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3-[(4-cyclobutyl-6-methylpyrimidin-2-yl)(methyl)amino]-N-methylpropanamide
N-[2-(dimethylamino)ethyl]-6-fluoro-N-[(2-methylphenyl)methyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
2-{2-[4-(5-chloronaphthalene-1-carbonyl)piperazin-1-yl]ethoxy}ethan-1-ol
2-(5-acetylthiophen-3-yl)-N-[(2,3-difluoro-4-methylphenyl)methyl]acetamide
N-methyl-2-[3-methyl-5-oxo-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-[1-(pyridin-3-yl)ethyl]acetamide
N-(2-methoxyethyl)-3-(piperidine-1-carbonyl)-N-(thiophen-2-ylmethyl)pyrazine-2-carboxamide
(1S,5R)-6-(2-methoxyethyl)-3-[3-(pyrrolidine-1-carbonyl)pyridin-2-yl]-3,6-diazabicyclo[3.2.2]nonan-7-one
(1R,5S,8S)-N-(4-ethenylphenyl)-8-hydroxy-3-azabicyclo[3.2.1]octane-3-carboxamide
2-oxo-N-[1-(thiophen-2-ylmethyl)-1H-pyrazol-5-yl]-1-oxa-3,8-diazaspiro[4.6]undecane-8-carboxamide
3-chloro-5-[1-(3-methylpyridin-4-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
1-[(5-amino-1,3,4-thiadiazol-2-yl)methyl]-3-(1-cyclopentyl-4-methyl-1H-pyrazol-5-yl)urea
1-[3-({2-[(3-methoxyphenyl)methyl]morpholin-4-yl}methyl)phenyl]ethan-1-one
(2,1,3-benzothiadiazol-5-ylmethyl)(methyl){[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}amine
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-(2-hydroxyethyl)-N-propylbenzamide
2-{4-[methyl(2-phenylethyl)amino]-6-oxo-1,6-dihydropyridazin-1-yl}-N-(propan-2-yl)acetamide
8-(butan-2-yl)-1-ethyl-3-(naphthalen-1-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(1H-imidazol-1-yl)-N-methyl-N-(thiophen-3-ylmethyl)benzamide
3-{[(1-{1,9-dioxaspiro[5.5]undecan-4-yl}piperidin-4-yl)oxy]methyl}pyridine
6-(4-fluorophenyl)-7-methyl-2-[(3R)-3-methylpiperazine-1-carbonyl]-7H,8H-imidazo[1,2-a]pyrazin-8-one
2-(4-methoxynaphthalen-1-yl)pyridine-3-carboxamide
3-(3-methoxyphenyl)-1-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]propan-1-one
4-(furan-2-yl)-2-[5-(propan-2-yl)-4-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]-1H-pyrazol-1-yl]pyrimidine
[(2-butyl-1H-imidazol-4-yl)methyl](ethyl){[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}amine
3-[2-(azepan-1-yl)-2-oxoethyl]-4-[(2-ethoxyphenyl)methyl]piperazin-2-one
1-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}but-3-en-1-one
1-{[4-(methylsulfanyl)phenyl]methyl}-4-[3-(pyrrolidine-1-carbonyl)phenoxy]piperidine
1'-(3,5-difluorobenzoyl)-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
5-(2-methoxyphenoxymethyl)-N-methyl-N-[2-(oxan-2-yl)ethyl]-1,2-oxazole-3-carboxamide
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-2-[2-oxo-5-(trifluoromethyl)-1,2-dihydropyridin-1-yl]acetamide
N-(2-methoxyethyl)-4-{2-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
4-(2,3,4-trimethoxyphenyl)-7H-pyrrolo[2,3-d]pyrimidine
2-methoxy-N-[4-(quinolin-3-yl)phenyl]acetamide
(5S)-5-({[(5-propylfuran-2-yl)methyl](pyridin-2-ylmethyl)amino}methyl)pyrrolidin-2-one
N-(1,3-benzoxazol-2-ylmethyl)-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
3-(hydroxymethyl)-1-({4-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)piperidin-3-ol
N-(3-{[(2-fluorophenyl)methyl]sulfanyl}propyl)-4-methyl-3,4-dihydro-2H-1,4-benzoxazine-2-carboxamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-1-[5-(methoxymethyl)thiophene-2-carbonyl]-N-methylpiperidin-3-amine
N-(2,3-dihydro-1H-inden-1-yl)-3-[5-(1H-indol-3-ylmethyl)-1,3,4-oxadiazol-2-yl]propanamide
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-[1-(pyrazin-2-yl)propan-2-yl]-1,2-oxazole-3-carboxamide
2-{1-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]-1,4-diazepan-6-yl}acetic acid
3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-2-[(2-phenylethyl)sulfanyl]pyridine
3-{3-[4-(1H-imidazol-1-ylmethyl)phenyl]phenyl}-1H-pyrazole
2-({[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}methyl)-6-methoxyphenol
3-(2,5-difluorophenyl)-5-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
3-hydroxy-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)pyridine-2-carboxamide
1-[(5-cyclopentylthiophen-2-yl)methyl]-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
8-[3-(4-methyl-1H-pyrazol-1-yl)propanoyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-ethyl-N-methyl-3-{[(2S)-2-(3-methyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]sulfonyl}benzamide
3-{2-[methyl(2-methylpropyl)amino]ethyl}-8-(1-methyl-1H-pyrazole-5-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one