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N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-2-(2-phenyl-1H-imidazol-1-yl)acetamide
N-[(3S,4R)-4-propyl-1-(quinoline-6-carbonyl)pyrrolidin-3-yl]acetamide
1-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
N,3-dimethyl-5-propyl-N-[2-(1H-pyrazol-4-yl)ethyl]-1-benzofuran-2-carboxamide
N,N-dimethyl-1-(5-propyl-1,3,4-oxadiazol-2-yl)azepan-4-amine
5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-ethyl-1H-pyrazole-4-carboxamide
N-[(4-hydroxyazepan-4-yl)methyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
3-[(1R,2R)-2-(benzyloxy)cyclopentyl]-1-(2-methoxyphenyl)urea
N-[4-(furan-2-yl)butan-2-yl]-3-propanamidobenzamide
2-[(1-methyl-1H-indol-3-yl)sulfanyl]-N-[(5-methylpyrazin-2-yl)methyl]acetamide
(3S,9aR)-8-(2-chlorobenzoyl)-3-[(1R)-1-hydroxyethyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)-1-benzofuran-5-carboxamide
N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-{methyl[2-(2-methyl-1H-imidazol-1-yl)ethyl]amino}-2-[4-(1H-pyrazol-1-yl)phenyl]acetic acid
(2S,4R)-4-(4-butyl-1H-1,2,3-triazol-1-yl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
methyl 3-(furan-3-amido)-5-({[4-(piperidin-1-ylmethyl)phenyl]formamido}methyl)benzoate
1-benzyl-N-(2,3-dihydro-1H-inden-2-yl)-N-methyl-1H-pyrazole-4-carboxamide
4-{[3-(2,3-dimethoxyphenyl)pyrrolidin-1-yl]methyl}-3-methyl-1-(prop-2-en-1-yl)-1H-pyrazole
(1S,4R)-2-[(3,4-dichlorophenyl)methyl]-2-azabicyclo[2.2.1]heptan-3-one
3-[2-(4-methoxy-4-phenylpiperidin-1-yl)-2-oxoethyl]-3,4-dihydroquinazolin-4-one
(4aS,7aR)-1-(2,5-dimethylbenzoyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[7-(cyclopropylmethyl)-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl]benzonitrile
2,6-diamino-4-(2-chloro-3,4-dimethoxyphenyl)-5,6,7,8-tetrahydroquinoline-3-carbonitrile
(3R,4R)-1-[(3-chloro-4-ethoxyphenyl)methyl]-4-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-3-ol
3-(azetidine-1-sulfonyl)-N-[3-(methylsulfanyl)propyl]benzamide
1-methyl-4-({5-[1-(prop-2-en-1-yl)pyrrolidin-2-yl]-1,2,4-oxadiazol-3-yl}methyl)piperidine
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(2-methoxyphenyl)propan-1-one
[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl](methyl)[1-(pyridin-2-yl)ethyl]amine
6-(4-{2-[(propan-2-yl)amino]pyrimidine-5-carbonyl}piperazin-1-yl)pyridine-3-carbonitrile
4-{[2-(benzylamino)pyrimidin-5-yl]methyl}piperazine-2-carboxylic acid
1-[1-(4-ethyl-5-methylpyrimidin-2-yl)piperidin-3-yl]pyrrolidin-2-one
N-{2-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]ethyl}-2-(2,5-dioxoimidazolidin-1-yl)acetamide
N-(3-{[(4-chlorophenyl)methyl]sulfanyl}propyl)pyrrolidine-3-carboxamide
1-[4-(8-methoxyquinolin-2-yl)phenyl]ethan-1-one
(3R,4R)-1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(morpholin-4-yl)piperidin-3-ol
3-({2-[1-(2-ethylbenzoyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
2-(2-hydroxypropyl)-9-(3-hydroxypyridine-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)pyrimidin-2-amine
N-[(3-methylphenyl)methyl]-3-(1-methylpiperidin-3-yl)-N-(propan-2-yl)propanamide
methyl 3-[(3S,4R)-1-[(2-hydroxy-5-methoxyphenyl)methyl]-4-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-3-yl]propanoate
[4-(4,6-dimethylpyrimidin-2-yl)phenyl]methanol
N-[(2-methylphenyl)methyl]-5-(phenoxymethyl)-N-(propan-2-yl)-1H-pyrazole-3-carboxamide
N-benzyl-2-[4-(4-{[2-(furan-2-yl)ethyl]amino}piperidin-1-yl)phenyl]acetamide
8-(2,3-dihydro-1-benzofuran-5-ylmethyl)-3-[(4-methoxyphenyl)methyl]-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-methyl-3-[3-(pyridin-2-yl)azetidine-1-carbonyl]-1,2,5,6,7,8-hexahydroquinolin-2-one
ethyl 4-{6-[2-(1,3-dioxo-2,3-dihydro-1H-isoindol-2-yl)acetyl]-6-azaspiro[2.5]octane-1-carbonyl}piperazine-1-carboxylate
5,5-dimethyl-3-{2-oxo-2-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethyl}imidazolidine-2,4-dione
N-ethyl-1-[(3-methoxyphenyl)methyl]-5-(quinoline-6-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)-3-(pyridin-3-yl)propan-1-one
5-cyclopropyl-N-methyl-1-[4-(5-methylfuran-2-yl)pyrimidin-2-yl]-N-[2-(pyridin-2-yl)ethyl]-1H-pyrazole-4-carboxamide