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5-butanoyl-N-(3-phenylpropyl)-1-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[(3R,4S)-1-(6-tert-butyl-2-oxo-2,3-dihydropyrimidine-4-carbonyl)-4-propylpyrrolidin-3-yl]acetamide
1-(cyclohexylmethyl)-5-[(furan-2-ylmethyl)(methyl)amino]-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(3R,5S)-N-[2-(dimethylamino)ethyl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
(3S)-1-[5-(4,4-difluoropiperidine-1-carbonyl)-1-methyl-1H-1,3-benzodiazol-2-yl]pyrrolidin-3-ol
2-{[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1H-1,3-benzodiazole
3-(2-methoxyethyl)-1-[2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]piperidine-3-carboxylic acid
N-[2-(benzyloxy)ethyl]-6-ethyl-2-oxo-1,2-dihydropyridine-4-carboxamide
1-(3,5-difluorophenyl)-3-{1-[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]ethyl}urea
2-ethoxy-N-[(2R,3R)-2-(pyridin-3-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
N-[(1-hydroxycyclohexyl)methyl]-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
N-[(3R,4S)-1-(2-aminopyrimidin-4-yl)-4-(propan-2-yl)pyrrolidin-3-yl]-4-cyanooxane-4-carboxamide
(1S,5R)-6-(2-methoxyethyl)-3-[(5-methyl-1,2-oxazol-4-yl)sulfonyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(2-benzylmorpholine-4-carbonyl)-6-phenyl-1,2-dihydropyridin-2-one
2-[(1S,5R)-3-(2-amino-6-ethyl-5-methylpyrimidin-4-yl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-(3-hydroxy-3-phenylpropyl)-N-methylacetamide
1-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-(furan-2-ylmethyl)-2-(6-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)-N-propylacetamide
11-{[(3,4-difluorophenyl)methyl]amino}-4-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-[cyclohexyl(methyl)amino]-3-{3-[({2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}amino)methyl]phenoxy}propan-2-ol
N-[3-(cyclohexyloxy)propyl]-1H-1,2,3-triazole-5-carboxamide
N-[5-carbamoyl-2-(3-methylpiperidin-1-yl)phenyl]-1-propyl-1H-pyrazole-5-carboxamide
2-[4-(2,1,3-benzoxadiazol-4-ylmethyl)-1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-2-yl]ethan-1-ol
N-(cyclohexylmethyl)-4-[(furan-2-ylmethyl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
5-fluoro-3-methyl-2-{[4-(pyridin-4-yl)piperidin-1-yl]methyl}-1H-indole
2-methyl-3-[3-(3-methylphenoxymethyl)piperidine-1-carbonyl]-4,5,6,7-tetrahydro-1H-indol-4-one
4-methyl-1-{[2-(trifluoromethyl)phenyl]methyl}-1,4-diazepan-5-one
2-(2-acetylphenyl)-N-(propan-2-yl)benzamide
2-[(2-amino-5-butyl-6-methylpyrimidin-4-yl)amino]-1-(pyrrolidin-1-yl)ethan-1-one
N-{2-[4-(2-fluorophenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]ethyl}-4-methylbenzamide
1-cyclohexyl-4-{5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
[(5-ethylpyridin-2-yl)methyl](methyl){[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amine
2-[4-methyl-2-(methylamino)-1,3-thiazole-5-carbonyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one
1-[2-(benzyloxy)ethyl]-1,2,3,4,5,6,7,8-octahydroquinolin-2-one
N-{2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}-2-[4-(2-oxoimidazolidin-1-yl)phenyl]acetamide
5,8-dimethyl-2-({[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]amino}methyl)quinolin-4-ol
1-[6-hydroxy-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]-3-(1-methyl-1H-pyrrol-2-yl)propan-1-one
3-(5-acetyl-2-methoxyphenyl)-1-methyl-1-[1-(4-methylpyridin-2-yl)propan-2-yl]urea
N,N,2-trimethyl-7-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}acetamide
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
4-({[3-(1H-1,2,3-benzotriazol-1-yl)propyl]carbamoyl}amino)-N-ethyl-3-methylbenzamide
1-(3-{4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}-3-oxopropyl)-1,2-dihydropyridin-2-one
1-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepan-4-yl]-2-(2,4,7-trimethyl-1H-indol-3-yl)ethan-1-one
N-methyl-4-(pyridin-3-yl)-N-{[3-(trifluoromethyl)phenyl]methyl}pyrimidin-2-amine
4-{1-[4-(5-chloropyrimidin-2-yl)piperazin-1-yl]-2-methylpropan-2-yl}morpholine
{9-[(3-methyl-1,2-oxazol-5-yl)methyl]-3-(1H-pyrrole-3-carbonyl)-3,9-diazaspiro[5.5]undecan-1-yl}methanol
3-{1-[(5-acetylthiophen-3-yl)methyl]piperidin-3-yl}-1-(4-methylpiperazin-1-yl)propan-1-one
3,4,5-trimethoxy-N-[(5-{[(3-methylphenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl]benzamide
N-{[4-amino-6-(dimethylamino)-1,3,5-triazin-2-yl]methyl}-6-methoxy-3-methyl-1-benzofuran-2-carboxamide