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N,6-dimethyl-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-2-(pyridin-3-yl)pyrimidin-4-amine
5-(4-methanesulfonylphenoxy)-1-azabicyclo[3.2.1]octane
{[6-chloro-2-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}(methyl)[(1-methyl-1H-imidazol-2-yl)methyl]amine
methyl 3-(cyclobutylmethoxy)-5-(4-methyl-1,4-diazepane-1-carbonyl)benzoate
N-{1-[(3-chlorophenyl)methyl]-3-methyl-1H-pyrazol-5-yl}-3-methoxypyrrolidine-1-carboxamide
2-(4-benzyl-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]acetamide
2-ethyl-8-[(4-methylphenyl)methanesulfonyl]-2,8-diazaspiro[5.5]undecan-3-one
N-[(3R,4R)-1-[(2-tert-butyl-5-carbamoylfuran-3-yl)methyl]-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
(4aR,7aS)-1-(2-hydroxyethyl)-4-[4-(2-oxopyrrolidin-1-yl)butanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-amine
(1R,3S)-3-[2-(dimethylamino)ethoxy]-7-(5-ethenylpyridin-2-yl)-7-azaspiro[3.5]nonan-1-ol
methyl(3-methylbut-2-en-1-yl){[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
1-[2-methoxy-4-({[(3-methylphenyl)methyl]amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
ethyl 3-{[3-(5-fluoro-2-methoxybenzoyl)piperidine-1-carbonyl]amino}propanoate
2-{methyl[(2-phenyl-1,3-thiazol-4-yl)methyl]amino}-N-(pyrazin-2-yl)acetamide
{[2-(2,2-dimethylpropanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
5-[4-(morpholin-4-yl)piperidine-1-carbonyl]-N-(propan-2-yl)pyridin-2-amine
methyl (2S,4R)-1-methyl-4-[2-(3-methyl-2-oxo-1,2,3,4-tetrahydroquinazolin-1-yl)acetamido]pyrrolidine-2-carboxylate
2-[4-(2-methoxyethoxy)phenyl]-3-(pyrrolidin-1-yl)pyrazine
2-chloro-4-{[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]methyl}phenol
2-methyl-5-{2-oxo-2-[(1R,5R)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethyl}-3,4-dihydropyrimidin-4-one
1-{imidazo[1,2-a]pyrimidine-2-carbonyl}-4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]piperidine
1-methyl-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]cyclopropane-1-carboxamide
(4aS,7aR)-4-benzyl-6,6-dioxo-N-(propan-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-1-(2-methoxyphenyl)-N-methyl-1H-pyrazole-4-carboxamide
5-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-2-amine
1-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(thiophen-3-yl)propan-1-one
2-amino-N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}acetamide
4-(2,5-dichlorophenyl)-2-(methylsulfanyl)pyrimidine
methyl (2S,4S,5R)-5-(2-chlorophenyl)-4-[(3-methoxy-3-oxopropyl)carbamoyl]-1,2-dimethylpyrrolidine-2-carboxylate
4-({[(3-ethyl-1,2-oxazol-5-yl)methyl](methyl)amino}methyl)-1-azatricyclo[7.3.1.05,13]trideca-3,5,7,9(13)-tetraen-2-one
3-{[(1-ethylcyclopropyl)carbamoyl]methyl}-N-(2-methoxyethyl)-4-methyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
2-{3-[(3,4-dimethoxyphenyl)amino]piperidin-1-yl}-6-methylpyridine-3-carbonitrile
N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]pyrimidin-4-amine
4-(hydroxymethyl)-1-{[2-(4-methoxyphenyl)imidazo[1,2-a]pyridin-3-yl]methyl}azepan-4-ol
(3R,5S)-1-[(3,4-dimethoxyphenyl)methyl]-N-[3-(morpholin-4-yl)propyl]-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
2-(dimethylamino)-2-(2-fluorophenyl)-1-(thiomorpholin-4-yl)ethan-1-one
2-[4-(1-benzofuran-2-ylmethyl)-1-cyclopentylpiperazin-2-yl]ethan-1-ol
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-5-fluoro-4-(morpholin-4-yl)pyrimidin-2-amine
(3S,4S)-4-cyclopropyl-1-[1-(2-methoxyphenyl)piperidin-4-yl]pyrrolidine-3-carboxylic acid
4-{4-[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carbonyl}-6-methylquinoline
methyl 6-(3,4-dimethylbenzoyl)-2-[(2-methylphenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-(dimethylamino)-7-[5-(pyrrolidin-2-yl)thiophene-2-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-(2,3-dihydro-1H-inden-2-yl)-3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
ethyl 1-[5-methyl-4-(4-methylpiperazin-1-yl)thieno[2,3-d]pyrimidine-6-carbonyl]piperidine-3-carboxylate
2-[1-(3-methoxypropyl)-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}acetamide
2-({4-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}methyl)pyridine
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(methyl)[(5-methylfuran-2-yl)methyl]amine
5-fluoro-2-{1-[4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]piperidin-4-yl}-1H-1,3-benzodiazole