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4-[2-(2-chlorophenyl)ethyl]-11-[(3-ethoxypropyl)amino]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
(3R,4R)-4-ethyl-1-{5-[(4-methylpiperazin-1-yl)methyl]furan-2-carbonyl}piperidine-3,4-diol
1-(4-{[(4-fluorophenyl)methyl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
4-[2-(4-fluorophenoxy)acetyl]-1-(4-methylphenyl)piperazin-2-one
4-{1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]piperidin-3-yl}-2-methyl-6-(pyrrolidin-1-yl)pyrimidine
2-(4-{[3-(trifluoromethyl)phenyl]methyl}morpholin-3-yl)acetic acid
(4aS,8aR)-6-(2-aminopyridine-4-carbonyl)-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
N-(2,1,3-benzoxadiazol-5-ylmethyl)-1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-amine
2-{4-[2-(2,4-dimethoxyphenyl)acetyl]-2-oxopiperazin-1-yl}benzonitrile
2-methyl-1-{[5-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}-1,4-diazepan-5-one
N-{4-[5,6-dimethyl-2-(trifluoromethyl)pyrimidin-4-yl]-1H-pyrrolo[2,3-b]pyridin-6-yl}piperidin-4-amine
2-(methylsulfanyl)-5-[(4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidin-1-yl)methyl]pyrimidine
N-{1-[1-(1,2-oxazol-3-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopentanecarboxamide
3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]propanamide
6-(5-aminopyridin-3-yl)-N-cyclopentylpyridazin-3-amine
N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)acetamide
(4aS,8aR)-1-(3-hydroxypropyl)-6-(4-methylpiperazine-1-carbonyl)-decahydro-1,6-naphthyridin-2-one
N-[(3S,7S,8aS)-3-(cyclohexylmethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,5-difluorobenzamide
6,7-dimethoxy-2-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]-1,2,3,4-tetrahydroisoquinoline
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-1-[(1S,4R)-7,7-dimethyl-2-oxobicyclo[2.2.1]heptan-1-yl]methanesulfonamide
(3aS,6aS)-2-methyl-5-({2-phenylimidazo[1,2-a]pyrimidin-3-yl}methyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(3-methoxy-1,5-dimethyl-1H-pyrazol-4-yl)-1-{2-[(3-methylpyridin-2-yl)amino]ethyl}urea
2-(2-chlorophenoxy)-1-{3-[5-(4-fluorophenyl)-2-methylpyrimidin-4-yl]piperidin-1-yl}ethan-1-one
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-2-(2,4-dioxoimidazolidin-1-yl)acetamide
N-{4-chloro-3-[3-(diethylamino)pyrrolidine-1-carbonyl]phenyl}acetamide
3-{7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decane-2-carbonyl}-4,6-dimethyl-1,2-dihydropyridin-2-one
1-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-3-(4H-1,2,4-triazol-3-yl)piperidine
3-[2-(morpholin-4-ylmethyl)phenyl]thiophene-2-carbonitrile
7-(5-acetylthiophene-2-carbonyl)-2,7-diazaspiro[4.4]nonane-1,3-dione
2,5,6-trimethyl-N-[(1-phenylpyrrolidin-3-yl)methyl]pyrimidin-4-amine
2-(dimethylamino)-N-(2-methoxyethyl)-2-(2-methylphenyl)-N-(1-methylpiperidin-4-yl)acetamide
2-(3-methoxyphenoxymethyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-[2-({methyl[(5-methyl-1H-pyrazol-3-yl)methyl]amino}methyl)phenyl]-6-(2-methylpropyl)-3,4-dihydropyrimidin-4-one
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(quinolin-2-ylmethyl)piperidin-3-yl]propanoic acid
(3-{2-[1-(5-ethyl-2,6-dimethylpyrimidin-4-yl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)dimethylamine
1-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}butan-1-one
4-ethyl-1-methyl-3-{1-[3-(1,2-oxazolidin-2-yl)propanoyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[4-(1H-imidazol-2-yl)piperidin-1-yl]-2-[3-(trifluoromethyl)phenyl]ethan-1-one
2-({benzyl[2-(dimethylamino)ethyl]amino}methyl)-4-(pyrimidin-5-yl)phenol
6-(2-fluoro-4-methoxyphenyl)-7-methyl-N-(oxan-4-ylmethyl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-(2,6-dimethylpyridin-3-yl)-3-[(2-methylphenyl)methoxy]azetidine-1-carboxamide
3-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-9-(thiophene-2-carbonyl)-3,9-diazaspiro[5.5]undecane
N-[3-(methylsulfanyl)phenyl]-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carboxamide
(3S)-N,N-dimethyl-1-[(4-phenyl-1,3-thiazol-2-yl)methyl]azepan-3-amine
N-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-1-phenyl-1H-1,2,3-triazole-5-carboxamide
(1S,6R)-3-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-3,9-diazabicyclo[4.2.1]nonane
1-ethyl-4-{3-[(2-methylphenyl)methoxy]azetidine-1-carbonyl}pyrrolidin-2-one
2-{3-[3-(6-methoxypyridazin-3-yl)phenyl]-1H-pyrazol-1-yl}acetamide
(3S,5R,9R)-5-hydroxy-11-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-1,7,11-triazatricyclo[7.4.0.03,7]tridecane-2,8-dione
5-methyl-4-(pyrrolidin-1-ylmethyl)-2-[3-(trifluoromethyl)phenyl]-1,3-oxazole