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4-(cyclohex-3-en-1-ylmethyl)-7-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
[5-({[(5,6-dimethyl-1H-1,3-benzodiazol-2-yl)methyl](methyl)amino}methyl)furan-2-yl]methanol
2-(pyridin-3-yl)-N-{[3-(pyrimidin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2-(pyrrolidin-1-yl)acetamide
2-{2-[7-(1-hydroxy-3-phenylpropyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}-2,3-dihydro-1H-isoindole-1,3-dione
4-({5-[4-(1H-pyrazol-1-yl)phenyl]-1H,4H-pyrazolo[3,4-d]imidazol-1-yl}methyl)pyridine
2-ethyl-4-methyl-5-(1-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1H-imidazol-2-yl)-1H-imidazole
5-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-1-(3-methylbutyl)-N-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
N-[(3R,7S,8aS)-3-benzyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-fluoro-4-methylbenzamide
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(pyrrolidine-1-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(1-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidin-3-yl)methanol
1-(4-ethylpiperazin-1-yl)-3-(3-{[(2-phenylethyl)amino]methyl}phenoxy)propan-2-ol
dimethyl[(4-methyl-5-{1-[(1-methyl-1H-indol-6-yl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methyl]amine
4-(2-ethylphenyl)-3-[(methylamino)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
6-(2-hydroxyethyl)-N-[(1-methylpiperidin-3-yl)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-(1,3-benzothiazol-2-ylmethyl)-N-methyl-1-phenyl-1H-1,2,3-triazole-4-carboxamide
ethyl 5-{[8-(2-hydroxyethyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]methyl}furan-2-carboxylate
7-[(3,4-difluorophenyl)methyl]-2-{[5-(hydroxymethyl)furan-2-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
N-[(3R,5S)-5-(ethylcarbamoyl)-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]-1,3-dimethyl-1H-pyrazole-4-carboxamide
6-[1-(4-ethylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-2-methyl-2,3-dihydropyridazin-3-one
3-[(2R,5R)-2,5-dimethylpyrrolidine-1-carbonyl]-5-(3-fluorophenoxymethyl)-1H-pyrazole
1-{[4-(furan-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperidin-4-ol
(1H-1,3-benzodiazol-2-ylmethyl)(ethyl)[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]amine
2-[4-(3-methoxypropyl)piperazin-1-yl]-4-(pyridin-3-yl)pyrimidine
3-{[1-(ethylcarbamoyl)ethyl]sulfamoyl}-N-(1-propylcyclopropyl)benzamide
2-[2-(methylsulfanyl)phenyl]pyridine-3-carboxamide
1-methyl-2,4-dioxo-N-{2-[5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-5-carboxamide
[(1-methylpiperidin-4-yl)methyl](2-phenylethyl)(quinolin-2-ylmethyl)amine
N-[(4-chlorophenyl)methyl]-3-{6-oxo-2,7-diazaspiro[4.5]decan-2-yl}propanamide
ethyl 4-(6-{2-[3-(trifluoromethyl)phenyl]acetyl}-6-azaspiro[2.5]octane-1-amido)piperidine-1-carboxylate
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
N-(3-chloro-4-methoxyphenyl)-3-[1-(5-methylthiophene-2-carbonyl)piperidin-3-yl]propanamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-1H-1,2,3-triazole-5-carboxamide
1-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]piperidin-4-amine
1-{[1-(2-methyl-6-propylpyrimidin-4-yl)piperidin-3-yl]methyl}pyrrolidin-2-one
(2-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridin-4-yl)methanol
N-cyclopropyl-1-[2-(4-methoxyphenyl)ethyl]-5-(2-methylpropanoyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(1-{2-[ethyl(methyl)amino]acetyl}piperidin-4-yl)-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
methyl (2S,4R)-1-[(2,5-dimethylphenyl)methyl]-4-(2-phenylquinoline-4-amido)pyrrolidine-2-carboxylate
methyl 3-[(3,3-dimethylbutanamido)methyl]-5-(quinoline-8-sulfonamido)benzoate
1-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
1-(2-chlorophenyl)-3-(1-{1-[1-(1-methylcyclopropyl)propan-2-yl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
2-{5-cyclopropyl-4-[4-(2-methoxyphenyl)piperazine-1-carbonyl]-1H-pyrazol-1-yl}-4-(2-fluorophenyl)pyrimidine
methyl 4-(5-{[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoate
3-[(2R,3R,6R)-5-(morpholine-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
5-methoxy-2-{[methyl({4-methyl-5-[(2-phenoxyethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)amino]methyl}phenol
4-({[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]amino}methyl)-1,2-dihydrophthalazin-1-one
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(1H-pyrazole-4-carbonyl)-2,7-diazaspiro[4.5]decane
5-(methanesulfonylmethyl)-2-(thiophen-3-yl)pyridine
2-(5-ethyl-1,3,4-thiadiazol-2-yl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one