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5-fluoro-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}quinazolin-4-amine
N-methyl-4-(2-methyl-1H-imidazol-1-yl)-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]butanamide
2-[2-(morpholin-4-yl)-2-oxoethyl]-7-propyl-2,7-diazaspiro[4.5]decan-6-one
2-(5-methylpyridine-3-carbonyl)-N-(oxolan-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
N-(3-hydroxy-3-phenylpropyl)-N-methyl-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
4-cyclopentyl-N-[1-(3-methylpyridin-2-yl)ethyl]pyrimidin-2-amine
N-(2,1,3-benzoxadiazol-5-ylmethyl)-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
1-[4-({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)-1,4-diazepan-1-yl]ethan-1-one
{[1-benzyl-2-(2-methoxyethanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)(2-phenylethyl)amine
4-(2-{9-oxa-2-azaspiro[5.5]undecan-2-yl}-2-oxoethyl)-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
2-(furan-2-yl)-2-oxo-N-[1-(pyrazin-2-yl)piperidin-3-yl]acetamide
2,3,5-trimethyl-N-[2-(pyrrolidine-1-sulfonyl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
2-(4-benzyl-2-oxopyrrolidin-1-yl)-N-ethyl-N-[(2-fluorophenyl)methyl]acetamide
5-(2-methoxyphenoxymethyl)-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,2-oxazole-3-carboxamide
4-[3-(2-methoxybenzoyl)piperidin-1-yl]-2-methyl-6-(1H-pyrazol-1-yl)pyrimidine
2-[1-(1,2,3,4-tetrahydronaphthalen-2-yl)-1H-imidazol-2-yl]pyridine
(2S)-S-(3-{2-azaspiro[4.4]nonane-2-carbonyl}phenyl)-2,3-dihydroxypropane-1-sulfonamido
[3-(2-phenoxyethyl)-1-(quinolin-2-yl)piperidin-3-yl]methanol
dimethyl(2-{2-[1-(5-propyl-1,3,4-thiadiazol-2-yl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)amine
3-(2,5-dioxoimidazolidin-4-yl)-N-{2-[(4-fluorophenyl)formamido]ethyl}propanamide
(3S)-1-{[4-(1H-imidazol-1-yl)phenyl]methyl}-N,N-dimethylazepan-3-amine
4-(2-methoxyphenoxy)-1-[(2S)-oxolane-2-carbonyl]piperidine-4-carboxylic acid
3-[4-(4-ethoxyphenyl)-1H-imidazol-2-yl]-2-methoxypyridine
3-chloro-4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}phenol
N-[4-chloro-3-(1,1-dioxo-1λ6-thiomorpholine-4-carbonyl)phenyl]acetamide
N,2-dimethyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-1H-1,3-benzodiazole-5-carboxamide
N-[(5-methoxy-1H-indol-2-yl)methyl]-6-oxo-1,6-dihydropyridine-3-carboxamide
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-3-[(2-methylprop-2-en-1-yl)oxy]benzamide
2-{[3-(3-chlorobenzoyl)piperidin-1-yl]methyl}-1,3-benzothiazole
4-(hydroxymethyl)-1-{[3-(pyridin-2-yl)phenyl]methyl}piperidin-4-ol
N-benzyl-N-cyclopentyl-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
1-{1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-2-{[1,2,4]triazolo[4,3-b]pyridazin-6-yloxy}ethan-1-one
2-butoxy-1-[(2R,3S,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
7-fluoro-1-(2-methylpropyl)-3-({[3-(morpholin-4-yl)propyl]amino}methyl)-1,2-dihydroquinolin-2-one
6-methyl-3-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
4-acetamido-N-[(2-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)benzamide
N-ethyl-2-[4-({3-methanesulfonylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)morpholin-3-yl]acetamide
2-methyl-4-{3-[3-(3-methylphenoxy)azetidine-1-carbonyl]phenyl}butan-2-ol
2-[4-(hydroxymethyl)phenyl]-1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}-N-(4-methylphenyl)piperidine-1-carboxamide
N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-N-methyl-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
N-[(3S,4R)-4-(4-methylphenyl)-1-[(6-methylpyridin-2-yl)methyl]pyrrolidin-3-yl]cyclopropanecarboxamide
methyl 6-(2-{[3-(2H-1,3-benzodioxol-5-yl)propanamido]methyl}-2,3-dihydro-1-benzofuran-7-yl)pyridine-3-carboxylate
8-[(2,2-difluoro-2H-1,3-benzodioxol-5-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
7-[2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}butane-1-sulfonamide
2-(6-{pyrazolo[1,5-a]pyridin-7-yl}pyridin-3-yl)acetic acid
1-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]-3-(pyridin-3-yl)propan-1-one
N6-cyclopropyl-N4-methyl-N4-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)pyrimidine-2,4,6-triamine
(1S,5R)-1,3,3-trimethyl-6-{[6-(4-methyl-1,4-diazepane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}-6-azabicyclo[3.2.1]octane