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N'-(2,5-dimethoxyphenyl)-N-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]propanediamide
1-{[4-methyl-5-(1-methylpiperidin-4-yl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-4-ol
2-{3-[2-(2-methylpropyl)-3-oxo-2,8-diazaspiro[4.5]decane-8-carbonyl]piperidin-1-yl}acetamide
(3aR,6aR)-2-(cyclobutylmethyl)-5-(2,4-difluorobenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(4-methoxyphenyl)-2,2-dimethyl-4-(1H-pyrrole-2-carbonyl)piperazine
(1S,4S)-2-{5-[2-(methylsulfanyl)phenoxymethyl]-1,2-oxazole-3-carbonyl}-2-azabicyclo[2.2.1]heptane
6-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]imidazo[2,1-b][1,3]thiazole-5-carboxamide
1-(4-{1-[(3-methylphenyl)methyl]-1H-pyrazol-4-yl}-1,2,3,6-tetrahydropyridin-1-yl)butan-2-ol
9-methoxy-7-[4-(methylsulfanyl)phenyl]-4-(thiophen-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-amino-6-{4-[(1-propyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}pyrimidin-4-ol
3-phenyl-1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}pyrrolidin-3-ol
N-cyclopentyl-3-[5-(pyrimidin-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanamide
ethyl 4-[(2-chlorophenyl)methyl]-1-(3-phenylprop-2-ynoyl)piperidine-4-carboxylate
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-1-[3-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(2-methoxy-5-methylbenzoyl)piperidin-3-ol
2-[2-(2H-1,3-benzodioxol-5-yloxy)acetyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
3-[3-(dimethylamino)propyl]-8-[(1-methyl-1H-indol-3-yl)methyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-methyl-5-{1-[(1-methyl-1H-imidazol-2-yl)methyl]pyrrolidin-2-yl}-N-(1H-pyrazol-5-ylmethyl)thiophene-2-carboxamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-1-(furan-2-ylmethyl)piperidine-4-carboxamide
2-(5-acetylthiophen-3-yl)-1-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]ethan-1-one
9-{[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(2-aminoethyl)-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}quinazolin-4-amine
6-(4-{[4-(1H-imidazol-1-yl)phenyl]methyl}piperazin-1-yl)pyrazine-2-carboxamide
2-(2-methoxyethyl)-9-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-2,9-diazaspiro[5.5]undecan-3-one
1-ethyl-2-{1-[3-(4H-1,2,4-triazol-4-yl)phenyl]-1H-imidazol-2-yl}-1H-1,3-benzodiazole
N-methyl-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
(3aS,6aS)-2-cycloheptyl-5-(3-methoxypropanoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-[4-(pyrrolidine-1-carbonyl)pyridin-2-yl]pyridin-3-amine
3-[2-(2,6-difluorophenyl)ethyl]-1-(2-ethoxyethyl)piperidine
1-[1-(2-chloro-6-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(pyridin-2-yl)propan-1-one
2-(3-butyl-4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-methyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]acetamide
7-(5-methylthiophen-2-yl)-4-(thiophen-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-{4-[4-(1,2-oxazolidine-2-carbonyl)piperidin-1-yl]piperidin-1-yl}-1,3-benzoxazole
N-{[2-(dimethylamino)-7-methoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)propanamide
3-[5-(2-methylbutan-2-yl)-1,3,4-thiadiazol-2-yl]-1-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]urea
(2S,4R)-N,N-diethyl-1-methyl-4-[3-(pyridin-4-yl)propanamido]pyrrolidine-2-carboxamide
4-{2-[(2-chlorophenyl)methyl]morpholin-4-yl}-N,N-dimethyl-4-oxobutanamide
1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-4-phenylazepane
5-ethyl-2-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]pyrimidin-4-amine
3-[(3R,4S)-1-(1H-indazole-3-carbonyl)-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
2-ethyl-4-methyl-N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)-1,3-oxazole-5-carboxamide
(3S,4R)-3-benzyl-4-methyl-1-(6-phenylpyridazin-3-yl)piperidin-4-ol
2-{1-[(4-phenyl-1,3-thiazol-2-yl)methyl]piperidin-3-yl}-1,2,3,4-tetrahydroisoquinoline
2-(2-ethylphenyl)-4,6-dimethoxy-1,3,5-triazine
N-[3-(furan-2-yl)-1H-1,2,4-triazol-5-yl]-4-(6-oxo-1,6-dihydropyridazin-4-yl)piperazine-1-carboxamide
2-[(furan-2-ylmethyl)(methyl)amino]-2-{4-[(morpholine-4-carbonyl)amino]phenyl}acetic acid
methyl N-[2-(3-methyl-3-phenylpiperidin-1-yl)-2-oxoethyl]carbamate
1-methyl-3-(thiomorpholine-4-carbonyl)-N-{[4-(trifluoromethyl)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-chloro-4-({[3-(1H-imidazol-1-yl)propyl](pyridin-4-ylmethyl)amino}methyl)-6-methoxyphenol
3-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]-2-methyl-4,5,6,7-tetrahydro-1-benzofuran-4-one