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2-[2-(3,4-dichlorophenyl)morpholin-4-yl]pyrimidin-4-amine
2-(2,3-dihydro-1H-inden-1-yl)-N-[2-(propane-2-sulfonyl)ethyl]acetamide
1-{5-[(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]imidazo[2,1-b][1,3]thiazole-6-carbonyl}azocane
N4-[2-(5-chloro-1H-1,3-benzodiazol-2-yl)ethyl]-6-methylpyrimidine-2,4-diamine
2-(1,2-benzoxazol-3-yl)-N-[2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)ethyl]acetamide
(1R,5R)-6-benzyl-3-(5-methyl-1,2-oxazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]thiophene-3-carboxamide
4-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1λ6-thiomorpholine-1,1-dione
6-ethyl-2-methyl-4-(3-phenoxyazetidine-1-carbonyl)quinoline
1-(cyclohexylmethyl)-6,7-dimethoxy-3-{[methyl(thiophen-3-ylmethyl)amino]methyl}-1,2-dihydroquinolin-2-one
1'-cyclobutanecarbonyl-5-methanesulfonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-N,N-dimethylpiperidine-1-carboxamide
ethyl 1-(1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
3-(1H-1,3-benzodiazol-1-yl)-N-[1-(3-phenylpropyl)piperidin-3-yl]propanamide
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-{[(1,3-thiazol-2-yl)carbamoyl]methyl}propanamide
3-({[2-(3-methylphenyl)pyrimidin-5-yl]methyl}amino)-1-[4-(propan-2-yl)piperazin-1-yl]propan-1-one
6-[4-(cyclobutylmethyl)piperazin-1-yl]-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide
3-{4-[3-(2-methylphenyl)-3-phenylpropanoyl]piperazin-1-yl}propanamide
methyl 4-[({2-[5-oxo-1-(thiophen-2-ylmethyl)pyrrolidin-2-yl]ethyl}amino)methyl]benzoate
3-methoxy-N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)propanamide
3-ethyl-5-methyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-1,2-oxazole-4-carboxamide
1-[3-(3-ethylphenoxy)azetidin-1-yl]-2-(morpholin-4-yl)butan-1-one
3-chloro-N-cyclopentyl-4-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}benzamide
(3S)-1-[4-(4-fluorophenyl)oxane-4-carbonyl]-N,N-dimethylazepan-3-amine
2-[(1-ethylpyrrolidin-2-yl)methyl]-2,3-dihydro-1,2-benzothiazol-3-one
1-{4-[1-methyl-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperazin-1-yl}ethan-1-one
1-[2-(4-methoxyphenyl)ethyl]-6-oxo-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
methyl 3-(cyclobutylmethoxy)-5-[(2R)-2-methylpiperazine-1-carbonyl]benzoate
2-[4-(5-ethyl-2-methylpyrimidin-4-yl)piperazin-1-yl]benzonitrile
1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-2-(propan-2-yl)-2,5-dihydro-1H-pyrrole
(1S,6R)-3-{[3-(morpholin-4-ylmethyl)phenyl]methyl}-3,9-diazabicyclo[4.2.1]nonane
8-[(2S)-2-amino-3-hydroxypropanoyl]-2-[(4-chlorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-[2-(4-fluorobenzenesulfonyl)ethyl]-3-(1-methyl-1H-pyrazol-5-yl)propanamide
3-{[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]amino}pyrrolidin-2-one
4-(4-methoxyphenyl)-4-oxo-N-[1-(2-phenylethyl)piperidin-3-yl]butanamide
[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl][(5-ethylpyridin-2-yl)methyl]methylamine
(1R,2S,9S)-11-(1,3-benzothiazol-2-yl)-7,11-diazatricyclo[7.3.1.02,7]tridecan-6-one
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(furan-2-yl)-2-oxoacetamide
7-methyl-2-[2-(4,6,7-trimethyl-1-benzofuran-3-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
5-(4-methanesulfonylpiperazine-1-carbonyl)-2-(2-methyl-1,3-thiazol-4-yl)pyrimidin-4-ol
1-(cyclohexylmethyl)-2-(methoxymethyl)-6-methyl-4-oxo-N-(pyridin-4-ylmethyl)-1,4-dihydropyridine-3-carboxamide
1-{[2-cyclohexylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-4-(cyclopropylmethyl)piperazine
5-{3-[4-(4-chlorophenyl)-4-hydroxypiperidin-1-yl]-3-oxopropyl}-5-{[4-(methylsulfanyl)phenyl]methyl}pyrrolidin-2-one
[(3R,4R)-4-[(dimethylamino)methyl]-1-(5-ethyl-2,6-dimethylpyrimidin-4-yl)pyrrolidin-3-yl]methanol
3-[1-(2,1,3-benzoxadiazol-5-ylmethyl)piperidin-4-yl]-N-(2-chlorophenyl)propanamide
1-methyl-3-({2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)pyrrolidin-2-one
2-[4-(dimethylamino)phenyl]-1-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
5-{[8-(6-methylpyridin-2-yl)-1,8-diazaspiro[4.5]decan-1-yl]methyl}-N-propylpyrimidin-2-amine
(3S,4R)-3-ethyl-4-methyl-1-{2-[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]-1,3-thiazole-4-carbonyl}piperidin-4-ol