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1-{2-[(pyrimidin-2-yl)amino]ethyl}piperidine-3-carboxamide
1-{4-methyl-2-[4-(thiophen-3-ylmethyl)piperazin-1-yl]pyrimidin-5-yl}ethan-1-one
6-{3-[(2,4-difluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}pyrazine-2-carboxamide
N-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}-2-(1H-pyrazol-1-yl)butanamide
dimethyl(2-{[1-(5-propyl-1,3,4-oxadiazol-2-yl)piperidin-4-yl]oxy}ethyl)amine
1-cyclobutanecarbonyl-3-[2-(2-methylphenyl)ethyl]piperidine
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-{4-[(2-hydroxyethyl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}propan-1-one
(3R,4R)-1-[3-(dimethylamino)pyrazin-2-yl]-3,4-dimethylpyrrolidin-3-ol
5-fluoro-2-{1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidin-2-yl}-1H-1,3-benzodiazole
5-[4-(2-methoxyphenyl)-2-methylpiperazine-1-carbonyl]-N,N,4-trimethylpyrimidin-2-amine
2-ethoxy-3-(2-{[(3S)-3-fluoropyrrolidin-1-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl)pyridine
2-[2-butyl-5-oxo-4-(3-phenylphenyl)piperazin-1-yl]-2-oxoacetamide
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(2-propyl-1,3-thiazole-4-carbonyl)piperidin-3-yl]propan-1-ol
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-1-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
7-fluoro-2-methyl-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}quinoline-4-carboxamide
N-ethyl-2-[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]pyridine-4-carboxamide
(3S,4R)-1-[3-(methylsulfanyl)propanoyl]-4-phenylpyrrolidine-3-carboxylic acid
3-(3-methoxy-1,5-dimethyl-1H-pyrazol-4-yl)-1-methyl-1-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}urea
(4aS,8aR)-1-(2-aminoethyl)-6-[(4-fluoro-3-methoxyphenyl)methyl]-decahydro-1,6-naphthyridin-2-one
[5-({[(5-chloro-2-methoxyphenyl)methyl](ethyl)amino}methyl)furan-2-yl]methanol
(3aR,5S,6S,7aS)-2-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-octahydro-1H-isoindole-5,6-diol
3-(3-cyclopropyl-1H-pyrazol-5-yl)-4-[(1R)-1-(4-fluorophenyl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-{[4-phenyl-5-(piperidin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl}-1,4-oxazepane
(2S,4R)-4-acetamido-N,N-diethyl-1-[2-(2-methyl-1H-imidazol-1-yl)acetyl]pyrrolidine-2-carboxamide
4-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}-1,4-diazepane-1-carbaldehyde
4-{[(2R)-1-hydroxybutan-2-yl]amino}-N-(pyridin-3-ylmethyl)pyridine-2-carboxamide
1-(2-methoxyphenyl)-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-1H-pyrazole-4-carboxamide
4-{4-[1-(furan-2-ylmethyl)piperidine-3-carbonyl]piperazin-1-yl}-6-methylpyrimidin-2-amine
N-{4-[1-(methoxymethyl)cyclobutaneamido]phenyl}-5-methylfuran-3-carboxamide
2-ethyl-N-[(3-fluorophenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
{5-[(2-butylpyrrolidin-1-yl)methyl]furan-2-yl}methanol
7-(cyclopropylmethyl)-2-[(2,4-dimethoxy-3-methylphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
1-[2-(3-methoxyphenyl)azetidin-1-yl]-2-(trimethyl-1H-pyrazol-1-yl)ethan-1-one
N-(propan-2-yl)-5-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}pyrimidin-2-amine
[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]bis(1,3-oxazol-4-ylmethyl)amine
2-{2-[3-(4-methylpiperazin-1-yl)-3-oxopropyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}propanamide
(3aR,7aS)-5-methyl-2-(5-propyl-1,2,4-oxadiazol-3-yl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole
(2S,4R)-N-ethyl-1-(1-propylpiperidin-4-yl)-4-({[4-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
ethyl 4-(cyclopropylmethyl)-1-[(2,5-dimethylthiophen-3-yl)sulfonyl]piperidine-4-carboxylate
5-[1-(4-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-1-methyl-1H-pyrazole
5-{[7-(2-methoxyphenyl)-4-oxo-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-2-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-[2-(1H-imidazol-1-yl)phenyl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N-methyl-2-(2-oxopiperidin-1-yl)acetamide
4-[4-(9H-fluoren-2-ylmethyl)piperazin-1-yl]-2-(3-methoxypropyl)-2,3-dihydro-1H-isoindole-1,3-dione
3-[4-(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)-1H-1,2,3-triazol-1-yl]propane-1,2-diol
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]-1-ethyl-6-oxopiperidine-3-carboxamide
3-{2-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
5-(2-methoxy-4-methylphenoxymethyl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1,2-oxazole-3-carboxamide
5-fluoro-1-methyl-N-[1-(methylcarbamoyl)cyclohexyl]-1H-indole-2-carboxamide
2-(dimethylamino)-N-(2-methoxyethyl)-4-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]pyrimidine-5-carboxamide