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N-(3-hydroxypropyl)-2-(1H-pyrazol-1-yl)-N-(thiophen-2-ylmethyl)benzamide
(2R,3R)-3-(1,2,3,6-tetrahydropyridin-1-yl)-1'-(thiophen-3-ylmethyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-(2,3-dihydro-1-benzofuran-7-yl)-2-[4-hydroxy-4-(pyridin-3-yl)piperidin-1-yl]acetic acid
1-[2-(2-methoxyphenyl)ethyl]-N,2,6-trimethyl-4-oxo-N-(thiophen-3-ylmethyl)-1,4-dihydropyridine-3-carboxamide
1-methyl-5-(1-methyl-1H-indazole-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-{1-[1-(3-hydroxypropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methoxy-2-phenylacetamide
(2S)-1-({3-[4-(3-methylpyrazin-2-yl)-6-oxo-1,6-dihydropyrimidin-2-yl]phenyl}methyl)pyrrolidine-2-carboxamide
N-[(2R,3R)-2-(2-methoxyethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]cyclobutanecarboxamide
6-(2-aminoethyl)-2-[4-({[1-(dimethyl-1,3-thiazol-4-yl)ethyl](methyl)amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
(2R)-1-{[7-methyl-2-(3-methylphenyl)quinolin-3-yl]methyl}pyrrolidine-2-carboxamide
N-(furan-3-ylmethyl)-N-methyl-1-[6-methyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-4-amine
N-{[4-(3-methylpiperidin-1-yl)phenyl]methyl}-1H-1,2,3-triazole-5-carboxamide
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-(2-methoxyethyl)pyrimidin-2-amine
ethyl 4-{[4-(2-methoxyphenyl)piperidine-1-carbonyl]amino}benzoate
8-[(8-methoxy-2H-chromen-3-yl)methyl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
5-{[4-(4-methoxybenzoyl)piperazin-1-yl]methyl}-2,1,3-benzothiadiazole
N-[4-(1H-pyrazol-1-yl)phenyl]-1-(pyridin-4-ylmethyl)piperidine-2-carboxamide
4-{1-[1-(thiophene-2-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}pyridine
1-{2-[1-(2-methylphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]ethyl}pyrrolidin-2-one
4-{[3-(pyrrolidine-1-carbonyl)-5-[3-(thiophen-3-yl)-1H-pyrazole-5-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-1-yl]methyl}pyridine
N-{4-[2-(dimethylamino)ethoxy]-1-(3-fluorophenyl)-1H-indazol-3-yl}-2-(methylsulfanyl)propanamide
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N,1-dimethyl-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
N-[4-(methylsulfanyl)phenyl]-6-[3-(2-oxopyrrolidin-1-yl)benzoyl]-6-azaspiro[2.5]octane-1-carboxamide
5-[4-(1-ethoxyethyl)phenyl]-1H-indazol-3-amine
1-[2-(4-methoxyphenyl)ethyl]-8-(1-methoxypropan-2-yl)-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-{3-[(3-fluorophenyl)amino]piperidine-1-carbonyl}-2-methoxyphenol
N-methyl-2-(3-methylpiperazine-1-carbonyl)-N-(2-phenylethyl)-2,3-dihydro-1H-inden-2-amine
3-(5-fluoro-2-methoxybenzoyl)-1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidine
7-(cyclobutylmethyl)-2-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetyl}-2,7-diazaspiro[4.5]decan-6-one
1,3-dimethyl 5-[(3-propylmorpholine-4-carbonyl)amino]benzene-1,3-dicarboxylate
1-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-yl]-4-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]butan-1-one
3-[(cyclobutylamino)methyl]-3-hydroxy-1-(2-phenylethyl)piperidin-2-one
N-[1-(3-phenylpropyl)piperidin-3-yl]piperidine-1-sulfonamide
ethyl 3-(3-{5-[(3-methylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamido)propanoate
5-(2-fluorophenyl)-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
4-methyl-1-({4-[methyl(phenyl)amino]phenyl}methyl)-1,4-diazepan-5-one
2,3-dimethoxy-N-({4-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)benzamide
N-methyl-2-(methylamino)-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-1,3-thiazole-4-carboxamide
9-(2,5-dimethylfuran-3-carbonyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
(3R)-1-(6-cyclopropylpyrimidin-4-yl)-3,4,4-trimethylpyrrolidin-3-ol
N-[(1-benzylpiperidin-4-yl)methyl]-N-methyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-(2,6-dimethylphenyl)-3-[2-(1H-pyrrol-1-yl)propanamido]benzamide
N-(1-cyclopentyl-4-methyl-1H-pyrazol-5-yl)-1,1-dioxo-1λ6-thiomorpholine-4-carboxamide
1-cyclopentanecarbonyl-N-methyl-N-(1,3-thiazol-2-ylmethyl)piperidine-4-carboxamide
2-(azocan-1-yl)-1-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}ethan-1-one
3-(pentan-2-yl)-8-[(1s,4s)-4-hydroxycyclohexanecarbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-2,8-dimethylquinoline-4-carboxamide
3-[(4aR,7aS)-6,6-dioxo-4-[(1-propyl-1H-imidazol-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
1-{2-[3-cyclopentyl-1-(4-fluorophenyl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-1-{4-[3-(pyrrolidin-1-yl)propyl]-1,4-diazepan-1-yl}ethan-1-one