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N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)pyridine-2-carboxamide
4-({4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-1-yl}methyl)-1H-pyrazole-3-carboxylic acid
3-(1-{1-[(3-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(2-methylphenyl)urea
4-[1-(3,6-dimethyl-1-benzofuran-2-carbonyl)azetidin-3-yl]pyridine
(2S,4R)-1-[3-(2-chlorophenyl)-5-methyl-1,2-oxazole-4-carbonyl]-4-(dimethylamino)pyrrolidine-2-carboxylic acid
6-(2-chlorophenyl)-N-[(2S)-1-hydroxypropan-2-yl]-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-[3-(4-fluorophenoxy)propyl]-4-(1H-1,2,3-triazole-5-carbonyl)piperazine
2-{4-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}pyridine-3-carboxamide
3-(azocan-1-yl)-1-[4-(oxan-4-yl)piperazin-1-yl]propan-1-one
1-(6-chloropyridazin-3-yl)-N-[1-(2-methylpropyl)piperidin-4-yl]piperidin-4-amine
4-[(5-methoxy-2-methyl-3-phenyl-1-benzofuran-6-yl)methyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(3aS,6aR)-3-[2-(4-fluorophenyl)ethyl]-5-[(1-methyl-1H-imidazol-2-yl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
3-[2-(3,4-difluorophenyl)ethyl]-1-(3-fluoropropyl)piperidine
N4-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-6-methylpyrimidine-2,4-diamine
2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)acetamide
7-[2-(2-chlorophenyl)acetyl]-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-(2-methyl-1-benzofuran-5-yl)-1-(1-methylpiperidin-4-yl)-1-(pyridin-4-ylmethyl)urea
5-(furan-2-ylmethyl)-5-{3-[(2S,6S)-4-methyl-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-3-oxopropyl}pyrrolidin-2-one
4-[(5-methanesulfonyl-2-methylpyrimidin-4-yl)amino]-1-(4-methoxyphenyl)pyrrolidin-2-one
4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-(1,2,3,4-tetrahydronaphthalene-2-carbonyl)piperidine
1-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]-4,4,4-trifluorobutan-1-one
2-(2-fluoro-4-methylphenyl)-2-{4-[(3-methoxyphenyl)methyl]piperazin-1-yl}acetic acid
methyl[2-(pyridin-2-yl)ethyl]{[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}amine
N-[(1-cyclopentylpiperidin-3-yl)methyl]-N-[2-(piperidin-1-yl)ethyl]-2-(1H-1,2,4-triazol-1-yl)acetamide
2-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridin-3-ol
1-[(2-methylphenyl)methyl]-N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
4-[2-(dimethylamino)-2-(4-fluorophenyl)acetamido]oxane-4-carboxylic acid
5-ethyl-2,3-dimethyl-N-[(5-methylfuran-2-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
methyl({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})[1-(1,2-oxazol-3-yl)ethyl]amine
8-(5-ethyl-1,2,4-oxadiazol-3-yl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
2-[(2-fluorophenyl)methyl]-N-methyl-N-(2-phenylethyl)-1,3-benzoxazole-6-carboxamide
2-(2-methyl-1H-imidazol-1-yl)-1-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
6-(3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyrimidine-2,4-diamine
5-ethyl-N-[2-(oxan-2-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
N,N-dimethyl-2-[methyl({4-[6-oxo-4-(pyridin-4-yl)-1,6-dihydropyrimidin-2-yl]phenyl}methyl)amino]acetamide
1-[(2-methyl-1H-imidazol-4-yl)methyl]-4-(pyrimidin-2-yl)-1,4-diazepane
N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-4-(pyridin-3-yl)pyrimidin-2-amine
[(1-methyl-1H-pyrazol-4-yl)methyl](2-methylpropyl){[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amine
N-[2-(3-methanesulfonamidopropanamido)-4-methylphenyl]cyclohexanecarboxamide
3-(1H-1,2,3-benzotriazol-1-yl)-5-(pyrrolidine-1-sulfonyl)benzoic acid
1-amino-N-({1-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]pyrrolidin-3-yl}methyl)cyclopentane-1-carboxamide
1-{3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-4-(thiophene-2-carbonyl)piperazine
3-({methyl[(3-methylpyridin-4-yl)methyl]amino}methyl)-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
2,5-dioxo-6-[3-(pyridin-3-yloxy)propyl]-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
4-{4-phenyl-1-[2-(pyrazin-2-yl)ethyl]-1H-imidazol-5-yl}benzoic acid
2-methoxy-N-[(4-methyl-1H-imidazol-2-yl)methyl]-2-phenylacetamide
3-(1-cyclopentanecarbonylpiperidin-4-yl)-1-[3-(2-methoxyethoxy)phenyl]urea
1-[(3-methoxyphenyl)methyl]-6-oxo-N-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]piperidine-3-carboxamide
N-[(2-ethoxypyridin-3-yl)methyl]-3-(1-methylpiperidin-2-yl)propanamide
5-methyl-1-[4-(4-{[(2R)-oxolan-2-ylmethyl]amino}piperidin-1-yl)phenyl]pyrrolidin-2-one