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2-methyl-4-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
ethyl (4aS,8aR)-6-[2-methyl-6-(1H-pyrazol-1-yl)pyrimidin-4-yl]-decahydro-1,6-naphthyridine-4a-carboxylate
[(3R,5R)-1-(1-ethyl-1H-pyrazole-3-carbonyl)-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
2-benzyl-8-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-2,8-diazaspiro[4.5]decan-1-one
2-{4-[(4-acetylpiperazin-1-yl)methyl]phenyl}-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-5-(1H-pyrazol-1-ylmethyl)furan-2-carboxamide
2-({3-[4-(4-chlorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)-4-methoxyphenol
N-({1-[(2-phenylethyl)carbamoyl]piperidin-3-yl}methyl)pyridine-3-carboxamide
3-[(3R,4S)-3-amino-4-propylpyrrolidine-1-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
4-[3-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-6-(methoxymethyl)pyrimidine
1-{1'-[(1S,3R)-3-aminocyclopentanecarbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}-2-methoxyethan-1-one
2-methyl-5-{3-[1-(pyridin-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}-1,3-benzoxazole
2-methyl-4-(4-{octahydro-1H-pyrido[1,2-a]piperazine-2-carbonyl}phenyl)butan-2-ol
6-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}pyridine-2-carboxylic acid
N-{1-[1-(4-methylbenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}oxolane-3-carboxamide
1-(2-methoxyphenyl)-N,N-dimethyl-1H-pyrazole-4-carboxamide
N-(dicyclopropylmethyl)-N-methyl-3-[(thiophen-2-ylmethyl)amino]benzamide
N-[(3R,4S)-4-cyclopropyl-1-{2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]acetyl}pyrrolidin-3-yl]methanesulfonamide
7-(2,2-dimethylpropyl)-2-(1,4-dithiepan-6-yl)-2,7-diazaspiro[4.5]decane
N-[2-(dimethylamino)ethyl]-5-(pyrrolidine-3-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)acetamide
3-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-1-[1-(propan-2-yl)-1H-1,2,3-triazol-4-yl]urea
N-{[5-(4-methoxyphenyl)-1,2-oxazol-3-yl]methyl}thiolan-3-amine
(1-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)(1-methyl-1H-imidazol-2-yl)methanol
7-[2-(2-methoxy-4-methylphenoxy)ethyl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
4-{5-[(N-methylmethanesulfonamido)methyl]furan-2-yl}-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxylic acid
2,7-dimethyl-N,N-bis(1,3-oxazol-4-ylmethyl)imidazo[1,2-a]pyridine-3-carboxamide
benzyl 7-(oxan-4-yl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxylate
9-[(1,3-dimethyl-1H-pyrazol-5-yl)sulfonyl]-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
8-[(3-methoxyphenyl)methyl]-1-(3-methoxypropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(3,5-dichloropyridin-4-yl)methyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane
1-(4-ethylpiperazin-1-yl)-3-(1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}piperidin-4-yl)propan-1-one
3-{1-[(2S)-2-hydroxypropanoyl]piperidin-4-yl}-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
2-ethyl-8-[6-methyl-2-(methylsulfanyl)pyrimidin-4-yl]-2,8-diazaspiro[4.5]decan-3-one
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
N-cyclopentyl-1-[1-(3-methylfuran-2-carbonyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
6-[2-(4-methoxy-3-methylphenyl)-1H-imidazol-1-yl]quinoxaline
4-methyl-6-[3-(1H-pyrazol-5-yl)piperidin-1-yl]pyrimidin-2-amine
3-(2-propyl-2,5-dihydro-1H-pyrrol-1-yl)-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraene
N-[(3R,4S)-1-acetyl-4-(propan-2-yl)pyrrolidin-3-yl]-3-chlorobenzene-1-sulfonamide
4,6-dimethyl-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}pyridine-3-carboxamide
4-[1-butyl-5-(1-methyl-1H-pyrazol-5-yl)-1H-1,2,4-triazol-3-yl]benzamide
N-[(1-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}piperidin-3-yl)methyl]-2H-1,3-benzodioxole-5-carboxamide
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
3-methyl-6-{5-[(2,2,3,3-tetrafluoropropoxy)methyl]-1,2,4-oxadiazol-3-yl}pyridazine
N-[3-(8-methoxyquinolin-5-yl)phenyl]acetamide
1-(2,6-dimethylpyridin-4-yl)-4-(5-methyl-1,2-oxazole-3-carbonyl)piperazine
3-[(1,2-oxazol-3-ylmethyl)sulfamoyl]-N-(2,2,2-trifluoroethyl)benzamide
2-{[4-(oxan-4-yl)piperazin-1-yl]methyl}-1H-1,3-benzodiazole