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N-[3-(methylsulfanyl)propyl]-3-(piperidine-1-carbonyl)pyrazine-2-carboxamide
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-2-(1H-imidazol-1-yl)propanamide
N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-5-(thiophen-2-yl)-1H-pyrazole-4-carboxamide
2-{2-[4-(2-methylphenoxy)piperidin-1-yl]ethyl}pyridine
N-[3-(furan-2-yl)-1H-1,2,4-triazol-5-yl]-4-(pyridin-3-yl)-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carboxamide
4-(6-amino-2-{[(2-methylphenyl)methyl]sulfanyl}pyrimidin-4-yl)-1-ethylpiperazin-2-one
N-methyl-6-(methylamino)-N-(quinolin-2-ylmethyl)pyridine-3-carboxamide
[(4-{1-azabicyclo[3.2.1]octan-5-yloxy}phenyl)methyl][(1-ethyl-1H-pyrazol-4-yl)methyl]amine
N-[(4-methoxyphenyl)methyl]-N-(pyridin-4-ylmethyl)-1-benzofuran-3-carboxamide
5-(2-butoxy-4-fluorophenyl)-3-(methoxymethyl)-1H-1,2,4-triazole
(3S,4S)-1-{[2-(difluoromethoxy)phenyl]methyl}-4-[methyl(pyrazin-2-ylmethyl)amino]pyrrolidin-3-ol
5-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidine-1-carbonyl]pyrazin-2-ol
N-[2-(3-methoxyphenyl)-1-[1-(1-methyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]ethyl]-N-methyl-3-(methylsulfanyl)propanamide
1-methyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}azepane-2-carboxamide
3-(2-ethyl-5-oxopyrrolidin-2-yl)-N-[3-(propan-2-yloxy)propyl]propanamide
2-(1-{[(2-methyl-2H-1,2,3-triazol-4-yl)carbamoyl]methyl}-1H-pyrazol-4-yl)benzamide
1-(2-{4-[5-methyl-2-(1H-pyrazol-1-yl)phenyl]-1H-1,2,3-triazol-1-yl}ethyl)imidazolidin-2-one
2-(1H-pyrazol-4-yl)-4-(trifluoromethyl)pyridine
(2S)-2-[3-(diphenylmethyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]propanoic acid
N-methyl-N-(pyrazin-2-ylmethyl)-3-(thiophen-3-yl)-1H-pyrazole-5-carboxamide
4-{[5-(1H-imidazol-4-yl)-4-phenyl-1H-imidazol-1-yl]methyl}benzene-1-sulfonamide
4-methyl-5-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-2-(propan-2-yl)pyrimidine
1-(2-methoxy-6-{[methyl(oxan-4-ylmethyl)amino]methyl}phenoxy)-3-(morpholin-4-yl)propan-2-ol
N-[2-(4-hydroxypiperidin-1-yl)-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl]pyridine-2-carboxamide
2-(1,3-dioxo-2,3-dihydro-1H-isoindol-2-yl)-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)acetamide
4-{1-[1-(3,6-dimethylpyrazin-2-yl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
4-fluoro-N-{3-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]-3-oxopropyl}benzamide
5-[4-(adamantan-1-yl)piperazine-1-carbonyl]-N,4-dimethyl-1,3-thiazol-2-amine
3-cyclopropyl-1-{spiro[azepane-4,2'-chromene]-1-yl}propan-1-one
1-{octahydro-1H-pyrido[1,2-a]piperazin-2-yl}-2-(2,4,7-trimethyl-1H-indol-3-yl)ethan-1-one
2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(3-methoxypropyl)acetamide
1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one
2-cyclopropyl-4-methyl-5-[4-(3-methylphenoxy)piperidine-1-carbonyl]pyrimidine
1-(4-chlorophenyl)-N-{[6-(dimethylamino)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-N-[2-(dimethylamino)ethyl]cyclopropane-1-carboxamide
3-hydroxy-1-[(3-methylphenyl)methyl]-3-[(propylamino)methyl]piperidin-2-one
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[2-(pyridin-3-yl)acetyl]pyrrolidine-3-carboxylic acid
ethyl 1-[(2-hydroxy-3-methoxyphenyl)methyl]-4-(2-phenoxyethyl)piperidine-4-carboxylate
1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine
2-(1-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)propan-2-ol
1-(azepan-1-yl)-3-(4-chloro-2-{[(2-methoxyethyl)(methyl)amino]methyl}phenoxy)propan-2-ol
5-methyl-N-{[7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1,2-oxazole-3-carboxamide
(1-{1-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}piperidin-3-yl)methanol
6-chloro-N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-N-methylimidazo[1,2-a]pyridine-2-carboxamide
1-[2-(4-{1H-pyrazolo[3,4-b]pyridin-1-yl}phenoxy)ethyl]-1H-imidazole
4-{[4-fluoro-3-(trifluoromethyl)phenyl]methyl}-3-methyl-1-(2-methylpropyl)piperazin-2-one
4-amino-N-(2-benzylphenyl)azepane-1-carboxamide
6,8-dimethyl-3-({methyl[2-(4-methyl-1,3-thiazol-5-yl)ethyl]amino}methyl)-1,2-dihydroquinolin-2-one
2-(dimethylamino)-2-(2-fluorophenyl)-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)acetamide
2-[1-(oxolan-3-ylmethyl)azetidin-3-yl]-1H-1,3-benzodiazole
(2S)-3-hydroxy-2-(methylamino)-1-[4-(2-methylphenyl)-1,4-diazepan-1-yl]propan-1-one