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2-ethyl-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
7-[1-benzyl-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-2,3-dimethyl-1H-indole
2-[4-(6-cyclopropylpyrimidin-4-yl)-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl]ethan-1-ol
N-(cyclopropylmethyl)-1-[(4-fluorophenyl)methyl]-5-(2-methoxyacetamido)-N-(oxolan-2-ylmethyl)-1H-1,3-benzodiazole-7-carboxamide
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}({[3-methoxy-4-(propan-2-yloxy)phenyl]methyl})amine
N-[(4-methoxy-2,5-dimethylphenyl)methyl]-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-(1-methanesulfonylpiperidin-4-yl)-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-(2-hydroxyethyl)-6-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]-1H,2H,3H,4H,5H,6H,7H-pyrazolo[3,4-c]pyridin-3-one
1-(azepan-1-yl)-3-{4-chloro-2-[(4-methylpiperazin-1-yl)methyl]phenoxy}propan-2-ol
2-[(4-chlorophenyl)methyl]-8-(2,2-dimethylpropanoyl)-2,8-diazaspiro[4.5]decan-3-one
1-(2-oxo-2-{4-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}ethyl)-1,2,3,4-tetrahydroquinolin-2-one
4-(1-benzylpiperidin-4-yl)piperazine-2-carboxylic acid
1-(3-{3-[(4-methoxyphenyl)amino]piperidin-1-yl}-3-oxopropyl)pyrrolidin-2-one
1-(2-methyl-1,3-thiazole-4-carbonyl)-4-(3-phenylpropyl)-1,4-diazepane
1-[4-(4-methylpiperazin-1-yl)benzoyl]-4-(3-methylpyridin-4-yl)piperazine
1-{1-[(2-fluoro-4-methoxyphenyl)methyl]azetidin-3-yl}piperidine
2-[6-hydroxy-4-(quinoline-3-carbonyl)-1,4-diazepan-1-yl]acetic acid
N-(pentan-3-yl)-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
4-ethyl-3-{[1-(2-methyl-6-propylpyrimidin-4-yl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N,4,6-trimethyl-N-[3-(oxolan-2-yl)propyl]pyrimidin-2-amine
(3R,4S)-4-cyclopropyl-1-(quinoline-2-carbonyl)pyrrolidin-3-amine
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)acetamide
4-methoxy-1-[5-(2-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]piperidine
2-{[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]amino}pyridine-3-carboxamide
1-[1-(4-aminopyrimidin-2-yl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-3-carboxamide
3-({3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)pyridine
4-methyl-2-[2-(pyridin-2-yl)-1H-imidazol-1-yl]pyridine
N-(1-methoxypropan-2-yl)-1-oxo-2-[2-(piperidin-1-yl)ethyl]-2,3-dihydro-1H-isoindole-5-carboxamide
3-ethyl-8-[4-(1H-pyrrol-1-ylmethyl)benzoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-[5-(2,3-dihydro-1,4-benzodioxin-2-yl)-1,2,4-oxadiazol-3-yl]pyridine
4-(1H-imidazol-1-yl)-1-[(1S,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]butan-1-one
5-cyclopropyl-N,3-dimethyl-N-{[3-(trifluoromethyl)phenyl]methyl}-1H-pyrazole-4-carboxamide
4-[1-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)piperidin-3-yl]benzoic acid
2-[1-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)pyrrolidin-2-yl]-5-fluoro-1H-1,3-benzodiazole
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-2-oxo-1,2-dihydroquinoline-4-carboxamide
5-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]quinoxaline
1-ethyl-3,8-dimethyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
8-methyl-2-propyl-N-(thiophen-3-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxamide
2-methyl-3-{9-oxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}-4,5,6,7-tetrahydro-1H-indol-4-one
1-(2-methanesulfonylethyl)-5-(2-methylprop-1-en-1-yl)-4-phenyl-1H-imidazole
4-cyclobutyl-6-methyl-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}pyrimidin-2-amine
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[1-(3-methylpyridin-2-yl)propan-2-yl]-1H-pyrazole-3-carboxamide
N6-(3-methoxypropyl)-N5-methyl-N5-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
(1S,5R)-3-{dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl}-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
ethyl 1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-4-(2-phenoxyethyl)piperidine-4-carboxylate
3-(azepane-1-carbonyl)-1-methyl-N-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}-3-(1,2-oxazolidin-2-yl)propan-1-one
methyl 1-{2-hydroxy-3-[3-({methyl[(5-methylfuran-2-yl)methyl]amino}methyl)phenoxy]propyl}piperidine-4-carboxylate
5-ethyl-4-({3-[3-(3-methylpyridin-4-yl)phenyl]-1H-pyrazol-1-yl}methyl)furan-2-carboxamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one