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5-ethyl-2-methyl-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}pyrimidin-4-amine
[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]({[2-(propylsulfanyl)pyrimidin-5-yl]methyl})amine
4-(1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}azetidin-3-yl)pyridine
(2S,4R)-4-amino-N-methyl-1-[6-(2-methylbutan-2-yl)-1-benzothiophene-3-carbonyl]pyrrolidine-2-carboxamide
2-[3-({[2-(pyrrolidin-1-yl)ethyl]carbamoyl}amino)phenyl]acetamide
1-{2-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyrimidin-4-yl}piperidin-4-ol
(3S,4S)-1-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}-4-(propan-2-yloxy)pyrrolidin-3-ol
3-[({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}amino)methyl]-1-[(4-fluorophenyl)methyl]-3-hydroxypiperidin-2-one
N-(2,3-dihydro-1H-inden-2-yl)-3-(2-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidin-2-yl)propanamide
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]acetamide
5-chloro-4,6-dimethyl-3-[3-(thiophene-2-carbonyl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
N-[2-({4-[(dimethylamino)methyl]phenyl}formamido)ethyl]acetamide
4-[(4-hydroxy-5-methoxypyridin-2-yl)methyl]-5-methyl-1-(4-methylphenyl)piperazin-2-one
4-{[1-cyclohexyl-5-(oxolan-3-yl)-1H-1,2,4-triazol-3-yl]methyl}-1-methylpiperidine
{4-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]morpholin-2-yl}methanamine
2-({1-[(1-methyl-1H-imidazol-5-yl)methyl]piperidin-3-yl}methyl)-1H-1,3-benzodiazole
N-(1-benzothiophen-2-ylmethyl)-5-[(3-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
1-[3-(cyclopentyloxy)phenyl]-3-(1H-pyrazol-3-ylmethyl)urea
1-{2-[2-(3-methoxypropyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-(2,5-dimethylphenyl)-N'-[(3,4,5-trimethoxyphenyl)methyl]propanediamide
7-methyl-4-{2-oxo-2-[3-(propoxymethyl)pyrrolidin-1-yl]ethyl}-3,4-dihydro-2H-1,4-benzothiazin-3-one
N-(propan-2-yl)-6-(quinolin-8-yl)pyrimidin-4-amine
ethyl 2-({[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]carbamoyl}amino)propanoate
(5S,9aS,9bS)-5-[(E)-2-(4-hydroxy-3-methoxyphenyl)ethenyl]-2-[(2-methylphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-methoxy-5-methyl-N-[2-(3-phenylpyrrolidin-1-yl)ethyl]thiophene-2-carboxamide
1-[2-(piperazin-1-yl)ethyl]-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}-1H-1,2,3-triazole-4-carboxamide
4-chloro-3-methyl-5-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}-1H-pyrazole
9-(3-hydroxypyridine-2-carbonyl)-2-[3-(1H-imidazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-1-[(3,4-dimethoxyphenyl)methyl]-N5-[2-(dimethylamino)ethyl]piperidine-3,5-dicarboxamide
2-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]pyrimidin-4-amine
methyl (1R,3S,3aR,6aS)-3-(4-fluoro-2-methylphenyl)-1,5-dimethyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
1-[5-({[2-(3-chlorophenyl)ethyl]amino}methyl)-2-methoxyphenoxy]-3-(diethylamino)propan-2-ol
2-(5-{[4-(1H-pyrrole-2-carbonyl)piperazin-1-yl]methyl}furan-2-yl)benzonitrile
2-[(1S,5R)-6-[4-(difluoromethoxy)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
7-(2-methoxyethyl)-2-({4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-2,7-diazaspiro[4.5]decan-6-one
2-methoxy-1-{4-[2-(phenoxymethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}ethan-1-one
N-methyl-2-(3-oxo-3,4-dihydro-2H-1,4-benzothiazin-4-yl)-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)acetamide
methyl 3-(2-methylbutanamido)-5-{[(5-methylthiophen-2-yl)methyl]amino}-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-1-(furan-2-ylmethyl)piperidine
4-{1-[4-(2,3-dichlorophenyl)-1H-1,2,3-triazol-1-yl]propyl}pyridine
2-[2-methyl-3-({[1-(2-propoxyphenyl)ethyl]amino}methyl)-1H-indol-1-yl]acetamide
1-(4-fluorophenyl)-N-{2-hydroxy-2-[2-(trifluoromethyl)phenyl]ethyl}cyclopropane-1-carboxamide
(1S,4S)-2-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-2-azabicyclo[2.2.1]heptane
4-(2,5-dimethoxyphenyl)-3-(1-methoxyethyl)-4H-1,2,4-triazole
2-(3-oxo-2,3-dihydro-1H-indazol-2-yl)-N-[(4-sulfamoylphenyl)methyl]acetamide
5-(propan-2-yl)-N-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methylthiophene-2-carboxamide
3-(4-chlorobenzoyl)-1-cyclohexylpiperidine
6-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carbonyl]-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-4-({[4-(benzyloxy)phenyl]methyl}amino)-1-(propan-2-yl)pyrrolidine-2-carboxamide