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{[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[1-(propan-2-yl)piperidin-3-yl]methyl}amine
1-{2-methyl-5-[2-(pyridin-3-yl)piperidine-1-carbonyl]phenyl}imidazolidin-2-one
3-(hydroxymethyl)-1-{[3-(2-methylphenyl)phenyl]methyl}piperidin-3-ol
(2S)-2-{[2-(4-ethylpiperazin-1-yl)-2,3-dihydro-1H-inden-2-yl]formamido}propanamide
4-{3-[4-(4-fluorophenyl)piperazine-1-carbonyl]piperidin-1-yl}-2-(thiophen-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
3-(3-methylbutyl)-8-(quinoline-6-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-{2-oxo-2-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]ethyl}imidazolidin-2-one
5-[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-{2-[(5-{1-[(2,4-difluorophenyl)methyl]piperidin-4-yl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}azepane
1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
7-methyl-2-[3-(piperazin-1-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
{[(1R,5S,6S)-3-[(6-methoxynaphthalen-2-yl)methyl]-3-azabicyclo[3.1.0]hexan-6-yl]methyl}dimethylamine
2-ethyl-N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-4-methyl-1,3-oxazole-5-carboxamide
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-2-methyl-1,3-thiazole-4-carboxamide
N-ethyl-2-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-amine
2-(3-hydroxypropyl)-9-(2,4,5-trimethylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-(dimethylamino)-2-(4-fluorophenyl)acetamide
1-[5-(dimethyl-1,2-oxazole-4-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl]-4-methylpiperazine
8-(3-phenoxybenzoyl)-2,8-diazaspiro[4.5]decan-3-one
1-(1,2-oxazole-3-carbonyl)-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
5-{3-[1-(oxan-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}pyrimidine
{4-[(3-fluorophenyl)methyl]-1-(1H-indol-3-ylmethyl)piperidin-4-yl}methanol
9-(2,3-difluorobenzoyl)-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
(4aS,7aR)-1-(4-hydroxybenzoyl)-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl][(dimethyl-1,2-oxazol-4-yl)methyl]methylamine
N-methyl-N'-[2-(methylsulfanyl)phenyl]-N-[1-(1,2-oxazol-3-yl)ethyl]butanediamide
1-[3-(difluoromethoxy)phenyl]-3-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]urea
1-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(morpholin-4-yl)ethan-1-one
3-{[cyclopropyl(3-methylbutyl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
2-{[(3aS,6aS)-5-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-octahydropyrrolo[2,3-c]pyrrol-1-yl]methyl}-6-methylpyridine
N-[2-(trifluoromethyl)phenyl]-2-oxa-7-azaspiro[4.5]decane-7-carboxamide
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-(prop-2-en-1-yl)-N-(pyridin-2-ylmethyl)propanamide
2-{3-[(2,6-dichlorophenyl)methyl]-5-(morpholin-4-ylmethyl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
(3S,9aR)-3-[(4-chlorophenyl)methyl]-8-(naphthalene-2-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-{2-[(2-amino-5,6-dimethylpyrimidin-4-yl)(methyl)amino]ethyl}piperidin-2-one
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[(6-methylpyridin-2-yl)methyl]-2,3-dihydro-1H-indene-2-carboxamide
6,8-dimethyl-2-({[(1r,4r)-4-hydroxycyclohexyl]amino}methyl)quinolin-4-ol
3,5-dichloro-N,4-dimethyl-N-[3-(oxolan-2-yl)propyl]benzamide
methyl 4-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]pentanoate
1-{4-[5-(3,4-dimethylphenyl)-4-phenyl-1H-imidazol-1-yl]piperidin-1-yl}ethan-1-one
[3-(pyridazine-4-carbonyl)-9-(pyridin-2-ylmethyl)-3,9-diazaspiro[5.5]undecan-1-yl]methanol
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-1-[(4-methylphenyl)methyl]-5-oxopyrrolidine-3-carboxamide
{[(3R,4S)-1-(4-methoxypyrimidin-2-yl)-4-propylpyrrolidin-3-yl]sulfamoyl}dimethylamine
1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-4-(pyridin-3-yl)piperidin-4-ol
N-cyclopropyl-N-{[2-(3-methoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-3-[(2-fluorophenyl)formamido]propanamide
methyl 2-{[(3-chlorophenyl)methyl]sulfamoyl}-6-(3-methylbutanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-(azocan-1-yl)-3-(2-{[ethyl(methyl)amino]methyl}-5-methoxyphenoxy)propan-2-ol
4-(3-ethyl-1H-pyrazole-4-amido)-N-phenylpiperidine-1-carboxamide
3-({2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}sulfamoyl)-N,N-dimethylbenzamide