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2-amino-4-(2-methoxypyrimidin-5-yl)-5-methyl-6-(5-methylfuran-2-yl)pyridine-3-carbonitrile
3,5-dimethyl-1-(1-{2-methyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl}pyrrolidin-3-yl)-1H-pyrazole
4-[(3aR,5R,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindole-2-carbonyl]-6-fluoro-1,2-dihydroquinolin-2-one
(1S,4S)-2-{5-[(4-ethylpiperazin-1-yl)methyl]-1,2-oxazole-3-carbonyl}-2-azabicyclo[2.2.1]heptane
N-[(1-methanesulfonylpiperidin-3-yl)methyl]-1-methyl-2-oxo-1,2-dihydroquinoline-3-carboxamide
4-{3-[3-(hydroxymethyl)-3-(prop-2-en-1-yl)piperidin-1-yl]propoxy}benzamide
1-(4-cyanopyridin-2-yl)-N-[4-(3-fluorophenyl)phenyl]piperidine-3-carboxamide
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-3-carboxamide
2-{4-[4-(furan-2-carbonyl)piperazine-1-carbonyl]piperidin-1-yl}-4-methyl-6-(propan-2-yl)quinazoline
3-{[3-(naphthalene-1-carbonyl)piperidin-1-yl]methyl}pyridine
2,3-dimethyl-5-[3-(2-methylpropyl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]benzene-1-sulfonamide
5-{2-[3-(3-fluorophenoxymethyl)piperidin-1-yl]-2-oxoethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-(pyrazin-2-yl)-2-{[2-(4-sulfamoylphenyl)ethyl]amino}acetamide
N-{[5-(2-amino-3-cyano-5,6,7,8-tetrahydroquinolin-4-yl)furan-2-yl]methyl}-N-methylmethanesulfonamide
4-methyl-2-{[5-(2-methylprop-1-en-1-yl)-4-phenyl-1H-imidazol-1-yl]methyl}-6-(trifluoromethyl)pyrimidine
N-{[7-chloro-5-(thiophen-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2,3,4-trimethoxybenzamide
N-[(2R,3R)-2-methoxy-1'-[2-(thiophen-2-yl)acetyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenoxyacetamide
N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-2-[(1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonan-3-yl]acetamide
(4aR,7aS)-1-acetyl-4-(2-methoxypyridine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{1'-[2-(4-hydroxyphenyl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
3-cyclopropyl-N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-1H-pyrazole-5-carboxamide
N-(furan-2-ylmethyl)-N-(3-methylbutan-2-yl)-2-(oxan-4-yl)acetamide
{[3-(2H-1,3-benzodioxol-5-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]methylamine
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-1-ethyl-1H-pyrazole-4-carboxamide
3-(4-{[3-(1H-indol-2-yl)phenyl]carbamoyl}piperidin-1-yl)propanoic acid
N-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]-3-(1H-pyrazol-1-yl)benzamide
1-[3-({3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}methyl)phenyl]ethan-1-one
4-{5-[2-(dimethylamino)-1,3-thiazol-5-yl]-4-phenyl-1H-imidazol-1-yl}butan-2-ol
N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-3-(1-methylpiperidin-2-yl)propanamide
(2S,4R)-4-amino-1-[3-chloro-4-(pyrrolidin-1-yl)benzoyl]-N-ethylpyrrolidine-2-carboxamide
5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-{imidazo[1,2-a]pyridin-3-ylmethyl}-1H-pyrazole-3-carboxamide
2-[(2-ethyl-1,3-thiazol-4-yl)methyl]-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
2-{[2-(1-{imidazo[1,2-a]pyrimidine-2-carbonyl}piperidin-4-yl)-1H-imidazol-1-yl]methyl}pyridine
1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazine
N-[(dimethyl-1,3-thiazol-2-yl)methyl]-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}[2-(pyrrolidin-1-yl)ethyl]amine
3-cyclohexyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1H-pyrazole-4-carboxamide
N-({7-[2-(trifluoromethyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)cyclopropanecarboxamide
2-[4-({4-[1-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}methyl)phenyl]ethan-1-amine
2-(4-methoxyphenyl)-5-[(2E)-2-methylbut-2-en-1-yl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
7-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-oxa-7-azaspiro[4.5]decan-8-one
2-[5-(2,3-dihydro-1H-inden-5-yl)-3-methyl-1H-1,2,4-triazol-1-yl]acetic acid
2-butyl-5-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]-1,3-benzoxazole
3-(azocane-1-carbonyl)-4-fluorobenzene-1-sulfonamide
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
7-methoxy-3-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carbonyl}-2,3,4,5-tetrahydro-1H-3-benzazepine
3-(2-ethylpiperidine-1-carbonyl)-N-(1,2-oxazol-3-ylmethyl)benzene-1-sulfonamide
N-methyl-N-(2-phenylethyl)-1-(thian-4-yl)piperidin-3-amine
5-oxo-1-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]pyrrolidine-3-carboxylic acid
2-[2-(2-butyl-4-methyl-3-oxopiperazin-1-yl)-2-oxoethyl]-5,6-dimethyl-2,3-dihydropyridazin-3-one