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methyl({[4-(5-methylpyridin-2-yl)piperidin-4-yl]methyl})(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)amine
N-(4-methyl-1,3-thiazol-2-yl)-5-[1-(1H-pyrrole-2-carbonyl)pyrrolidin-2-yl]thiophene-2-carboxamide
6-[4-(aminomethyl)piperidin-1-yl]-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide
1-tert-butyl-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-5-oxopyrrolidine-3-carboxamide
7-(propan-2-yl)-N-[(4-sulfamoylphenyl)methyl]-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
2-(dimethyl-1,2-oxazol-4-yl)-1-{4-[4-({methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}methyl)phenoxy]piperidin-1-yl}ethan-1-one
5-{[2-(oxolan-3-yl)-1H-imidazol-1-yl]methyl}-3-(propan-2-yl)-1,2-oxazole
4-(2-methoxyphenyl)-6-(1H-pyrazol-1-yl)pyrimidine
1-(azocan-1-yl)-3-[2-methoxy-4-({[(3-methylphenyl)methyl]amino}methyl)phenoxy]propan-2-ol
2-{2-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethoxy}ethan-1-ol
1-{1-azabicyclo[2.2.2]octan-3-yl}-3-(8-chloro-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)urea
N-cyclopropyl-N-({4-[3-(dimethylamino)propoxy]phenyl}methyl)pyridine-2-carboxamide
4-(1-benzothiophene-5-carbonyl)thiomorpholine
5-fluoro-N4,N4-dimethyl-N2-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}pyrimidine-2,4-diamine
6-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-ethylpyridine-3-carboxamide
1-[(5-ethylpyridin-2-yl)methyl]-4-(pyrimidin-2-yl)-1,4-diazepane
5-{[1-(2-carboxyethyl)-1H-pyrazol-4-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
[(4-ethyl-5-{1-[1-(propan-2-yl)piperidin-4-yl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2,5-dimethylfuran-3-carboxamide
1-acetyl-N-[2-(azepan-1-yl)ethyl]-N-(propan-2-yl)piperidine-4-carboxamide
2-amino-6-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-4-{2-[(propan-2-yl)amino]pyrimidin-5-yl}pyridine-3-carbonitrile
[1-(1H-indol-3-ylmethyl)-4-(2-phenoxyethyl)piperidin-4-yl]methanol
(2S)-2-{[5-(3-acetylphenoxymethyl)-1,2-oxazol-3-yl]formamido}propanamide
3-(2-aminoethyl)-N-[3-(4-chlorophenyl)phenyl]piperidine-1-carboxamide
3-(1-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-2-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{4-[1-(2H-1,3-benzodioxol-5-yl)-3-methyl-1H-1,2,4-triazol-5-yl]phenyl}acetamide
N'-{[4-(cyclobutylmethoxy)phenyl]methyl}-N'-cyclopropyl-N,N-dimethylbutanediamide
{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(prop-2-en-1-yl)(prop-2-yn-1-yl)amine
1-{2-[9-methoxy-7-(3-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}-4-phenylpyrrolidin-2-one
3-(1-{3-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}pyrrolidin-2-yl)-4-methyl-1,2,5-oxadiazole
2-{5-[2-(2-fluorophenyl)ethyl]-1,2,4-oxadiazol-3-yl}pyrazine
1-(1-propyl-1H-pyrazole-5-carbonyl)-N-(pyridin-4-ylmethyl)piperazine-2-carboxamide
2,6-difluoro-4-methoxy-N-propyl-N-(pyridin-3-ylmethyl)benzamide
3-ethyl-4-methyl-N-(3-{[(3-methylphenyl)methyl]sulfanyl}propyl)-1H-pyrazole-5-carboxamide
1-(5-cyclobutyl-1,3,4-oxadiazol-2-yl)-4-(pyridin-4-ylmethyl)-1,4-diazepane
1-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
6-{4-[(5-methylnaphthalen-1-yl)methyl]piperazin-1-yl}pyrazine-2-carboxamide
N-[4-methyl-2-(4H-1,2,4-triazol-4-yl)phenyl]cyclopentanecarboxamide
2-{2-[(dimethylamino)methyl]-4-(pyrimidin-2-yl)phenoxy}-N-[1-(1,3-thiazol-2-yl)ethyl]acetamide
ethyl 1-(2-amino-6-methylpyrimidine-4-carbonyl)-4-[(4-chlorophenyl)methyl]piperidine-4-carboxylate
2-(4-cyclohexanecarbonylmorpholin-3-yl)-N-[(2-methoxyphenyl)methyl]acetamide
4-[3-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-(2-methoxyethyl)-2-methyl-N-(thiophen-2-ylmethyl)imidazo[1,2-a]pyrimidine-3-carboxamide
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(4-methyl-1,3-thiazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
7-methyl-4-(2-methylpyrrolidine-1-carbonyl)-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline
2-{2-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-ylmethyl]phenoxy}acetic acid
N-[3-(1H-imidazol-1-yl)propyl]-2,6,8-trimethylquinoline-4-carboxamide
2-[1-(3,5-dimethylphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]-5-methyl-1,3,4-oxadiazole
1,3-dimethyl-6-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-{[3-(3-methylphenoxy)azetidin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid