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2-(4-methoxyphenyl)-N-[(3S,5S)-1-methyl-5-(morpholine-4-carbonyl)pyrrolidin-3-yl]acetamide
1-cyclopentyl-N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
3-[4-(methylsulfanyl)benzoyl]-1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidine
5-[3-(benzyloxy)azetidine-1-carbonyl]-1-ethylpiperidin-2-one
2-[(1S,5R)-3-(2-ethoxypyridine-3-carbonyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-5-(methoxymethyl)furan-2-carboxamide
1-[3-(2-methoxybenzoyl)piperidin-1-yl]-2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethan-1-one
3-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidine-1-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
4-({3-oxo-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-4-yl}methyl)benzene-1-sulfonamide
N-[(2-amino-1,3-thiazol-4-yl)methyl]-6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
3-cyclopropyl-N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-1H-pyrazole-5-carboxamide
4-(cyclohex-3-en-1-yl)-1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-1H-1,2,3-triazole
1-{1-[4-(furan-2-yl)phenyl]piperidin-4-yl}piperidin-4-amine
N-[1-methyl-4-(pyridin-3-yloxy)-1H-indazol-3-yl]-1,1-dioxo-1λ6-thiolane-3-carboxamide
2-[3-oxo-9-(quinolin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-2-yl]acetamide
(4aS,8aS)-2-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-decahydroisoquinolin-4a-ol
(1S,5R)-3-(2-hydroxy-3-methylbenzoyl)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[(4-methylpiperazin-1-yl)sulfonyl]-5-phenyl-N-[2-(pyridin-2-yl)ethyl]benzamide
ethyl 3-(2-methoxyethyl)-1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidine-3-carboxylate
4-{[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]methyl}benzonitrile
3-(3,4-dimethoxyphenyl)-N-(3-methoxypropyl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}[(4-phenyl-1,3-thiazol-2-yl)methyl]amine
2-amino-N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-3-ethyl-N-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
4-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}-5-(thiophen-2-yl)-1H-pyrazole
1-[(2-methoxyphenyl)methyl]-4-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperazine
{1-[5-(2-chloro-4-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]piperidin-2-yl}methanol
(3S,4S)-1-{[3,5-dimethyl-2-(1H-pyrazol-1-yl)phenyl]methyl}-4-methylpiperidine-3,4-diol
1-(2,3-difluoro-6-methoxybenzoyl)-4-(thiophen-2-ylmethyl)-1,4-diazepane
5-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidine-1-carbonyl}-3,4-dihydropyrimidin-4-one
[(3R,4S)-1-{[4-(cyclopentyloxy)phenyl]methyl}-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
2-(4-{[4-(5-methylpyridin-2-yl)piperidin-4-yl]methyl}piperazin-1-yl)benzonitrile
2-methyl-6-[(2S)-2-(morpholine-4-carbonyl)pyrrolidine-1-carbonyl]-1,3-benzoxazole
3-{1-[(1-ethyl-1H-pyrazol-3-yl)methyl]piperidin-3-yl}benzoic acid
8-fluoro-2-[({[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}amino)methyl]quinolin-4-ol
4-{2-[2-(furan-2-yl)pyrimidin-5-yl]-1H-imidazol-1-yl}benzene-1-sulfonamide
{5-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1H-1,3-benzodiazol-2-yl}methanol
8-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-1-(2-methoxyethyl)-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}(methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-2-(4-ethyl-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-1-yl)acetamide
3-[1-(5-ethyl-1,3,4-oxadiazol-2-yl)piperidin-4-yl]phenol
4-(cyclopropylmethyl)-3-(propan-2-yl)-1-[3-(4H-1,2,4-triazol-4-yl)propanoyl]-1,4-diazepan-5-one
3-[(2-fluorophenyl)formamido]-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}propanamide
3-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]-4,5,6,7-tetrahydro-1-benzofuran-4-one
3-(1-ethyl-1H-imidazol-2-yl)-1-(furan-2-carbonyl)piperidine
methyl 4-{[3-(2-methylpyrimidin-4-yl)phenyl]carbamoyl}piperazine-1-carboxylate
3-[(2-fluorophenyl)formamido]-N-methyl-N-[1-(pyrimidin-4-yl)ethyl]propanamide
N-cyclobutyl-3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propanamide
5-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidine-1-carbonyl]-1,2-dihydropyridin-2-one
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-1-[3-(morpholin-4-yl)propyl]-6-oxopiperidine-3-carboxamide
(2S,4S)-1-[(2-chlorophenyl)methyl]-N-ethyl-4-[(1-methylpiperidin-4-yl)amino]pyrrolidine-2-carboxamide