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(3aS,6aR)-5-(1-benzofuran-2-ylmethyl)-3-[(2-methoxyphenyl)methyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-[2-hydroxy-2-(4-hydroxyphenyl)ethyl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
6-[3-(methylsulfanyl)phenyl]-3,4-dihydroquinazolin-4-one
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-1-(pyridin-2-yl)piperidine-3-carboxamide
N-[2-(3-methoxyphenyl)-1-[1-(quinoline-2-carbonyl)piperidin-4-yl]ethyl]-N-methylcyclopropanecarboxamide
2-{[3-(5-fluoro-2-methoxybenzoyl)piperidin-1-yl]methyl}-1-methyl-1H-1,3-benzodiazole
N-{[3-(pyrrolidin-1-yl)phenyl]methyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
N-(3,5-dimethoxyphenyl)-2-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]acetamide
7-(2-chloro-3-methylbenzoyl)-N,N,2-trimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-[2-methoxy-4-(1,4-oxazepan-4-ylmethyl)phenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
N-(2-ethylphenyl)-4-(furan-3-carbonyl)-1,4-diazepane-1-carboxamide
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-(2-methoxyethyl)-N-methylpiperidine-3-carboxamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-6-oxo-1,6-dihydropyrimidine-5-carboxamide
(3S,4S)-1-(1H-1,2,3-benzotriazole-5-carbonyl)-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
3-(hydroxymethyl)-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}piperidin-3-ol
2-ethoxy-5-{2-[(1-methoxypropan-2-yl)amino]pyrimidin-4-yl}benzoic acid
2-{2-[(4aR,8aR)-6-(3-methylbutyl)-decahydro-1,6-naphthyridin-1-yl]-2-oxoethyl}-4-benzyl-1,2-dihydrophthalazin-1-one
1-{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}-4-methylpiperidine
1-[(1S,5R)-3-benzoyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-[(trifluoromethyl)sulfanyl]ethan-1-one
N-(isoquinolin-5-ylmethyl)-N-methyl-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)benzamide
3-chloro-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]benzamide
N-({1-[(3,4-dimethylphenyl)methyl]piperidin-3-yl}methyl)pyrimidine-4-carboxamide
9-(cyclopropylmethyl)-4-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2,2-dimethyl-4-{4-[1-(3-methylphenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}morpholine
N-({6-[3-(trifluoromethyl)phenyl]pyridin-3-yl}methyl)acetamide
({6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[2,1-b][1,3]thiazol-5-yl}methyl)[(4-methoxyphenyl)methyl]amine
(3aR,7aS)-2-[6-(propan-2-yl)-2-(trifluoromethyl)pyrimidin-4-yl]-2,3,3a,4,7,7a-hexahydro-1H-isoindole
3-hydroxy-5-[3-(1H-pyrazol-1-yl)phenyl]benzoic acid
N-(2,3-dihydro-1H-inden-5-yl)-4-(pyridin-3-ylmethoxy)piperidine-1-carboxamide
ethyl 4-{4-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]benzoyl}piperazine-1-carboxylate
2-({4-[4-(oxolan-2-ylmethyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)phenol
1-[(4-fluorophenyl)methyl]-4-(1-methylcyclopropanecarbonyl)-2-(propan-2-yl)-1,4-diazepane
2-[5-(1-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carbonyl}piperidin-4-yl)-1H-pyrazol-3-yl]acetic acid
3-[1-(1-methyl-1H-pyrrole-2-carbonyl)piperidin-4-yl]-N-(oxolan-2-ylmethyl)propanamide
(1R,3S)-3-[2-(dimethylamino)ethoxy]-7-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-7-azaspiro[3.5]nonan-1-ol
2-{2-[3-(3-fluorophenoxymethyl)piperidin-1-yl]-2-oxoethyl}-1,2-dihydrophthalazin-1-one
N-{2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N,2,6-trimethylquinoline-4-carboxamide
1-{2-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-2-oxoethyl}-3-methoxy-1,2-dihydropyridin-2-one
1-(4-{1-[methyl(pyridin-4-ylmethyl)amino]-2-phenylethyl}piperidin-1-yl)-3-phenoxypropan-1-one
4-{2-oxo-2-[3-(thiophene-2-carbonyl)piperidin-1-yl]ethyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
2-ethyl-N-[(5-methoxy-1,3-benzoxazol-2-yl)methyl]pyrimidine-5-carboxamide
N-[(3S,4R)-1-{[2-(morpholin-4-yl)pyrimidin-5-yl]methyl}-4-propylpyrrolidin-3-yl]acetamide
1-[4-(1,3-benzoxazol-2-yl)piperidin-1-yl]-3-(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propan-1-one
3-(1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}piperidin-4-yl)-N-[(1-ethylpyrrolidin-2-yl)methyl]propanamide
{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}[(1,2-dimethyl-1H-imidazol-5-yl)methyl]amine
N-{[3-(methylsulfanyl)phenyl]methyl}-N-(propan-2-yl)-2-(pyrrolidin-3-yl)acetamide
2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetic acid
N,N-dimethyl-5-[(4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazin-1-yl)methyl]-1,3-thiazol-2-amine
2-(2-hydroxyethyl)-9-{[4-(propan-2-yloxy)phenyl]methyl}-2,9-diazaspiro[5.5]undecan-3-one