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5-methyl-N-[1-(3-methylpyridin-2-yl)propan-2-yl]-3-phenyl-1,2-oxazole-4-carboxamide
5-methyl-2-(methylamino)-N-{[1-(pyridin-2-ylmethyl)pyrrolidin-3-yl]methyl}benzamide
2-{6-chloro-2-methylimidazo[1,2-a]pyridine-3-carbonyl}-7-methyl-2,7-diazaspiro[4.5]decan-6-one
(4aS,8aR)-6-(4-methoxycyclohexanecarbonyl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
2-cyclopropyl-9-(3-methoxy-2-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
3-hydroxy-3-{[(2-methylpropyl)amino]methyl}-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
3-[(2-fluorophenyl)formamido]-N-methyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
3-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]-3H,4H-pyrido[3,4-d]pyrimidin-4-one
N-(5-hydroxyadamantan-2-yl)-5-methyl-4-{[3-(morpholin-4-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
1-(furan-2-carbonyl)-N-[1-methyl-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidin-3-amine
N6-cyclopropyl-N4-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N4-methylpyrimidine-2,4,6-triamine
3-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-N-(furan-2-ylmethyl)-N-(1-hydroxybutan-2-yl)propanamide
(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-8-[(4-methyl-1H-imidazol-5-yl)methyl]-8-azabicyclo[3.2.1]octane
1-(3-{[3-(2-hydroxyethyl)-4-methylpiperazin-1-yl]methyl}phenyl)ethan-1-one
4-methoxy-3-{7-methyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl}benzene-1-sulfonamide
4-[2-(2-chloro-4-fluorophenyl)acetyl]-1-[(3-fluorophenyl)methyl]piperazin-2-one
(3S,4R)-1-(3-methyl-4-oxo-3,4-dihydroquinazoline-7-carbonyl)-4-phenylpyrrolidine-3-carboxylic acid
(3S,4R)-1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-4-phenylpyrrolidine-3-carboxylic acid
3-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]-1-methyl-1,2-dihydroquinolin-2-one
N-(3-{2-oxo-2-[2-(propan-2-yl)-2,5-dihydro-1H-pyrrol-1-yl]ethoxy}phenyl)propanamide
(2S,4S)-N-ethyl-4-{[(9-ethyl-9H-carbazol-3-yl)methyl]amino}-1-(propan-2-yl)pyrrolidine-2-carboxamide
1-[(4aR,8aS)-1-(cyclohex-1-ene-1-carbonyl)-decahydro-1,6-naphthyridin-6-yl]-3-phenoxypropan-1-one
7-cyclopropanecarbonyl-N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
5-methyl-1-(2-phenylphenyl)-4-(1,3-thiazole-4-carbonyl)piperazin-2-one
4-methoxy-2-[(3-{[4-(pyrrolidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)methyl]phenol
2-(furan-2-yl)-N,7-dimethyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-(3-hydroxy-3-methylbutyl)-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]benzamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-4H,5H,6H,7H,8H-cyclohepta[b]thiophene-2-carboxamide
1-[(3,5-dimethylphenyl)methyl]-4-[2-(4-fluorophenyl)-2-hydroxyacetyl]piperazin-2-one
1-[1-(2-ethylbutanoyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
1-(oxan-4-yl)-N-[2-(pyridin-2-yl)ethyl]piperidine-4-carboxamide
6-[(3-ethyl-1,2-oxazol-5-yl)methyl]-5,6-dihydro-1,6-naphthyridin-5-one
6-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-5,6,7,8-tetrahydro-1,6-naphthyridine
N3-cyclooctyl-4-oxo-1-(oxolan-2-ylmethyl)-N5-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
3-[(5-chloro-1,2,3,4-tetrahydroisoquinolin-2-yl)methyl]pyridin-2-amine
N,N-dimethyl-3-[3-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]aniline
1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-4-(3-methylpyridin-4-yl)-1,4-diazepane
N-[1-(1H-indol-1-yl)propan-2-yl]-4-(4H-1,2,4-triazol-4-yl)benzamide
9-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-3-oxa-9-azaspiro[5.5]undecane
(2S,4S)-4-amino-N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-1-methylpyrrolidine-2-carboxamide
1-[(5-methylfuran-2-yl)methyl]-N-[4-(1H-pyrazol-5-yl)phenyl]piperidine-3-carboxamide
(1S)-1-[1-(3,4-dimethylphenyl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]ethan-1-ol
1-{1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carbonyl}azonane
4-{[5-(1-ethyl-1H-pyrazol-3-yl)-1-(3-fluorophenyl)-1H-1,2,4-triazol-3-yl]methyl}-1-methylpiperidine
1-({5-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
2-(2-oxo-2-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}ethyl)-1,2-dihydrophthalazin-1-one
(1S,4S)-2-(5-chloro-2-methoxyphenyl)-5-[2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)acetyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]-2-(pyridin-2-ylsulfanyl)propanamide
7-fluoro-3-methyl-2-[4-(pyridin-3-ylmethyl)-1,4-diazepane-1-carbonyl]-1H-indole
2-acetyl-8-(3-methoxy-2-methylbenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid