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4-{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-2,2-dimethylmorpholine
N-[2-(dimethylamino)-2-(furan-2-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
2-{4-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-4-methoxyphenyl]phenyl}-N-methylacetamide
ethyl 6-[9-oxo-8-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-2-yl]pyridine-3-carboxylate
1-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
2-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-N,N-dimethylacetamide
3-(2-{4-[(2-fluorophenyl)methyl]piperidin-1-yl}-2-oxoethyl)-2,3-dihydro-1H-isoindol-1-one
(1R,2R,6S,7S)-4-{2-[2-(3-methoxyphenyl)ethyl]benzoyl}-10-oxa-4-azatricyclo[5.2.1.02,6]decane
3-ethyl-6-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]-3H-imidazo[4,5-b]pyridin-2-amine
N'-(2,4-dimethoxyphenyl)-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}propanediamide
(3S,4S)-1-(carboxymethyl)-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
2-(3-fluorophenyl)-5-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyridine
4-{2-[4-(2-methylpyrimidin-4-yl)piperidin-1-yl]-2-oxoethyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
4,6-dimethyl-2-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}pyridine-3-carbonitrile
1-[(4-methanesulfonylphenyl)methyl]-N,N-dimethylazepan-4-amine
2-(3,5-difluorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidin-1-yl]ethan-1-one
3-[(4-fluorophenyl)formamido]-N-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}propanamide
2-amino-4-{[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]amino}quinazoline-6-carboxylic acid
N-(2,1,3-benzothiadiazol-5-ylmethyl)-5-propylpyrazolo[1,5-a]pyrimidin-7-amine
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-4-(piperidin-3-yl)benzamide
1-[5-(2-chloro-3-methylbenzoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl]pyrrolidine
3-(1-{[1-(thiophene-3-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-1-ol
1-{1-[(2,6-difluorophenyl)methyl]piperidin-3-yl}-4-(2-fluorophenyl)piperazine
N-methyl-4-oxo-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
3-methyl-6-(5-{1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazol-4-yl}-1,2,4-oxadiazol-3-yl)pyridazine
3-(azetidine-1-carbonyl)-N-(2-methoxyethyl)-N-(thiophen-3-ylmethyl)benzene-1-sulfonamide
5-chloro-3-[1-(pyrazin-2-yl)propan-2-yl]-3,4-dihydroquinazolin-4-one
N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-N-(propan-2-yl)-2H-1,3-benzodioxole-5-carboxamide
4-(3-phenoxyphenyl)-3-(1H-1,2,3,4-tetrazol-5-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-cyclopropyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-2,3-dihydro-1H-inden-2-amine
3-methyl-1-(1-{2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetyl}piperidin-3-yl)butan-1-one
1-[(4-fluorophenyl)methyl]-3-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)urea
(1S,5R)-6-methyl-3-{1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[(4-fluorophenyl)methyl]-5-(1H-imidazole-5-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-[2-(1H-imidazol-2-yl)benzoyl]-4-(thiophen-2-ylmethyl)-1,4-diazepane
2-(2-{1-[4-(1H-imidazol-1-yl)benzoyl]piperidin-4-yl}-1H-imidazol-1-yl)acetamide
N-[1-(thiophen-2-ylmethyl)piperidin-3-yl]-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
N-(4-{[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)carbamoyl}phenyl)-2-methylfuran-3-carboxamide
2-{1-[(2-phenyl-1,3-oxazol-4-yl)methyl]pyrrolidin-3-yl}benzoic acid
N-[(2R,3R)-1'-[(2E)-3-(4-hydroxy-3-methoxyphenyl)prop-2-en-1-yl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
4-(2,6-dimethylpyridin-3-yl)-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]pyrimidin-2-amine
2-[2-(4-methanesulfonylphenyl)phenyl]-5-methyl-1,3,4-oxadiazole
(4aR,7aS)-1-methyl-4-[3-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)propanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(1-{1-[(3,4-difluorophenyl)methyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)pyridine
1-(6-methyl-3-{[methyl(1,2-oxazol-5-ylmethyl)amino]methyl}quinolin-2-yl)piperidin-3-ol
(3aS,6aS)-1-(6,7-diethoxy-3-methyl-1-benzofuran-2-carbonyl)-octahydropyrrolo[2,3-c]pyrrole
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carboxamide
3-(1-methyl-1H-imidazol-4-yl)-5-(3-phenyl-1H-pyrazol-4-yl)-1,2,4-oxadiazole
4-[2-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)ethyl]morpholine
5-methoxy-4-oxo-N-[1-(5,6,7,8-tetrahydronaphthalen-2-yl)ethyl]-1,4-dihydropyridine-2-carboxamide