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N-[(2-chlorophenyl)methyl]-1-(cyclohexylmethyl)-6-oxopiperidine-3-carboxamide
4-(1-{2-[(propan-2-yl)carbamoyl]ethyl}piperidin-3-yl)benzoic acid
N-ethyl-6-methyl-5-{5-[(3-methyl-1H-pyrazol-1-yl)methyl]-1,2,4-oxadiazol-3-yl}-1,2,3,4-tetrahydro-2,7-naphthyridine-2-carboxamide
3-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-3-methyl-1-(6-methylpyridin-3-yl)urea
N-{2-[(pyridin-3-yl)amino]ethyl}quinoxaline-5-carboxamide
3-[2-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-oxoethyl]-4-(propan-2-yl)piperazin-2-one
1-({5-[(4-fluoro-3-methylphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
N-({1-[(6-chloropyridin-3-yl)methyl]pyrrolidin-3-yl}methyl)propane-1-sulfonamide
1-(2-phenoxyethyl)-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperazine
1-(4-chloro-2-methoxy-5-methylphenyl)-3-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-3-methylurea
[(3R,4S)-4-[(4-ethylpiperazin-1-yl)methyl]-1-[(2-ethylpyrimidin-5-yl)methyl]pyrrolidin-3-yl]methanol
methyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}amine
6-(4-methanesulfonylphenyl)-2-methyl-1H-imidazo[4,5-b]pyridine
N,N,2-trimethyl-7-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
3-{2-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
N-methyl-1-(1-methylpiperidin-4-yl)-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}piperidine-3-carboxamide
2-(3-methylphenyl)-5-(3-phenylpiperazine-1-carbonyl)pyrimidin-4-ol
{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}({2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl})amine
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-4-(4-methylphenoxy)piperidine-4-carboxamide
2-[(3R,4S)-3-{2-[4-(hydroxymethyl)phenyl]acetamido}-4-(propan-2-yl)pyrrolidin-1-yl]-N-methylacetamide
1-(furan-2-yl)-2-{3-oxo-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-9-yl}ethane-1,2-dione
3-[5-(benzylsulfanyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-[(4-methoxyphenyl)methyl]piperidine
9-(2-methoxybenzenesulfonyl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
N-({3-[(dimethylamino)methyl]phenyl}methyl)-N-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-(furan-2-ylmethyl)-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)piperidine-4-carboxamide
(4aS,7aR)-1-(3-methoxybenzenesulfonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(2-chloro-4-fluorophenyl)methyl]-4-[4-(piperidine-1-carbonyl)phenoxy]piperidine
2-{4-[(E)-2-phenylethenyl]-1H-pyrazol-1-yl}-N-(1-propyl-1H-1,2,3-triazol-4-yl)acetamide
methyl 3-(furan-2-amido)-5-[(1-hydroxypropan-2-yl)amino]-1-(3-methylbutyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-{[1-(2-{[1,2,4]triazolo[4,3-b]pyridazin-6-yloxy}acetyl)piperidin-3-yl]methyl}furan-2-carboxamide
N-(1,4-dioxan-2-ylmethyl)-2-[4-(trifluoromethyl)phenyl]-1,3-benzoxazole-5-carboxamide
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
(2R,3R,6R)-5-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
N1,N1-dimethyl-N3-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}piperidine-1,3-dicarboxamide
3-fluoro-N-{1-[1-(thian-4-yl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
4-{4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
(2E)-1-{4-[(2-chlorophenyl)methyl]-4-(hydroxymethyl)piperidin-1-yl}-4-methylpent-2-en-1-one
8-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
2-(2-phenylethyl)-N-(2,2,2-trifluoroethyl)-1,3-benzoxazole-5-carboxamide
N-tert-butyl-2-(4-{[methyl(1H-pyrazol-3-ylmethyl)amino]methyl}phenoxy)acetamide
2-amino-3-ethyl-N-methyl-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-3H-imidazo[4,5-b]pyridine-6-carboxamide
5-[1-(1-benzylpyrrolidin-3-yl)-1H-1,2,3-triazol-4-yl]-2-methoxypyridine
3-[(2R,3R,6R)-5-(pyridine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
2-amino-6-cyclobutanecarbonyl-4-(4-hydroxy-2,6-dimethylphenyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-(2H-1,3-benzodioxol-5-ylmethyl)-6-({methyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
5-methanesulfonyl-1'-(oxolane-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
methyl 4-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}piperazine-1-carboxylate
methyl 6-{[4-(1,3-benzoxazol-2-yl)piperazin-1-yl]methyl}pyridine-2-carboxylate
1-[2-(4-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]-2-phenylpiperazine
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-2-oxo-1,3-oxazolidine-4-carboxamide