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2-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}phenol
(3R,4R)-1-{2-[cyclohexyl(methyl)amino]pyridine-3-carbonyl}-4-ethylpiperidine-3,4-diol
N-(6-phenoxypyridin-3-yl)-1-(1,3-thiazol-2-ylmethyl)piperidine-4-carboxamide
N-[2-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)ethyl]-4-(1H-pyrazol-3-yl)benzamide
9-(3-methylthiophene-2-carbonyl)-2-[2-(pyridin-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[(4aR,8aR)-4a-hydroxy-7-[(4-methylnaphthalen-1-yl)methyl]-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
(2S,4S)-N-ethyl-1-(1H-imidazol-4-ylmethyl)-4-[2-(thiophen-2-yl)acetamido]pyrrolidine-2-carboxamide
3-{1-[(3-hydroxy-4-methoxyphenyl)methyl]piperidin-4-yl}-1-(morpholin-4-yl)propan-1-one
(1S,4S)-5-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-2-(2-methoxy-5-phenylphenyl)-2,5-diazabicyclo[2.2.1]heptan-3-one
3-(4-phenyl-1H-pyrazol-5-yl)-1-(2-propyl-1,3-thiazole-4-carbonyl)piperidine
4-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}morpholine-2-carboxylic acid
1-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-4-(pyrrolidin-3-yl)piperazine
N-[(4-fluorophenyl)methyl]-N-(3-methoxypropyl)-2,3-dimethyl-1H-indole-7-carboxamide
5-cyclopropanecarbonyl-1'-(furan-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
[(1-ethyl-1H-imidazol-2-yl)methyl](methyl){[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}amine
1-(1-benzoylpiperidin-3-yl)-4-[3-(trifluoromethyl)phenyl]piperazine
3-(4-methoxy-2-methylbenzoyl)-1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidine
N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1-(propan-2-yl)piperidine-4-carboxamide
N-[2-(2-chlorophenyl)-1-{1-[(3,4-dimethoxyphenyl)methyl]piperidin-4-yl}ethyl]-N-methylfuran-2-carboxamide
N-(3-fluoro-5-methylphenyl)-3-[(methylsulfanyl)methyl]piperidine-1-carboxamide
2-{2-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}pyridine
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(1,3-thiazol-4-ylmethyl)pyrrolidin-3-yl]-4-methyl-1,3-thiazole-5-carboxamide
3-[(3S,7S,8aS)-3-[(2S)-butan-2-yl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,6-dichlorophenyl)urea
5-{[(1-cyclopropanecarbonylpiperidin-4-yl)formamido]methyl}thiophene-2-carboxylic acid
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
1-(3-methylfuran-2-carbonyl)-4-(2-methylpropyl)-1,4-diazepan-5-one
N-methyl-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}-1,3-benzothiazole-2-carboxamide
5-methyl-4-(1-methyl-1H-1,2,4-triazol-5-yl)-N-[2-(2-methyl-1H-indol-1-yl)ethyl]pyrimidin-2-amine
1-[3-(3-methoxyphenoxy)azetidin-1-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
4-[4-(2,6-dimethoxyphenyl)phenyl]-1,3-thiazol-2-amine
4-{1-[1-(oxolan-2-ylmethyl)piperidin-4-yl]-1H-imidazol-2-yl}pyridine
3,7-dimethyl-11-{[4-(pyridin-2-yl)phenyl]methyl}-3,7,11-triazaspiro[5.6]dodecane
(1S,5R)-3-(1H-indole-5-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(3-acetyl-1H-indol-1-yl)-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]butanamide
4-methyl-2-[1-(4-methyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]-1H-1,3-benzodiazole
2-[2-(1H-imidazol-4-yl)ethyl]-9-[2-(3-methylphenyl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
8-[(2-hydroxyphenyl)methyl]-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(3R,4R)-1-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
1-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-N-(4-fluorophenyl)piperazine-2-carboxamide
N-cyclohexyl-6-(2-methoxyphenyl)-N-(prop-2-yn-1-yl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-[4-(ethylsulfanyl)phenyl]-1,3-dimethyl-2,4-dioxo-1,3,8-triazaspiro[4.5]decane-8-carboxamide
N-(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-3-azaspiro[5.5]undecan-9-amine
1-(4-methoxyphenyl)-4-{1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}piperazine
ethyl 4-(2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamido)piperidine-1-carboxylate
1-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)piperidin-3-ol
3-[4-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)piperazin-1-yl]-1,2-benzothiazole
[3-(3-methoxypropyl)-1-[4-methyl-6-(methylamino)pyrimidin-2-yl]piperidin-3-yl]methanol
2-[4-(4-{[(4-phenyl-1,3-thiazol-5-yl)methyl]amino}piperidin-1-yl)phenyl]-N-(pyridin-2-ylmethyl)acetamide
[(1S,3S,3aS,6aR)-5-methyl-1-phenyl-3-[3-(1H-pyrazol-1-yl)phenyl]-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
N-{[6-(dimethylamino)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-3-(4-methylphenyl)-N-(oxolan-2-ylmethyl)propanamide