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[1-(2,1,3-benzoxadiazol-4-ylmethyl)-4-benzylpiperidin-4-yl]methanol
2-(3,4-difluorophenyl)-N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]acetamide
4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(propan-2-yl)piperidine
(3aS,7aR)-5-methyl-2-[2-(pyridin-4-yl)-1,3-thiazole-4-carbonyl]-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
1-{4-[(cycloheptylamino)methyl]-2-methoxyphenoxy}-3-(4-ethylpiperazin-1-yl)propan-2-ol
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-3-(methylsulfanyl)propanamide
1-[(3S,4R)-4-amino-3-methoxypiperidin-1-yl]-3-(2H-1,3-benzodioxol-5-yl)propan-1-one
3-{5-[(6-methoxy-1H-indazol-3-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
2-(3-fluorophenyl)-8-methoxy-5-(pyridin-4-ylmethyl)-2,3,4,5-tetrahydro-1,5-benzothiazepine
1-{2-[1-(3-fluorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]phenyl}-1,3-diazinane-2,4-dione
4-benzyl-3-ethyl-1-(isoquinoline-5-carbonyl)-1,4-diazepan-5-one
N-[2-(4-fluorophenyl)ethyl]-3-(1H-pyrazol-4-yl)benzamide
N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]quinoxaline-6-carboxamide
(4aS,8aR)-6-[(2-phenyl-1,3-oxazol-4-yl)methyl]-1-propyl-decahydro-1,6-naphthyridin-2-one
methyl (1R,3S,3aR,6aS)-3-(6-methoxy-2H-1,3-benzodioxol-5-yl)-1,5-dimethyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-(1H-1,3-benzodiazol-2-ylmethyl)-N-methyl-2-(3-phenylpropyl)-1,3-benzoxazole-5-carboxamide
{1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-3-(2-phenylethyl)piperidin-3-yl}methanol
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-methyl-N-[(5-phenyl-1H-pyrazol-3-yl)methyl]acetamide
N-(1-{2-[cyclohexyl(methyl)amino]-4-methylpyrimidin-5-yl}ethyl)-5-oxo-2,5-dihydro-1H-pyrazole-3-carboxamide
N-[2-fluoro-5-({methyl[3-(oxolan-2-yl)propyl]carbamoyl}amino)phenyl]acetamide
1-(cyclopropylmethyl)-N-methyl-N-(1,3-thiazol-4-ylmethyl)-5-[2-(thiophen-3-yl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(1R,4S)-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-1,7,7-trimethyl-3-oxo-2-oxabicyclo[2.2.1]heptane-4-carboxamide
3-(1-{1-[(2-ethoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(2-methoxyphenyl)urea
1-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-N-[1-(2-methylpropyl)cyclopropyl]piperidin-4-amine
1-cyclohexyl-N-cyclopentyl-4-oxo-5-(pyrrolidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
2-(propan-2-yl)-4-{1-[2-(pyridin-2-ylsulfanyl)ethyl]-1H-imidazol-2-yl}pyrimidine
3-methyl-N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
7-cyclohexyl-6-oxo-N-phenyl-2,7-diazaspiro[4.5]decane-2-carboxamide
3-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-1-[3-methoxy-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
5-[methoxy(phenyl)methyl]-3-(oxan-4-yl)-1H-1,2,4-triazole
3-(dimethyl-1,2-oxazol-4-yl)-N,N-bis(1,3-oxazol-4-ylmethyl)propanamide
N-methyl-2-{2-[2-(morpholin-4-yl)pyrimidin-5-yl]-1H-imidazol-1-yl}ethane-1-sulfonamide
1-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carbonyl}-4-(thian-4-yl)piperazine
5-{[2-(diethylamino)ethyl](ethyl)amino}-N,N-dimethyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
3-[(5-chlorothiophen-2-yl)methyl]-8-(trifluoromethyl)-3,4-dihydroquinazolin-4-one
1-(2-{1-[2-(1H-1,2,4-triazol-1-yl)benzoyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
1-(azetidin-1-yl)-2-(morpholin-4-yl)-2-(pyridin-3-yl)ethan-1-one
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-(2-methoxyphenyl)piperazine
1-{5-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]thiophen-2-yl}ethan-1-one
N-{[5-(dimethylcarbamoyl)furan-2-yl]methyl}-3,5,7-trimethyl-1H-indole-2-carboxamide
4-(2-{8-[2-(dimethylamino)ethyl]-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-2-oxoethyl)-1,2,3,6-tetrahydropyridazine-3,6-dione
7-methoxy-N-[2-(pyrrolidine-1-sulfonyl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-(2-methylphenyl)-3-phenyl-N-{2-[(pyridin-3-yl)amino]ethyl}propanamide
(3S,4R)-3-methoxy-1-[4-(1H-pyrazol-3-yl)benzoyl]piperidin-4-amine
4-oxo-6-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}-1,4-dihydroquinoline-3-carboxylic acid
[(3S,5R)-1-(dimethyl-1,3-thiazole-5-carbonyl)-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
(1S,5R)-6-(2-methoxyethyl)-3-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
(1R,5R)-6-(5-chloro-2-hydroxybenzoyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-(cyclopentylmethyl)-3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-(4-{2-oxo-1-oxaspiro[4.5]decane-4-carbonyl}piperazin-1-yl)pyridine-3-carbonitrile