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6-methoxy-2-{5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}-1,2,3,4-tetrahydroisoquinoline
1-{4-chloro-1H-pyrrolo[2,3-b]pyridin-6-yl}-4-(piperidin-1-yl)piperidine-4-carboxamide
1-[4-ethoxy-3-(1H-pyrrol-1-yl)phenyl]-3-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}urea
4-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N-benzyl-3-(1-ethyl-1H-imidazol-2-yl)-N-methylpiperidine-1-sulfonamide
2-benzyl-8-[2-(2-hydroxyethoxy)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
1-(3-propyl-1H-pyrazole-5-carbonyl)-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylcyclobutanamine
4-(1-{5-[(benzyloxy)methyl]-4-phenyl-1H-imidazol-1-yl}ethyl)pyrimidine
N-[2-(3-fluorophenyl)ethyl]-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-{1-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-1H-imidazol-2-yl}benzoic acid
4-(1H-imidazol-1-ylmethyl)-1-[4-(1H-pyrazol-3-yl)benzoyl]piperidin-4-ol
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-1-(5-ethyl-2-methylpyrimidin-4-yl)piperidin-4-amine
1-{5-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]thiophen-2-yl}ethan-1-one
(2R)-2-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]pyrrolidine
(3aR,6aR)-2-methyl-N-[(4-oxo-3,4-dihydrophthalazin-1-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N-[(3S,4R)-4-(propan-2-yl)-1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}pyrrolidin-3-yl]acetamide
1-(4-{[1-(3,5-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]amino}piperidin-1-yl)ethan-1-one
6-fluoro-4-methyl-2-[2-(trifluoromethyl)morpholin-4-yl]quinoline
(1,4-dioxan-2-ylmethyl)({[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})amine
N,6-dimethyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-2-oxo-4-(pyridin-3-yl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-2-methylpyrido[2,3-d]pyrimidin-4-amine
N-{2-methyl-4-[(2S)-2-phenylbutanamido]phenyl}pentanamide
3-({3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}methyl)-N-methyl-1,2,4-oxadiazole-5-carboxamide
N-[(3R,4R)-3-hydroxy-1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]piperidin-4-yl]pyridine-4-carboxamide
(3aR,7aS)-2-[1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
N-(2-ethylphenyl)-3-[(2,3,5,6-tetramethylphenyl)formamido]propanamide
2-(cyclopentylmethyl)-1-(3-methoxypropyl)-6-methyl-4-oxo-N-(pyridin-3-ylmethyl)-1,4-dihydropyridine-3-carboxamide
(1S,4S)-2-[4-(4-chlorophenoxy)piperidine-4-carbonyl]-2-azabicyclo[2.2.1]heptane
N-methyl-5-oxo-1-(prop-2-en-1-yl)-N-(pyrazin-2-ylmethyl)pyrrolidine-3-carboxamide
2-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-6-methylpyridine
methyl 4-({[(3S,5S)-1-{[4-(diethylamino)phenyl]methyl}-5-[(pyridin-3-ylmethyl)carbamoyl]pyrrolidin-3-yl]amino}methyl)benzoate
6-[1-(4-chloro-2-methylphenoxy)ethyl]-3-cyclopropyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
4-ethyl-3-(1-{1H-pyrazolo[1,5-a]imidazole-7-carbonyl}piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{1-[(3-chlorophenyl)methyl]piperidin-3-yl}-4-(4-fluorophenyl)piperazine
4-(2-methoxyphenoxy)-1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidine
methyl (2S,4R)-1-[(3-chlorophenyl)methyl]-4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzamido]pyrrolidine-2-carboxylate
(2S,4S)-4-[(adamantan-2-yl)amino]-N-ethyl-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
2-(2-ethyl-1H-imidazol-1-yl)-1-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
N,N-dimethyl-2-[(1S,5R)-6-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
(1S,5R)-3-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(2-methoxyacetyl)-N-{2-[3-(propan-2-yloxy)phenyl]ethyl}piperidine-4-carboxamide
2-({3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}methyl)-5-methoxy-4H-pyran-4-one
[(3R,4R)-4-(azepan-1-ylmethyl)-1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}pyrrolidin-3-yl]methanol
N-(oxolan-3-ylmethyl)-3-[(pyrimidin-4-ylmethyl)sulfamoyl]benzamide
N,N-dimethyl-2-[(thiolan-3-yl)amino]ethane-1-sulfonamide
1-(2,3-dihydro-1H-inden-5-yl)-3-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]urea
4-methoxy-N-{[1-(2-methylpyridine-3-carbonyl)piperidin-3-yl]methyl}benzene-1-sulfonamide
N5-[2-(cyclohex-1-en-1-yl)ethyl]-1-[(2-methoxyphenyl)methyl]-N3,N3-dimethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-[(3R,5S)-5-(diethylcarbamoyl)-1-methylpyrrolidin-3-yl]-6-methylpyridine-3-carboxamide