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1-{[1-(4-fluorophenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]methyl}-1H-1,2,3,4-tetrazole
4-{[(2R,5S)-5-(pyridin-4-ylmethyl)oxolan-2-yl]methyl}-1,4-oxazepane
N-{3-[benzyl(2-carbamoylethyl)carbamoyl]phenyl}pentanamide
3-[({[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)methyl]pyridin-2-amine
N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
3-(2,5-dimethoxyphenyl)-1-(2-ethoxybenzoyl)pyrrolidine
7-(cyclobutylmethyl)-2-[2-(1H-pyrazol-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
5-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-2-methyl-3,4-dihydropyrimidin-4-one
(3R,4S)-3,4-dimethyl-1-[1-(4-methylphenyl)cyclopropanecarbonyl]piperidin-4-ol
N-methyl-N-[2-(oxan-2-yl)ethyl]-5-propyl-1,2-oxazole-3-carboxamide
(5S,9aS,9bS)-2-[(2-methoxyphenyl)methyl]-5-phenyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-[(1S,3S,3aR,6aS)-3-(hydroxymethyl)-5-methyl-3-phenyl-octahydropyrrolo[3,4-c]pyrrol-1-yl]-2,6-dimethylphenol
2-{2-[3-(4-fluorophenoxy)piperidin-1-yl]-2-oxoethyl}-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
2-ethyl-9-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-6-ethyl-2-methylquinoline-4-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-4-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazine
(1R,3S)-7-(1H-indazole-3-carbonyl)-3-methoxy-3-methyl-7-azaspiro[3.5]nonan-1-ol
2-(2-hydroxyethyl)-9-(4-methylpyridine-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[1-(3,4-dimethoxybenzoyl)piperidin-4-yl]-2-(methoxymethyl)-5-(trifluoromethyl)-1H-1,3-benzodiazole
6-methyl-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
N-[4-(4-methoxyphenyl)butan-2-yl]-2,2,6,6-tetramethylpiperidin-4-amine
N-({5-[(3-fluoro-2,4-dimethylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methoxyacetamide
N-{[1-(2-fluorophenyl)pyrrolidin-3-yl]methyl}-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
[3-(hydroxymethyl)-1-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl]methanol
N-[(3,4-dimethoxyphenyl)methyl]-N-methyl-3-(5-methylfuran-2-yl)benzamide
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-methyl-3-(1H-pyrazol-1-yl)propan-1-one
N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-3-(3-fluorophenyl)-1H-pyrazole-4-carboxamide
1-[(3-fluorophenyl)methyl]-4-(2-methyl-1,3-thiazole-5-carbonyl)piperazine
1-methyl-5-(4-methylpyrimidin-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-cyclopentyl-6-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
4-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-N-methylpyridin-2-amine
4-{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}piperazine-1-carbaldehyde
N-methyl-N-[1-(1,3-thiazol-5-yl)ethyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
7-[(2,3-difluorophenyl)methyl]-2-[(2-methylpyrimidin-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
4-[1-(3-methyl-4,5-dihydro-1,2-oxazole-5-carbonyl)piperidin-4-yl]pyridine
2-[4-(2-propyl-1,3-thiazole-4-carbonyl)piperazin-1-yl]-1,3-benzoxazole
(3R)-1-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]pyrrolidin-3-ol
2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}acetamide
2-(adamantan-1-yl)-N-{3-[3-(hydroxymethyl)piperidin-1-yl]propyl}acetamide
1-{2-[5-(6-ethoxypyridin-3-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}piperidin-4-ol
1,9-dimethyl-4-[(4-methylthiophen-2-yl)sulfonyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
1-[1-(pent-2-yn-1-yl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
N-[(3,4-dimethoxyphenyl)methyl]-4-methyl-5-[1-(pyridin-4-ylmethyl)-1H-pyrazol-3-yl]-1,3-thiazol-2-amine
N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
2-{2-[methyl(quinolin-2-ylmethyl)amino]pyrimidin-4-yl}pyridine-4-carboxylic acid
N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]-1-(pyrrolidin-1-yl)cyclopentane-1-carboxamide
N-ethyl-3-[2-(hydroxymethyl)phenyl]benzamide
2-{[7-(5,8-dimethoxy-4-methylquinolin-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}phenol
5-fluoro-3-methyl-N-(prop-2-en-1-yl)-N-(pyridin-3-ylmethyl)-1H-indole-2-carboxamide
1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-methoxyethoxy)piperidine