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3-ethyl-8-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-(3,4-dimethoxybenzoyl)-1-(3-phenylbenzoyl)piperidine
7-[(2,3-dimethoxyphenyl)methyl]-2-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]-2,7-diazaspiro[4.5]decane
N-[(1-benzylpiperidin-4-yl)methyl]-N,1,3-trimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
3-methyl-8-(1,2,3,4-tetrahydroquinoline-8-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
5-chloro-2-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyridine
(3R,4S)-1-(2,6-dimethylpyrimidine-4-carbonyl)-4-(4-methoxyphenyl)pyrrolidin-3-amine
8-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-(1-cyclopentanecarbonylpyrrolidin-3-yl)-1-[(2,3-difluorophenyl)methyl]piperidine
N-(2-methylpropyl)-N-(3-phenylprop-2-yn-1-yl)-3-(trimethyl-1H-pyrazol-4-yl)propanamide
N-[3-(dimethylamino)-2,2-dimethylpropyl]-3-[5-(5-methylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]propanamide
7-cyclohexyl-2-[6-(dimethylamino)pyridine-3-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
({1-[(4-fluorophenyl)methyl]-1H-1,2,4-triazol-5-yl}methyl)(methyl)(pyridin-4-ylmethyl)amine
N-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-4-[(2-methyl-3-oxopiperazin-1-yl)methyl]benzamide
ethyl 4-({[(7S,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]carbamoyl}amino)benzoate
4-({4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}methyl)phenol
N-{3-hydroxy-1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-1-oxopropan-2-yl}acetamide
2,6-dihydroxy-N-methyl-N-(thiophen-3-ylmethyl)benzamide
(4aS,7aR)-1-(3-cyclopropyl-1,2-oxazole-5-carbonyl)-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{5-[1-(2-methoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]thiophen-2-yl}ethan-1-one
N,N-dimethyl-2-[(1S,5R)-6-(3-phenylpropanoyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
2-(3-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}-3-oxopropyl)-2,3-dihydro-1H-isoindol-1-one
1-[2-(1H-imidazol-1-yl)acetyl]-N-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-4-carboxamide
(3S,4R)-1-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-methyl-N-[(3-methylthiophen-2-yl)methyl]benzamide
9-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
4-{[1-benzyl-5-(dimethyl-1,3-oxazol-5-yl)-1H-1,2,4-triazol-3-yl]methyl}-1-methylpiperidine
1-{4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}-1H-imidazole
N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-N-methyl-3-(piperidin-4-ylmethyl)benzamide
N5-[2-(2-chlorophenyl)ethyl]-1-(cyclohexylmethyl)-N3,N3-dimethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-[2-(1-methanesulfonylpiperidin-2-yl)ethyl]-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-4-(pyrrolidine-1-carbonyl)pyridine
3-methyl-1-(2-methylpropyl)-4-(5-methylthiophene-3-carbonyl)piperazin-2-one
3-(5-{3,6-dimethyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)propanoic acid
5-(2,4-dimethoxyphenyl)-N-[3-(morpholin-4-yl)propyl]-1,2,4-triazin-3-amine
2-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]acetamide
1-(diethylamino)-3-[4-({[2-(3-fluorophenyl)ethyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
N-[2-(4-hydroxyphenyl)-2-oxoethyl]-N-methyl-2-(1-propylpiperidin-4-yl)acetamide
2-tert-butyl-4-hydroxy-N-[2-(3-methoxyphenyl)ethyl]pyrimidine-5-carboxamide
N-propyl-3-({[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}sulfamoyl)benzamide
(3S,4S)-1-(2,3-dihydro-1-benzofuran-5-ylmethyl)-4-(4-fluorophenyl)piperidin-3-ol
4-benzyl-3-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
(2S,4R)-N-cyclopropyl-1-[1-(2-phenylethyl)piperidin-4-yl]-4-(pyridin-2-ylsulfanyl)pyrrolidine-2-carboxamide
5-(2-{[(4-methoxyphenyl)methyl]amino}ethyl)-1-[2-(pyridin-4-yl)ethyl]pyrrolidin-2-one
3-[(4aR,7aS)-4-[(1-ethyl-1H-pyrazol-4-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
3-(2,3-dimethoxyphenyl)-5,6-dimethyl-1,2-dihydropyridin-2-one
1-{[1-(3-fluorophenyl)-3-(furan-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-4-methyl-1,4-diazepane
N-{2-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}acetamide
4-[1-(pyridin-4-yl)-2-[2-(pyridin-4-yl)-1H-imidazol-1-yl]ethyl]morpholine
1-[5-({[2-(1-ethylpiperidin-4-yl)ethyl]amino}methyl)-2-methoxyphenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol