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3-(2,4-difluorophenyl)-4-(1H-imidazol-2-yl)-1H-pyrazole
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-[1-(4-methylpyridin-2-yl)propyl]acetamide
1-[(3S)-1-benzylpyrrolidin-3-yl]-5-(2-methyl-1H-imidazol-4-yl)-4-phenyl-1H-imidazole
N-cyclopentyl-6-methyl-5-[5-(1-methylcyclopropyl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine-2-carboxamide
(3S,4R)-N-(4-chloro-2-methylphenyl)-3-methanesulfonamido-4-(propan-2-yl)pyrrolidine-1-carboxamide
(3R)-3,4,4-trimethyl-1-(pyridin-4-yl)pyrrolidin-3-ol
6-{3-[(2-fluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}pyridine-3-carbonitrile
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}but-3-enamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(1H-indol-3-yl)acetamide
N-[5-(4-fluorophenyl)-1,3,4-thiadiazol-2-yl]-2-(pyridin-3-yl)piperidine-1-carboxamide
5-{1-[3-(1H-imidazol-1-yl)propyl]-1H-imidazol-2-yl}-2-phenyl-1,3-thiazole
5-fluoro-N-(pyrimidin-4-ylmethyl)quinazolin-4-amine
7,7-dimethyl-2-[3-(pyrrolidin-1-yl)propyl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(2-methoxyethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-hydroxy-1-[(3-methoxyphenyl)methyl]-3-({[2-(1H-1,2,3-triazol-1-yl)ethyl]amino}methyl)piperidin-2-one
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-1-(oxan-4-yl)piperidine-3-carboxamide
5-(4-{[methyl(oxan-2-ylmethyl)amino]methyl}phenoxymethyl)furan-2-carboxylic acid
5-methanesulfonyl-2-(2-methyl-1,3-thiazol-4-yl)-4-(piperidin-3-yl)pyrimidine
3-{1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidin-4-yl}-1-(4-phenylpiperazin-1-yl)propan-1-one
N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-2-(methylsulfanyl)acetamide
1-[(2-methyl-1H-imidazol-4-yl)methyl]-3-(3-methylthiophene-2-carbonyl)piperidine
N,N,4-trimethyl-5-(5,6,7,8-tetrahydro-1,6-naphthyridine-6-carbonyl)pyrimidin-2-amine
N-(cyclopropylmethyl)-4-oxo-3,4-dihydroquinazoline-2-carboxamide
2-(3-methoxypropyl)-8-[(3-methylphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-[(3-methoxyphenyl)methyl]-3-(1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperidin-3-yl)propanamide
4-(4H-1,2,4-triazol-4-yl)-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]benzamide
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-4-(pyridin-2-yl)pyrimidin-2-amine
1-methyl-4-(2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carbonyl)piperazine-2-carboxylic acid
7-(2-methylphenyl)-4-(pyridine-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-cyclohexyl-3-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidine-1-carboxamide
N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
1-(1,3-thiazol-2-yl)-4-{2,5,7-trimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}piperazine
2-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-2-azaspiro[4.5]decan-3-one
1,3,6-trimethyl-N-[1-(3,4,5-trimethoxyphenyl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-{5-[1-(thiophene-2-sulfonyl)pyrrolidin-2-yl]-1,2,4-oxadiazol-3-yl}pyridine
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-1-methyl-5-oxopyrrolidine-3-carboxamide
8-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
7-(2-methoxyacetamido)-1-methyl-2-phenyl-N-{spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-5-ylmethyl}-1H-1,3-benzodiazole-5-carboxamide
N-(3-chloro-4-ethoxyphenyl)-3-(2-methylpiperidin-1-yl)azetidine-1-carboxamide
2-{4-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1-(3-phenylpropyl)piperazin-2-yl}ethan-1-ol
N-({7-[(2E)-3-(2,5-difluorophenyl)prop-2-enoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)oxane-4-carboxamide
{4-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-1,4-oxazepan-6-yl}methanol
N-[3-(2-chlorophenoxy)propyl]-N,2,4-trimethylpyrimidine-5-carboxamide
1-(3-fluoro-5-methylphenyl)-3-[(1R,2R)-2-hydroxycyclohexyl]-3-propylurea
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-5-(3-fluorophenoxymethyl)-N-methyl-1H-pyrazole-3-carboxamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-methylacetamide
(1S,5R)-6-(3-chloro-5-fluorobenzoyl)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonane
2-[2-(2H-1,3-benzodioxol-4-ylmethyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]-6-methylpyridine
1-(2,1,3-benzoxadiazol-4-ylmethyl)-4-phenoxypiperidine-4-carboxylic acid
ethyl 3-[(2,4-difluorophenyl)methyl]-1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]piperidine-3-carboxylate