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(4aS,7aR)-1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
8-[5-(1,5-dimethyl-1H-pyrazol-4-yl)-1,2-oxazole-3-carbonyl]-1-oxa-8-azaspiro[4.5]decane
2-methoxy-N-[1-(2-phenylethyl)-5-(4-phenylpiperidine-1-carbonyl)-1H-1,3-benzodiazol-7-yl]acetamide
2-{4-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-1-[(4-methoxy-3-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
5-cyclopropyl-N-(3-ethoxypropyl)-1-{9-methoxy-5H,6H-benzo[h]quinazolin-2-yl}-1H-pyrazole-4-carboxamide
4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]-1-(5-methyl-1,2-oxazole-3-carbonyl)piperidine
2-[1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-3-yl]-1H-1,3-benzodiazole
(1R,5R)-6-(cyclopropylmethyl)-3-{pyrazolo[1,5-a]pyridine-3-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
3-chloro-N-(4-{4-[(2-methoxyethyl)amino]piperidin-1-yl}phenyl)benzamide
(3S,4S)-1-[(2-fluoro-4-methoxyphenyl)methyl]-4-(3-methoxyphenyl)piperidin-3-ol
8-[5-(methoxymethyl)thiophene-2-carbonyl]-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
N-(5-oxo-1-phenylpyrrolidin-3-yl)-2-[3-(trifluoromethyl)phenyl]acetamide
7-[(1-ethyl-1H-indol-6-yl)methyl]-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
10-{4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]piperidine-1-carbonyl}-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraen-9-one
3-hydroxy-3-{[(2-methanesulfonylethyl)amino]methyl}-1-[(3-methylphenyl)methyl]piperidin-2-one
N-[1-(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)piperidin-4-yl]pyridin-2-amine
2-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]methyl}-5-methoxy-3-methyl-1H-indole
(4aR,6R,8aS)-8a-(methoxymethyl)-2-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-6-(morpholin-4-yl)-decahydroisoquinoline
1-{2-oxo-2-[(1S,5R)-7-oxo-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethyl}-1,4-dihydroquinolin-4-one
N-[2-(dimethyl-1H-1,2,4-triazol-1-yl)ethyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
3-{[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]amino}-N-(pyridin-2-ylmethyl)-5-(pyrrolidine-1-sulfonyl)benzamide
N3-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)-N5-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
2-[4-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)phenyl]-3,4,5,6,7,8-hexahydroquinazolin-4-one
4-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridin-2-amine
N-(cyclopropylmethyl)-3-(5-methylthiophen-2-yl)-5-(morpholine-4-sulfonyl)benzamide
1-[(3R,5S)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]-3-(4-phenylphenyl)propan-1-one
1-(2H-1,3-benzodioxol-5-yl)-5-[(2,4-dimethoxyphenyl)methyl]-1H-1,2,4-triazole
N4-[2-(3,5-dimethoxyphenyl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
1-{4-[(2-methylpyridin-3-yl)oxy]piperidine-4-carbonyl}azetidin-3-amine
1-[6-hydroxy-4-(4-methylquinolin-2-yl)-1,4-diazepan-1-yl]-2-methoxyethan-1-one
1-(4-aminobutanoyl)-4-(2,3-dihydro-1H-inden-5-yloxy)piperidine-4-carboxylic acid
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-[(4-fluorophenyl)methyl]-5-(2-methoxyacetamido)-1H-1,3-benzodiazole-7-carboxamide
1-[1-(1-benzofuran-5-ylmethyl)piperidin-4-yl]-3-(pyrrolidine-1-carbonyl)piperidine
3-(4-hydroxyphenyl)-1-[(1S,5R)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
5-tert-butyl-4-[(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)methyl]furan-2-carboxamide
2-acetyl-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]benzamide
2-(1H-1,2,3,4-tetrazol-1-yl)-1-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
2-{5-[1-(1H-pyrazol-1-yl)propan-2-yl]-3-(thiophen-2-ylmethyl)-1H-1,2,4-triazol-1-yl}pyridine
N-(dimethyl-1H-1,2,4-triazol-3-yl)-4-{[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}benzamide
4-[3-(2-chlorophenoxy)azetidine-1-carbonyl]-1-cyclopentylpyrrolidin-2-one
3-(3-{1-[(1-ethyl-1H-imidazol-5-yl)methyl]-1H-pyrazol-3-yl}phenyl)-6-methoxypyridazine
3-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]-1,2-dihydropyridin-2-one
N-[2-(3-hydroxypiperidin-1-yl)ethyl]-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetamide
ethyl 1-(3-chlorobenzenesulfonyl)-4-[(4-methoxyphenyl)methyl]piperidine-4-carboxylate
(3aS,6aS)-2-cyclopentanecarbonyl-5-[2-(1,3-thiazol-4-yl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{[2-(2H-1,3-benzodioxol-5-yl)-8-methoxy-2,3,4,5-tetrahydro-1,5-benzothiazepin-5-yl]methyl}-5-methoxyphenol
2-(difluoromethoxy)-N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]benzamide
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-(2,2,2-trifluoroethyl)acetamide
N'1-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}cyclopropane-1,1-dicarboxamide