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N-[2-(3-ethoxyphenoxy)ethyl]-N-methyl-2-(propan-2-yloxy)propanamide
3-(3,4-dimethylphenyl)-1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]propan-1-one
N-[(2-chloro-6-fluorophenyl)methyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
4-(2,5-dimethylphenyl)-3-propyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
5-[3-({[5-(pyrimidin-2-ylsulfanyl)furan-2-yl]methyl}amino)propyl]-1,3,4-thiadiazol-2-amine
3,3-dimethyl-4-[3-(2-methylphenyl)-3-phenylpropanoyl]piperazin-2-one
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-[(1-methylpyrrolidin-3-yl)methyl]acetamide
1-(2,5-dimethylfuran-3-carbonyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N,1-dimethyl-6-propyl-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
5-[(1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonane-9-carbonyl]-2,1,3-benzoxadiazol-1-ium-1-olate
2-(dimethylamino)-N-({2-[(dimethylamino)methyl]phenyl}methyl)-2-(3-fluorophenyl)-N-methylacetamide
2-[(4aR,7aS)-4-[(5-methylthiophen-2-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N,N-dimethylacetamide
2-(dimethylamino)-7-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-[3-cyclopropyl-1-(3,4-dimethylphenyl)-1H-1,2,4-triazol-5-yl]-6-(4H-1,2,4-triazol-4-yl)pyridine
1-{1-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]piperidin-4-yl}-1,4-diazepane
N-ethyl-6-[3-(1H-imidazol-2-yl)piperidin-1-yl]-N-methylpyridine-3-carboxamide
2-{1-[4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]piperidin-4-yl}-1H-1,3-benzodiazole
N-[2-(5-hydroxypyrazine-2-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]oxolane-2-carboxamide
N-(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
N,1-dimethyl-2-oxo-N-(quinolin-5-ylmethyl)imidazolidine-4-carboxamide
1-(2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}-5-methoxyphenyl)-3,5-dimethyl-1H-pyrazole
2-{4-[2-(thiophen-2-yl)ethyl]piperazin-1-yl}phenol
2-cyclopropyl-8-[(3,5-difluoro-4-methoxyphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
(4aS,7aR)-1-[2-(methylamino)-1,3-thiazole-4-carbonyl]-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
{[2-(cyclopentanesulfonyl)-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}bis(prop-2-en-1-yl)amine
3-{2-cyclopropyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-N,N-dimethylpropanamide
N-[2-(2-chlorophenyl)-2-(dimethylamino)ethyl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-N-[(4-methyl-1,3-thiazol-2-yl)methyl]pyridin-2-amine
5-(methoxymethyl)-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1H-pyrazole-4-carboxamide
4-(3-methylphenoxy)-1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperidine-4-carboxylic acid
3-bromo-5-[(propan-2-yl)sulfamoyl]benzoic acid
2-{[3-(diethylcarbamoyl)piperidin-1-yl]methyl}pyridine-3-carboxylic acid
N-[(3R,4S)-1-methanesulfonyl-4-(propan-2-yl)pyrrolidin-3-yl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propanamide
5-tert-butyl-N-{[4-(piperidine-1-carbonyl)phenyl]methyl}-1,3,4-oxadiazol-2-amine
1-cyclopentyl-4-oxo-5-(piperidine-1-carbonyl)-N-[2,2,2-trifluoro-1-(furan-2-yl)ethyl]-1,4-dihydropyridine-3-carboxamide
5-ethyl-4-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-methylpyrimidine
2-({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}sulfonyl)-2,8-diazaspiro[4.5]decane
5-{[4-(2,2-dimethyloxan-4-yl)-1H-1,2,3-triazol-1-yl]methyl}thiophene-2-carboxylic acid
5-({3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}methyl)-N-(propan-2-yl)pyrimidin-2-amine
(1S,5R)-6-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
[1-(3-chloro-5-fluorobenzoyl)-3-(2-methoxyethyl)piperidin-3-yl]methanol
N-[3-(1-oxo-2,3-dihydro-1H-inden-5-yl)phenyl]acetamide
1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
6-fluoro-4-{3-[(1-propylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}-1,2-dihydroquinolin-2-one
N-{[2-(diethylamino)pyridin-3-yl]methyl}-2,3-dihydro-1,4-benzodioxine-2-carboxamide
2-{1-cyclohexyl-4-[(2,5-dimethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
6-(2-methoxyethyl)-2-(4-{[methyl(pyridin-2-ylmethyl)amino]methyl}phenyl)-3,4-dihydropyrimidin-4-one
(1S,5R)-3-[2-(phenylsulfanyl)acetyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-[4-(5-{[(3-fluorophenyl)carbamoyl]amino}-1H-pyrazol-1-yl)piperidin-1-yl]acetamide
3-{[4-methyl-6-({2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}amino)pyrimidin-2-yl]amino}phenol