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N-[(3-ethoxyphenyl)methyl]-3-hydroxy-N-(prop-2-en-1-yl)pyridine-2-carboxamide
3-(azepane-1-carbonyl)-1-ethyl-N-[2-(2-methoxyphenyl)ethyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-(pyridin-3-ylmethyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
2-(2-chloro-4-fluorophenyl)pyridine-3-carbonitrile
4-(2-methoxybenzoyl)-9-[(1-methylpiperidin-3-yl)methoxy]-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(propan-2-yl)-1-[(1s,4s)-4-(5-phenoxyfuran-2-amido)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
2-{3-[2-(3-fluorophenyl)piperidin-1-yl]-3-oxopropyl}-2,3-dihydro-1H-isoindol-1-one
N-cyclopentyl-4-oxo-4-{4-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]piperazin-1-yl}butanamide
1-[(2S,4S)-1-(2,2-dimethylpropyl)-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carbonyl]azepane
1-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}azepan-2-one
2-cyclopropyl-9-(ethanesulfonyl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
1-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]ethan-1-one
8-(furan-3-ylmethyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-{1-oxaspiro[4.5]decan-3-yl}acetamide
N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
3-{2-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-2-oxoethyl}-1λ6-thiolane-1,1-dione
3-benzyl-1-(3-methoxypropyl)-8-(quinoxalin-5-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-(2-methoxypyridin-3-yl)-2,3-dihydro-1λ6-thiophene-1,1-dione
N-cyclobutyl-4-[(3-ethylpiperazin-1-yl)sulfonyl]benzamide
6-[3-(hydroxymethyl)phenyl]-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
2-{[4-(2-amino-6-methylpyrimidin-4-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]amino}acetic acid
N-({7-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)pyrazine-2-carboxamide
2-(3-fluorophenyl)-1-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]azepane
N-[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-[4-(morpholin-4-yl)-6-oxo-1,6-dihydropyridazin-1-yl]acetamide
(4aR,7aS)-1-(cyclopropylmethyl)-4-(3-methoxy-4-methylbenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[2-methyl-2-(piperidin-1-yl)propyl]-4-(2-phenoxyethyl)piperazine
3-{4-[(2-methylphenyl)sulfanyl]piperidine-1-carbonyl}pyridazine
N-[2-(1-methyl-1H-1,2,4-triazol-5-yl)ethyl]-3-(1-methylpiperidin-2-yl)propanamide
(2S,4R)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-(propan-2-yl)-4-({[4-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-[2-(4-methoxyphenyl)ethyl]acetamide
N-cycloheptyl-1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidine-4-carboxamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-methyl-4-phenylpyrimidine-5-carboxamide
N-{2-methoxy-4-[2-(1-phenylethyl)-1H-imidazol-1-yl]phenyl}acetamide
2-methoxy-N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}pyridine-3-carboxamide
5-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
2-[2-chloro-4-({methyl[1-(pyridin-3-yl)ethyl]amino}methyl)phenoxy]acetamide
N-[(2,5-difluorophenyl)methyl]-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
7-chloro-3-{[(2-methoxyethyl)amino]methyl}-1-(2-phenoxyethyl)-1,2-dihydroquinolin-2-one
N-(2-hydroxyethyl)-5-methyl-N-(propan-2-yl)-4-[(1,2,3,4-tetrahydronaphthalen-1-yl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
1-[(2-aminopyridin-3-yl)methyl]-4-(oxane-4-carbonyl)-1,4-diazepan-6-ol
N-benzyl-2-{1-[(3,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
3-[1-(1,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-{1-[(3-fluorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}urea
2-(3-hydroxyadamantan-1-yl)-1-{9-methyl-3,9-diazaspiro[5.6]dodecan-3-yl}ethan-1-one
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-(azocan-1-yl)-3-[4-({ethyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
2-(2,5-dioxoimidazolidin-4-yl)-N-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-5-[methyl(2-phenylethyl)amino]-2,3-dihydropyridazin-3-one
2-cyclohexyl-5-{[4-(1H-pyrrole-2-carbonyl)piperazin-1-yl]methyl}pyrimidine
3-[(dimethylamino)methyl]-3-(hydroxymethyl)-N-(3-phenoxyphenyl)piperidine-1-carboxamide
N,N-dimethyl-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}azepan-4-amine