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N-(3-methylphenyl)-3-[1-(thiophene-3-sulfonyl)piperidin-4-yl]propanamide
9-(5-acetylthiophene-3-carbonyl)-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
3-(2-fluorophenyl)-N-(2-methoxyethyl)-3-phenylpropanamide
5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}pyridin-2-amine
2-(furan-2-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-amino-6-cyclopentyl-4-[1-(2-hydroxyethyl)-3,5-dimethyl-1H-pyrazol-4-yl]-5-methylpyridine-3-carbonitrile
4-[(2-fluoro-4-methoxyphenyl)methyl]-3-[2-oxo-2-(piperidin-1-yl)ethyl]piperazin-2-one
4-[5-chloro-2-(methylamino)benzamido]-N-ethylpiperidine-1-carboxamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-4-(2-methyl-1H-imidazol-1-yl)butanamide
N,4-dimethyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
4-[4-({3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}methyl)phenyl]-2-methylbut-3-yn-2-ol
5-{2-[3-(2-chlorophenoxy)azetidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
2-[(4-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-yl}-1H-1,2,3-triazol-1-yl)methyl]pyridine
8-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}-1,3-dioxa-8-azaspiro[4.5]decan-2-one
2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(6-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]acetamide
3-[(3S,4R)-1-benzyl-4-(pyrrolidin-1-yl)piperidin-3-yl]-N-[2-(1H-imidazol-4-yl)ethyl]propanamide
1-(2-ethoxyethyl)-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
4-[(2-fluorophenyl)methyl]-1-(1H-indol-2-ylmethyl)-1,4-diazepan-5-one
{1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}[(2,3,4-trimethoxyphenyl)methyl]amine
N-ethyl-N-{[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}oxan-4-amine
2-({1-tert-butyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)-6-methylpyridine
N-cyclopropyl-N-[(2-methoxyphenyl)methyl]-2-(1H-1,2,4-triazol-3-ylsulfanyl)acetamide
N-(1-{2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}pyrrolidin-3-yl)acetamide
4-[4-(1H-pyrazol-1-yl)phenyl]-1H-pyrazole-3-carbonitrile
N-methyl-2-[2-oxo-3-(trifluoromethyl)-1,2-dihydropyridin-1-yl]-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
1-cyclopentyl-N-(1,2-diphenylethyl)-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
{[2-chloro-5-ethoxy-4-(propan-2-yloxy)phenyl]methyl}[(5-methylpyrazin-2-yl)methyl]amine
8-[6-(4-methylpiperazin-1-yl)pyridazin-3-yl]quinoline
5-[5-(3-methoxyphenyl)furan-2-yl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-[(5-{[2-(dimethylamino)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]-3-methylthiophene-2-carboxamide
N-(4-{1-[2-(3-fluorophenyl)ethyl]-1H-imidazol-2-yl}phenyl)acetamide
N-(3-{8-methyl-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}phenyl)propanamide
methyl 3-{[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]sulfonyl}thiophene-2-carboxylate
N-[2-(dimethylamino)ethyl]-N-{[2-(4-methoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}-2-methyl-1,3-thiazole-4-carboxamide
4-(3-hydroxy-3-methylbutyl)-N-[(4-methyl-1H-imidazol-2-yl)methyl]benzamide
3-(3-phenoxypropyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)-N'-(4-methylphenyl)propanediamide
9-(benzenesulfonyl)-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
N-[(3R,4S)-1-(cyclobutylmethyl)-4-(propan-2-yl)pyrrolidin-3-yl]-5-methyl-1,3-oxazole-4-carboxamide
3-(4-{2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)benzonitrile
2-chloro-4-{[(3-hydroxypropyl)[(5-methylthiophen-2-yl)methyl]amino]methyl}-6-methoxyphenol
1-[1-ethyl-5-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]-4-phenylpiperazine
N-(2-hydroxy-3-methoxypropyl)-N,1-dimethyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-[9-(2-amino-6-methylpyrimidin-4-yl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]acetamide
2-{4-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperazin-1-yl}-5-methyl-1,3-benzoxazole
5-cyclopropyl-N,N-diethyl-1-[4-(3-fluoro-4-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
(1S,6R)-3-[2-(5-chloro-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-oxoethyl]-3,9-diazabicyclo[4.2.1]nonan-4-one
1-{4-[(2S,4S)-4-amino-1-methylpyrrolidine-2-carbonyl]piperazin-1-yl}-2-phenoxyethan-1-one
1-(furan-2-carbonyl)-4-(oxan-4-yl)-1,4-diazepane-6-carboxylic acid
(3S,4R)-1-(6-aminopyridine-3-carbonyl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid