-yl]-2-oxoethyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
1-(propane-2-sulfonyl)spiro[azepane-4,2'-chromene]
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
(3S,9aR)-3-ethyl-8-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3,7-dimethyl-11-(1-methyl-1H-indole-2-carbonyl)-3,7,11-triazaspiro[5.6]dodecane
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-cyclopropyl-6-oxo-1,6-dihydropyrimidine-5-carboxamide
3-phenyl-N-[1-(1-{[4-(propan-2-yloxy)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]propanamide
[(3R,4R)-1-{[4-(difluoromethoxy)phenyl]methyl}-4-[(dimethylamino)methyl]pyrrolidin-3-yl]methanol
(3aR,6aS)-5-[(2Z)-5-methyl-2-phenylhex-2-en-1-yl]-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1,5-dimethyl-3-{4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine-1-carbonyl}-1H-indazole
8-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N,2,7-trimethylimidazo[1,2-a]pyridine-3-carboxamide
N-[3-(benzylsulfanyl)propyl]-2,2-dimethylcyclopropane-1-carboxamide
1-(morpholin-4-yl)-3-[1-(quinolin-4-ylmethyl)piperidin-4-yl]propan-1-one
1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}-4-{[3-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
(3R,4R)-1-(3-chlorothiophene-2-carbonyl)-3,4-dimethylpyrrolidin-3-ol
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-3-azaspiro[5.5]undecan-9-amine
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-[3-(methylsulfanyl)propyl]piperidine-4-carboxamide
3-(4-methoxyphenyl)-3-phenyl-1-[4-(pyridin-4-yl)piperazin-1-yl]propan-1-one
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-1-(prop-2-en-1-yl)pyrrolidine-2-carboxamide
2-[3-(1H-pyrazol-1-yl)phenyl]-1H-1,3-benzodiazole-6-carboxylic acid
1-{6-methyl-3-[(4-propylpiperazin-1-yl)methyl]quinolin-2-yl}piperidin-3-ol
[(3R,4R)-4-[(4-ethylpiperazin-1-yl)methyl]-1-[6-methyl-4-(trifluoromethyl)pyridin-2-yl]pyrrolidin-3-yl]methanol
N-(2-methoxyethyl)-1-(1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-4-yl)piperidine-3-carboxamide
4-benzyl-3-ethyl-1-(3-methylfuran-2-carbonyl)-1,4-diazepan-5-one
N-({1-[(6-ethoxy-2,3-dihydro-1H-inden-5-yl)methyl]pyrrolidin-3-yl}methyl)acetamide
1-(dimethyl-1,3-oxazole-4-carbonyl)-4-(3-phenylpropyl)-1,4-diazepane
1-{[5-(3-methoxyphenyl)-1,2-oxazol-3-yl]methyl}-4-(oxolan-3-yl)-1H-1,2,3-triazole
9-(3,4-dihydro-2H-1-benzopyran-2-carbonyl)-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-{[7-(5-acetyl-2-fluorophenyl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}furan-2-carboxamide
N-[(2S)-1-hydroxy-3-phenylpropan-2-yl]-1-benzofuran-3-carboxamide
(1R,5S,6S)-6-({4-[(3-chlorophenyl)methyl]piperazin-1-yl}methyl)-3-azabicyclo[3.1.0]hexane
1-[(2,4-dimethylphenyl)methyl]-3-(2-methoxyethyl)piperidine
8-(1-benzofuran-2-ylmethyl)-3-[(4-methoxyphenyl)methyl]-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(4-chlorophenyl)methyl]-N-ethyl-6-oxo-N-(pyridin-4-ylmethyl)piperidine-3-carboxamide
N-{[1-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)piperidin-3-yl]methyl}thiophene-2-sulfonamide