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4-(4-cyclopropanecarbonyl-1,4-diazepan-1-yl)-N-[2-(methylsulfanyl)phenyl]-4-oxobutanamide
N-(5-chloro-2-methoxyphenyl)-3-[1-(1H-imidazole-4-carbonyl)piperidin-3-yl]propanamide
3-[({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]-1,2,4-oxadiazole-5-carboxamide
3-({[(2-amino-1,3-thiazol-4-yl)methyl]amino}methyl)-3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
N-(2-aminoethyl)-N'-(2-ethoxyphenyl)propanediamide
(4-{[2-(morpholin-4-yl)butyl]amino}quinazolin-2-yl)methanol
2-[(3-methoxyphenyl)methyl]-4-(3-methyl-1H-pyrazole-4-carbonyl)morpholine
(3R,4S)-4-{ethyl[(6-methoxypyridin-3-yl)methyl]amino}oxolan-3-ol
N'-(2,5-dimethylphenyl)-N-[3-(pyrrolidin-1-yl)propyl]propanediamide
N-cyclobutyl-5-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-amine
2-[3-(2-methoxypyridin-3-yl)-1H-indazol-1-yl]-N-(1-methyl-1H-pyrazol-5-yl)acetamide
(3aR,7aS)-2-(3-methanesulfonylbenzoyl)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindole
(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-(quinolin-4-ylmethyl)piperidin-3-ol
N-[2-(dimethylamino)ethyl]-5-(2-methoxyphenoxymethyl)-N-methyl-1H-pyrazole-3-carboxamide
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxamide
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]acetamide
N-cyclohexyl-4-[(1-hydroxypropan-2-yl)amino]piperidine-1-carboxamide
N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
5-[1-(2-cyclopentylacetyl)piperidin-4-yl]-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
3-(2,2-difluoro-2H-1,3-benzodioxol-4-yl)-1-(oxolan-2-ylmethyl)urea
1-[2-(1H-pyrazol-1-yl)ethyl]-4-[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]-1H-1,2,3-triazole
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-(2-methyl-1-benzofuran-5-carbonyl)piperidine
7,8-dimethyl-3-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]-3,4-dihydroquinazolin-4-one
8-chloro-N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]quinoline-2-carboxamide
N-cycloheptyl-1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}piperidine-4-carboxamide
N-methyl-3-(6-methylquinolin-3-yl)pyrazin-2-amine
methyl[(3-methylthiophen-2-yl)methyl]{[5-(propane-1-sulfonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}amine
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-(2-phenylethyl)-1,3-benzoxazole-5-carboxamide
3-[3-(azepane-1-carbonyl)phenyl]-1-[(3-methoxyphenyl)methyl]urea
3-(3-benzyl-1H-1,2,4-triazol-5-yl)-4,6-dimethyl-1,2-dihydropyridin-2-one
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-1-methylcyclopropane-1-carboxamide
4-(2-butyl-1H-imidazol-4-yl)-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-[2-(pyrazin-2-yl)ethyl]-2-[4-(trifluoromethyl)phenyl]-1,3-benzoxazole-5-carboxamide
1-(2-methoxyethyl)-4-{4-[3-(propan-2-yloxy)phenyl]-1H-imidazol-2-yl}pyrrolidin-2-one
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
3-(3,5-dimethylphenyl)-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]propanamide
(3S,4R)-4-(2-methoxyphenyl)-1-[2-(4-methyl-1H-pyrazol-1-yl)acetyl]pyrrolidine-3-carboxylic acid
2-{4-[2-(methylamino)pyridine-4-carbonyl]piperazin-1-yl}benzonitrile
2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-ylmethyl)pyridine-3-carboxylic acid
2-(2-{3-[3-(4-fluorophenyl)oxolan-3-yl]-1,2,4-oxadiazol-5-yl}ethyl)-1,2-oxazinane
4-(4,6-dimethylpyrimidin-2-yl)-N-(4-methanesulfonylphenyl)piperazine-1-carboxamide
N-{[3-(cycloheptyloxy)-4-methoxyphenyl]methyl}-N-cyclopropyl-2-(dimethyl-1,2-oxazol-4-yl)acetamide
1-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-4-phenyl-3-(piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
ethyl 4-[6-(4H-1,2,4-triazol-4-yl)pyridine-2-amido]piperidine-1-carboxylate
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-1-[3-(methoxymethyl)pyrrolidin-1-yl]propan-1-one
N-[1-(cyclohex-1-en-1-yl)ethyl]-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
1-(azocan-1-yl)-3-[4-({[(3,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)-2-methoxyphenoxy]propan-2-ol
{2-[2-(3-ethyl-1,2-oxazol-5-yl)-1H-imidazol-1-yl]ethyl}dimethylamine
3-[(3R,4S)-4-(morpholin-4-yl)-1-(4-oxo-4-phenylbutanoyl)piperidin-3-yl]propanoic acid
1-[(2-hydroxy-5-phenylphenyl)methyl]-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol