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5-(2H-1,3-benzodioxole-5-carbonyl)-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
9-(2-fluorobenzoyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[(4aS,8aS)-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-3-cyclohexylpropan-1-one
5-({4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}methyl)-N,N-dimethylpyridin-2-amine
4-benzyl-3-[1-(dimethyl-1,3-oxazole-4-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
[1-(2-ethoxyethyl)-3-(prop-2-en-1-yl)piperidin-3-yl]methanol
(3R,4R)-1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
(3R,4R)-4-ethyl-1-{[5-(3-fluorophenyl)-1,3,4-oxadiazol-2-yl]methyl}piperidine-3,4-diol
N3-[1-(furan-2-yl)ethyl]-4-oxo-N5-(2-phenylethyl)-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
4-[(3R,4R)-3-cyclopropyl-3-hydroxy-4-methylpyrrolidine-1-carbonyl]-1λ6-thiane-1,1-dione
3-(2-methylphenyl)-5-(morpholine-4-sulfonyl)benzoic acid
2-amino-N-methyl-N-[(3-methyl-1H-indol-2-yl)methyl]-5,6,7,8-tetrahydroquinazoline-4-carboxamide
7-(cyclopropylmethyl)-2-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-1-[2-(pyridin-2-yl)ethyl]piperidin-2-one
1-(1-methylpiperidin-4-yl)-N-[1-(thiophen-3-yl)ethyl]piperidine-4-carboxamide
N-methyl-2-{8-methyl-3-oxo-2,8-diazaspiro[4.5]decan-2-yl}-N-{[3-(methylsulfanyl)phenyl]methyl}acetamide
N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-4-(1H-pyrazol-3-yl)benzamide
2-(4-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}piperazin-1-yl)ethan-1-ol
methyl 2-(2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamido)acetate
2-(2-hydroxyethyl)-9-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[(2-chlorophenyl)methyl]-7-fluoro-3-({[2-(1H-imidazol-1-yl)ethyl]amino}methyl)-1,2-dihydroquinolin-2-one
(1,3-benzothiazol-2-ylmethyl)(methyl){[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}amine
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]pyrrolidin-3-yl]methanol
{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}(methyl)(pyridin-3-ylmethyl)amine
7-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carbonyl}-3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
(2S)-1-[4-(4-chlorophenoxy)piperidine-4-carbonyl]-N,N-dimethylpyrrolidine-2-carboxamide
(3R,4S)-1-[(1,5-dimethyl-1H-indol-2-yl)methyl]-3,4-dimethylpiperidin-4-ol
4-cyclopentyl-N-(1,3-thiazol-2-ylmethyl)pyrimidin-2-amine
1-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-{[(4-fluorophenyl)methyl](methyl)amino}ethan-1-one
N-[(3-ethoxyphenyl)methyl]-6-oxo-N-(prop-2-en-1-yl)-1,6-dihydropyridine-3-carboxamide
ethyl 4-[3-(methylcarbamoyl)-6-oxo-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl]-1H-pyrazole-3-carboxylate
1-cyclohexyl-1-(pyridin-2-ylmethyl)-3-{[1,2,4]triazolo[4,3-a]pyridin-8-yl}urea
3,5-dimethyl-1-(1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}azetidin-3-yl)-1H-pyrazole
({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)(methyl)[1-(4-methyl-1,3-thiazol-2-yl)ethyl]amine
1-[(4-fluorophenyl)methyl]-4-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-1,4-diazepane
N,N-diethyl-1-[(1s,4s)-4-(4-acetamidobenzamido)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3-(2-chlorophenyl)-3-(3-hydroxyphenyl)-N-methyl-N-(pyrimidin-4-ylmethyl)propanamide
(1R,2S)-2-{[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}cyclopentane-1-carboxamide
7-[3-(thiophen-2-yl)propanoyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
(3S,4S)-4-(piperidin-1-yl)-1-[3-(1H-pyrazol-1-yl)benzoyl]pyrrolidin-3-ol
(3R,4R)-1-{[3-(furan-2-yl)phenyl]methyl}-4-(4-methylpiperazin-1-yl)piperidin-3-ol
1-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-4-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperazine
2-[2-(3-methyl-4H-1,2,4-triazol-4-yl)ethyl]-2-azatricyclo[6.3.1.04,12]dodeca-1(12),4,6,8,10-pentaen-3-one
3-(2,5-dioxoimidazolidin-4-yl)-N-[2-(4-fluorophenoxy)ethyl]propanamide
6-({3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}methyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-ethyl-2-(4-{[3-(3-methoxyphenyl)phenyl]methyl}piperazin-1-yl)acetamide
2-methoxy-1-[(1S,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
1-(methoxymethyl)-N,N-bis(pyridin-3-ylmethyl)cyclobutane-1-carboxamide
2-[4-(cyclohexylmethyl)-1-cyclopentylpiperazin-2-yl]ethan-1-ol
1-methyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carboxamide