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N-[(1R,3R)-3-aminocyclopentyl]-6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
4-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-4-methoxyphenyl]thiophene-2-carboxamide
2-(dimethylamino)-N-[2-(4-ethylpiperazin-1-yl)-2-methylpropyl]-2-(2-methylphenyl)acetamide
1-propyl-3-(pyrrolidine-1-carbonyl)-N-(quinolin-3-ylmethyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(5S,9aS,9bS)-2-(1-methylpiperidin-4-yl)-5-[3-(trifluoromethyl)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(1R,5R)-6-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane
ethyl 2-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-2,7-diazaspiro[4.5]decane-7-carboxylate
4-(3-chloro-5-fluoro-4-methoxyphenyl)-7-hydroxy-1,2,3,4-tetrahydroquinolin-2-one
1-(4-methylpiperazin-1-yl)-3-(4-{[3-(pyridin-2-yl)azetidin-1-yl]methyl}phenoxy)propan-2-ol
2-({4-[4-(4-methoxypyrimidin-2-yl)piperazine-1-carbonyl]phenyl}sulfanyl)ethan-1-ol
N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-methylbenzamide
(4aS,8aR)-6-[(2-methyl-1H-imidazol-4-yl)methyl]-1-[2-(5-methylfuran-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
3-(1-benzoylpiperidin-4-yl)-4-benzyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-(5-acetamido-2-methoxyphenyl)-3-(2-methylpiperidin-1-yl)azetidine-1-carboxamide
N-[3-(furan-2-yl)propyl]-2-propyl-1,3-thiazole-4-carboxamide
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-6-[2-(hydroxymethyl)phenyl]pyridine-3-carboxamide
N-(1-{1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-4-phenylbutanamide
methyl 2-{2-[2-(cyclopentylcarbamoyl)ethyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}acetate
4-ethyl-3-{1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
4-(5-{[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]methyl}thiophen-2-yl)-2-methylbut-3-yn-2-ol
4-(2-methoxyethoxy)-1-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}piperidine
(2S)-1-[(4-methyl-1,3-thiazol-5-yl)methyl]-N-[3-(3-methylphenyl)phenyl]pyrrolidine-2-carboxamide
4-[4-(3-methoxyphenyl)-1H-pyrazol-5-yl]-1-[(2-methylphenyl)methyl]piperidine
3-[2-(cyclohexylmethyl)morpholine-4-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
[7-(quinolin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
1-{1-[3-(1H-imidazol-1-yl)propyl]piperidin-4-yl}-3-(pyrrolidine-1-carbonyl)piperidine
(2S)-2-({5-[(quinolin-6-yloxy)methyl]-1,2-oxazol-3-yl}formamido)propanamide
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-(pyridin-3-ylmethyl)piperidine-2-carboxamide
2-(pyridin-3-yl)-7-[2-(1H-1,2,4-triazol-1-yl)propanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-({1-[(2-fluorophenyl)methyl]pyrrolidin-3-yl}methyl)-2-(3-methyl-1,2-oxazol-5-yl)acetamide
N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-7H-pyrrolo[2,3-d]pyrimidin-4-amine
2-{[5-cyclopropyl-4-(2,5-dimethoxyphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
N-{[1-(3-cyclopentylpropyl)piperidin-3-yl]methyl}methanesulfonamide
N-{4-[2-(2H-1,3-benzodioxol-5-yl)acetamido]-2-chlorophenyl}propanamide
3-(1H-imidazol-2-yl)-1-(5-methyl-2-phenylfuran-3-carbonyl)piperidine
3-{1-[(4-methoxynaphthalen-1-yl)methyl]piperidin-3-yl}-1-(pyrrolidin-1-yl)propan-1-one
1-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)-3-propylpiperidine-3-carboxylic acid
({2-[6-(azepan-1-yl)pyridazin-3-yl]phenyl}methyl)dimethylamine
1-({5-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3,3-dimethylurea
{[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}[(1-ethyl-1H-imidazol-2-yl)methyl]methylamine
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-{3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}propan-1-one
1-methyl-5-(3-phenylpiperazine-1-carbonyl)-1H-pyrrole-3-carbonitrile
2-butyl-N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-1,3-benzoxazole-5-carboxamide
3-(2-chloro-4,6-dimethylphenyl)-1-(3-hydroxypropyl)-1-(pyridin-4-ylmethyl)urea
1-[2-(benzenesulfonyl)ethyl]imidazolidin-2-one
1-[1-methyl-3-(thiophen-2-yl)-1H-pyrazole-5-carbonyl]azepan-4-amine
N-[1-(2,4-dimethoxyphenyl)ethyl]-4-(3-hydroxy-3-methylbutyl)-N-methylbenzamide
3-(2-methoxyethyl)-1-methyl-5-[4-(pyrrolidin-1-yl)phenyl]-1H-1,2,4-triazole
3-[(2R,3R,6R)-5-(3-methoxybenzoyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
5-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-1H-imidazole-4-carboxylic acid