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1-methyl-3-[3-(2-methylphenyl)phenyl]-1-[4-(morpholin-4-yl)butyl]urea
6-{[(2R)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}-N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
1-methyl-5-[4-(4-methylphenyl)piperazin-1-yl]-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
2-methyl-5-{4-[2-(2-methyl-5-oxopyrrolidin-1-yl)acetyl]piperazin-1-yl}-2,3-dihydropyridazin-3-one
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-5-methoxy-N-methyl-1H-indole-2-carboxamide
2-[({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)amino]pyridine-3-carboxamide
(4aR,7aS)-1-ethyl-4-[2-(2-methoxyethoxy)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(4-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}-1,4-diazepan-1-yl)ethan-1-one
1-[(4aR,8aS)-1-(5-chloro-2-fluorobenzoyl)-decahydro-1,6-naphthyridin-6-yl]ethan-1-one
8-(5-amino-1H-pyrazole-3-carbonyl)-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-[2-(2,6-difluorophenyl)ethyl]-1-methanesulfonylpiperidine
1-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidine-1-carbonyl]cyclopropane-1-carboxamide
4-[hydroxy(pyridin-2-yl)methyl]-N-(5,6,7,8-tetrahydronaphthalen-1-yl)piperidine-1-carboxamide
4-cyclopentyl-3-{[3-(1-methyl-1H-imidazol-4-yl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-2-one
5-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-methyl-2-(4H-1,2,4-triazol-4-yl)pyridine
1-benzyl-4-(8-methoxyquinolin-2-yl)-1,4-diazepan-6-ol
1-[1-(hydroxymethyl)-9-[(3-hydroxyphenyl)methyl]-3,9-diazaspiro[5.5]undecan-3-yl]-2-(methylsulfanyl)ethan-1-one
2-[(1S,5R)-3-[2-(2-hydroxyphenyl)acetyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
3-[1-(1-tert-butyl-1H-pyrrole-3-carbonyl)piperidin-3-yl]benzoic acid
3-[3-(2H-1,3-benzodioxol-5-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,5-dimethyl-1H-pyrazole
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-methoxyacetamide
8-[(2S)-3-hydroxy-2-(methylamino)propanoyl]-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-(2-ethoxyphenyl)-2-[2-(morpholin-4-yl)ethyl]piperidine-1-carboxamide
4-[3-fluoro-5-(trifluoromethyl)phenyl]-6-(4-methylpiperazin-1-yl)pyrimidin-2-amine
8-[2-(methylsulfanyl)benzoyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(oxan-4-ylmethyl)-3-(thiomorpholine-4-sulfonyl)benzamide
4-({1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}oxy)-N-(pyridin-2-ylmethyl)benzamide
(1R,7S)-3-[(4-fluorophenyl)methyl]-N-methyl-N-(1,2-oxazol-3-ylmethyl)-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
3-methyl-5-(2-{3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidin-1-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(pyridin-4-yl)-N-{[3-(trifluoromethyl)phenyl]methyl}pyrimidine-5-carboxamide
4-(3,4-diethoxybenzoyl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
2-{[3-(naphthalene-1-carbonyl)piperidin-1-yl]methyl}-1H-1,3-benzodiazole
2-(adamantan-1-yl)-N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}acetamide
3-(4-{[2-(carbamoylmethyl)piperidin-1-yl]methyl}-1H-pyrazol-1-yl)propanoic acid
(5S,9aS,9bS)-2-[(3-methoxyphenyl)methyl]-5-[5-(propan-2-yl)-1H-pyrazol-3-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N3-[2-(dimethylamino)ethyl]-N3-(thiophen-3-ylmethyl)piperidine-1,3-dicarboxamide
(1S,5R)-6-benzyl-3-[(4-fluoro-3-methylphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
[(3S,5R)-1-[(5-chlorothiophen-2-yl)methyl]-5-[(dimethylamino)methyl]piperidin-3-yl]methanol
4-benzyl-3-ethyl-1-[2-oxo-2-(piperidin-1-yl)ethyl]-1,4-diazepan-5-one
2-(dimethylamino)-2-(4-fluorophenyl)-N-{[(propan-2-yl)carbamoyl]methyl}acetamide
1-[4-(2,3-dihydro-1H-isoindol-2-yl)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
4-[2-(propan-2-yl)-1,3-benzoxazol-5-yl]isoquinoline
4-(2-hydroxyethyl)-N-[2-(2-methoxyphenoxy)phenyl]piperazine-1-carboxamide
2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-4-methyl-3,4-dihydro-2H-1,4-benzoxazine
2-(2-methoxyethyl)-5-{[2-methyl-4-(4-methylphenyl)piperazin-1-yl]methyl}pyrimidine
6-methyl-N-{[5-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}imidazo[2,1-b][1,3]thiazole-5-carboxamide
5-[butyl(methyl)amino]-1-ethyl-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
ethyl 3-[(2,4-difluorophenyl)methyl]-1-(1,5-dimethyl-1H-pyrazole-3-carbonyl)piperidine-3-carboxylate
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-2-(pyridin-4-yl)quinoline-4-carboxamide
3-[1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)piperidin-2-yl]pyridine