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methyl 2-(azepane-1-sulfonyl)-6-(2,4-difluorobenzoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-(4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]methyl}-1H-pyrazol-1-yl)propanoic acid
1-methyl-9-(prop-2-en-1-yl)-4-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-1,4,9-triazaspiro[5.6]dodecan-10-one
N-(furan-2-ylmethyl)-4-[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]pyridine-2-carboxamide
4-[1-benzyl-5-(prop-2-en-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]morpholine
S-[3-(azetidine-1-carbonyl)phenyl]-N-ethyl-4-hydroxybutane-1-sulfonamido
1-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]-2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
3-(1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}piperidin-3-yl)-N-(2-fluorophenyl)propanamide
(1S,5R)-6-(2-methoxyethyl)-3-{[2-(2-methoxyphenyl)pyrimidin-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane
4-(5-{[1-(2-methylphenyl)-1H-pyrrol-2-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl)-1H-imidazole
N-benzyl-N-methyl-3-[1-(oxan-3-ylmethyl)piperidin-4-yl]propanamide
3-{2-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
1-methyl-4-[2-(methylamino)pyrimidine-5-carbonyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
5-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridine-2-carbonitrile
3-[4,5-dimethyl-1-(4-methylpyridin-2-yl)-1H-1,3-benzodiazol-2-yl]propanoic acid
ethyl 2-[2-(trifluoromethyl)morpholin-4-yl]pyridine-3-carboxylate
N-[1-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-4-hydroxy-2-(pyridin-3-yl)pyrimidine-5-carboxamide
9-(cyclopropylmethyl)-4-{imidazo[1,2-a]pyridin-2-ylmethyl}-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-methyl-8-[6-(propan-2-yl)pyrimidin-4-yl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(2,1,3-benzoxadiazol-5-ylmethyl)({[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})amine
N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-2-(2,3,6-trimethylphenoxy)acetamide
4-{[2-(4-chlorophenyl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}piperazin-2-one
N-(1-{1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-2-(3-methoxyphenyl)ethyl)-N-methylfuran-2-carboxamide
4-{7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-6-methylpyrimidin-2-amine
(3S,4S)-3-hydroxy-N-(2-phenoxyphenyl)-4-(pyrrolidin-1-yl)pyrrolidine-1-carboxamide
N-benzyl-3-{[(3-fluoropyridin-2-yl)amino]methyl}-N-methylpyridin-2-amine
N-cyclopentyl-4-(pyrazin-2-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
(3S,4S)-4-methyl-1-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]piperidine-3,4-diol
9-methyl-2-({4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}methyl)-4H-pyrido[1,2-a]pyrimidin-4-one
1-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]urea
(2S,4R)-N-ethyl-4-{imidazo[1,2-a]pyrimidine-2-amido}-1-(2-methoxyacetyl)pyrrolidine-2-carboxamide
1-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(2,5-dimethylphenyl)ethan-1-one
1-[(3S,4R)-3-cyclopropyl-4-(dimethylamino)pyrrolidin-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
1-[2-hydroxy-2-(pyridin-3-yl)ethyl]-3-[5-(2-phenylethyl)-1,3,4-thiadiazol-2-yl]urea
N-cyclopentyl-2-{[4-methyl-5-(piperidin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}butanamide
1-cyclopropanecarbonyl-4-(4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}phenoxy)piperidine
(2S)-2-amino-4-(1-tert-butyl-3-phenyl-1H-1,2,4-triazol-5-yl)butanoic acid
1-(pyridin-2-ylmethyl)-4-[4-(2,2,2-trifluoroethyl)piperazine-1-carbonyl]pyrrolidin-2-one
(1S,5R)-3-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(2-methylpropyl)-N-(thiophen-3-ylmethyl)-3-(4H-1,2,4-triazol-4-yl)benzamide
N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-5-[3-(trifluoromethyl)phenoxymethyl]-1H-pyrazole-3-carboxamide
N-benzyl-N-(1,3-thiazol-2-ylmethyl)-1H-imidazole-2-carboxamide
3-(2-methoxyethyl)-5-[2-(1H-pyrazol-1-yl)phenyl]-1,2,4-oxadiazole
3-(3-fluorophenyl)-4-(4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)piperazin-2-one
N-(carbamoylmethyl)-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
7,7-dimethyl-2-(1-phenylpyrrolidin-3-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-amino-1-{7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}ethan-1-one
9-[(4-ethoxyphenyl)methyl]-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
N-{2-[ethyl(methyl)amino]-2-methylpropyl}-2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
7-(2-amino-4-ethyl-1,3-thiazole-5-carbonyl)-N2,N2,N4,N4-tetramethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine